CAS 30392-41-7

Bitolterol mesylate

Description:

Bitolterol mesylate is a synthetic compound primarily used as a bronchodilator in the treatment of asthma and chronic obstructive pulmonary disease (COPD). It functions as a beta-adrenergic agonist, specifically targeting beta-2 adrenergic receptors in the bronchial smooth muscle, leading to relaxation and dilation of the airways. This compound is characterized by its ability to provide rapid relief from bronchospasm, making it effective in managing respiratory conditions. Bitolterol mesylate is typically administered via inhalation, allowing for direct delivery to the lungs, which enhances its therapeutic effects while minimizing systemic side effects. The mesylate salt form improves its solubility and stability, facilitating its formulation in aerosolized delivery systems. Additionally, it is important to note that while Bitolterol mesylate is effective, it may also have side effects, including increased heart rate and nervousness, which are common with beta-agonists. Overall, Bitolterol mesylate represents a valuable option in respiratory therapy, particularly for patients requiring bronchodilation.

Formula: C₂₈H₃₁NO₅·CH₄O₃S

InChI: InChI=1S/C28H31NO5.CH4O3S/c1-18-6-10-20(11-7-18)26(31)33-24-15-14-22(23(30)17-29-28(3,4)5)16-25(24)34-27(32)21-12-8-19(2)9-13-21;1-5(2,3)4/h6-16,23,29-30H,17H2,1-5H3;1H3,(H,2,3,4)

InChI key: InChIKey=HODFCFXCOMKRCG-UHFFFAOYSA-N

SMILES: O(C(=O)C1=CC=C(C)C=C1)C2=C(OC(=O)C3=CC=C(C)C=C3)C=CC(C(CNC(C)(C)C)O)=C2.S(C)(=O)(=O)O

Synonyms:

• (tert-Butyl)[β-hydroxy-3,4-bis(p-toluoyloxy)phenethyl]ammonium methanesulfonate
• 4-[2-(Tert-Butylamino)-1-Hydroxyethyl]Benzene-1,2-Diyl Bis(4-Methylbenzoate) Methanesulfonate (1:1)
• Benzoic acid, 4-methyl-, 1,1′-[4-[2-[(1,1-dimethylethyl)amino]-1-hydroxyethyl]-1,2-phenylene] ester, methanesulfonate (1:1)
• Benzoic acid, 4-methyl-, 4-[2-[(1,1-dimethylethyl)amino]-1-hydroxyethyl]-1,2-phenylene ester, methanesulfonate (salt)
• Biterol
• Bitolterol Mesylate
• Bitoterol methanesulfonate
• Effectin
• Tornalate
• Win 32784
• p-Toluic acid, 4-[2-(tert-butylamino)-1-hydroxyethyl]-o-phenylene ester methanesulfonate (salt)

Bitolterol Mesylate

CAS: 30392-41-7

Applications Bitolterol Mesylate is a β2-adrenergic receptor agonist used for the relief of bronchospasm in conditions such as asthma and COPD.
References Friedel, H., et al.: Drugs., 35, 22 (1988); Cronin, M.T.D., et al.: J. Chem. Info. Comp. Sci., 42, 869 (2002); Shargel, L., et al.: Drug. Meta. Disp., 4, 72 (1976);

Formula: C₂₉H₃₅NO₈S

Color and Shape: Off-White To Light Beige

Molecular weight: 557.66

Ref: TR-B591400

Bitolterol mesylate

CAS: 30392-41-7

Bitolterol mesylate is a bronchodilator that belongs to the group of pharmacological agents. It is a beta-2 adrenergic receptor agonist and a potent bronchodilator with a rapid onset of action. Bitolterol mesylate acts by binding to beta-2 adrenergic receptors in the lungs, which causes relaxation of the smooth muscle in the airways and an increase in airflow to the lungs. This drug can be used for treating asthma, chronic obstructive pulmonary disease, and other conditions involving lung inflammation. Side effects may include chest pain, heart palpitations, headache, dizziness, or nausea. Bitolterol mesylate has also been shown to have antimicrobial activity against bacteria that cause inflammatory bowel disease.

Formula: C₂₉H₃₅NO₈S

Purity: Min. 95%

Color and Shape: Off-White Powder

Molecular weight: 557.66 g/mol

Ref: 3D-FB156857

Bitolterol mesylate

CAS: 30392-41-7

Bitolterol mesylate is a Bronchodilator.

Formula: C₂₉H₃₅NO₈S

Purity: 98%

Color and Shape: Solid

Molecular weight: 557.66

Ref: TM-T25161

Bitolterol Mesylate

CAS: 30392-41-7

Formula: C₂₈H₃₁NO₅

Molecular weight: 461.56

Ref: ST-EA-CP-B548003