CAS 2166387-65-9

Formula: C24H29ClN6O3

InChI: InChI=1S/C24H29ClN6O3/c1-14-7-15(2)12-31(11-14)24-27-10-18(25)22(29-24)28-17-5-6-19-16(8-17)9-20(23(33)30(19)4)34-13-21(32)26-3/h5-6,8-10,14-15H,7,11-13H2,1-4H3,(H,26,32)(H,27,28,29)/t14-,15+

InChI key: GXTJETQFYHZHNB-GASCZTMLSA-N

SMILES: C[C@@H]1C[C@@H](CN(C1)C2=NC=C(C(=N2)NC3=CC4=C(C=C3)N(C(=O)C(=C4)OCC(=O)NC)C)Cl)C

BI-3802

CAS: 2166387-65-9

BI-3802

Formula: C₂₄H₂₉ClN₆O₃

Purity: ≥95%

Molecular weight: 484.98

Ref: 54-BUP04733

cis-2-((6-((5-chloro-2-(3,5-dimethylpiperidin-1-yl)pyrimidin-4-yl)amino)-1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)oxy)-N-methylacetamide

CAS: 2166387-65-9

Formula: C₂₄H₂₉ClN₆O₃

Purity: 98%

Color and Shape: Solid

Molecular weight: 484.9785

Ref: IN-DA01FNV7

BI-3802

CAS: 2166387-65-9

cis-2-((6-((5-chloro-2-(3,5-dimethylpiperidin-1-yl)pyrimidin-4-yl)amino)-1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)oxy)-N-methylacetamide

Formula: C₂₄H₂₉ClN₆O₃

Purity: 98%

Molecular weight: 484.98

Ref: IN-DG00794058

BI-3802

CAS: 2166387-65-9

BI-3802, a highly potent BCL6 degrader, targets and inhibits the Bric-à-brac (BTB) domain of BCL6, exhibiting an IC50 value of ≤3 nM.

Formula: C₂₄H₂₉ClN₆O₃

Purity: 97.93% - 99.48%

Color and Shape: Solid

Molecular weight: 484.978

Ref: TM-T5408

BI-3802

CAS: 2166387-65-9

BI-3802 is a small-molecule drug that is designed to target ubiquitin ligases. These enzymes are involved in the regulation of protein homeostasis, including the control of cell growth and proliferation. BI-3802 has been shown to regulate cellular growth by inhibiting the ubiquitin ligase activity of GPR55 and other related proteins. This inhibition leads to a reduction in lipid peroxide levels, which may be due to its ability to inhibit the production of reactive oxygen species.

Formula: C₂₄H₂₉ClN₆O₃

Purity: Min. 95%

Molecular weight: 485 g/mol

Ref: 3D-RLD38765