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CAS 3052947-04-0

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Formula:C25H22N4O4S
InChI:InChI=1S/C25H22N4O4S/c30-21-9-8-20(23(32)27-21)29-14-17-7-6-16(11-19(17)24(29)33)12-22(31)28-25-26-13-18(34-25)10-15-4-2-1-3-5-15/h1-7,11,13,20H,8-10,12,14H2,(H,26,28,31)(H,27,30,32)
InChI key:IDDUCAFDQHUAFX-UHFFFAOYSA-N
SMILES:C1CC(=O)NC(=O)C1N2CC3=C(C2=O)C=C(C=C3)CC(=O)NC4=NC=C(S4)CC5=CC=CC=C5
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    GRK2 degrader-1

    CAS:
    GRK2 degrader-1 (compound 1) is a potent and orally active GRK2 degrader. It facilitates the degradation of GRK2 via the ubiquitin-proteasome pathway. In a pulmonary arterial hypertension (PAH) mouse model, GRK2 degrader-1 inhibits right ventricular remodeling and the increase in pulmonary arterial pressure. This compound is suitable for research in pulmonary arterial hypertension (PAH).
    Formula:C25H22N4O4S
    Molecular weight:474.54

    Ref: TM-TYD-05426

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