CAS 2226517-76-4

Formula: C18H17BrN2O3

InChI: InChI=1S/C18H17BrN2O3/c1-22-16-9-12(10-17(23-2)18(16)24-3)21-15-6-7-20-14-5-4-11(19)8-13(14)15/h4-10H,1-3H3,(H,20,21)

InChI key: AUOSKLDNVNGKRR-UHFFFAOYSA-N

SMILES: COC1=CC(=CC(=C1OC)OC)NC2=C3C=C(C=CC3=NC=C2)Br

SGC-GAK-1

CAS: 2226517-76-4

SGC-GAK-1

Formula: C₁₈H₁₇BrN₂O₃

Purity: ≥98%

Molecular weight: 389.24

Ref: 54-BUP10395

SGC-GAK-1

CAS: 2226517-76-4

SGC-GAK-1

Formula: C₁₈H₁₇BrN₂O₃

Purity: 98%

Molecular weight: 389.24318

Ref: 54-BISN0080

SGC GAK 1

CAS: 2226517-76-4

Formula: C₁₈H₁₇BrN₂O₃

Purity: 98%

Color and Shape: Solid

Molecular weight: 389.2432

Ref: IN-DA01ENHE

SGC-GAK-1

CAS: 2226517-76-4

6-Bromo-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine

Formula: C₁₈H₁₇BrN₂O₃

Purity: 98%

Molecular weight: 389.24

Ref: IN-DG01111372

SGC-GAK-1

CAS: 2226517-76-4

SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).

Formula: C₁₈H₁₇BrN₂O₃

Purity: 99.85%

Color and Shape: Yellow Solid

Molecular weight: 389.243

Ref: TM-T5169

SGC GAK 1

CAS: 2226517-76-4

A potent and selective inhibitor of cyclin G-associated kinase (GAK) with Ki of 3.1 nM. The compound has more than 50-fold selectivity over the closest off-target kinase RIPK2, making it a potent tool for the study of GAK biology. SGC-GAK-1 was tested in vitro in human prostate carcinoma cell lines and showed strong growth inhibition in cell lines with androgen-dependent growth.

Formula: C₁₈H₁₇BrN₂O₃

Purity: Min. 95%

Color and Shape: Solid

Molecular weight: 388.04226

Ref: 3D-FB166265

SGC-GAK-1

CAS: 2226517-76-4

Purity: 98%

Molecular weight: 388.042

Ref: 10-F864210