CAS 2225868-19-7

123B9

Formula: C₅₈H₈₂ClFN₁₂O₂₀

Synonyms:

• 123B9

123B9

CAS: 2225868-19-7

123B9 is a tumor-homing agent characterized as a potent and selective agonist for EphA2 with a dissociation constant (Kd) of 4.0 μM. It specifically targets the ligand-binding domain of the EphA2 tyrosine kinase receptor. Notably, 123B9 does not significantly inhibit the ligand-binding domains of closely related receptors EphA3 and EphA4.

Formula: C₅₈H₈₂ClFN₁₂O₂₀

Molecular weight: 1321.79

Ref: TM-TP2771