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CAS 496849-46-8

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H-Tyr-Cyclo(-D-Dab-Arg-Phe-Phe-D-Trp-Lys-Thr-Phe)

Description:
The chemical substance H-Tyr-Cyclo(-D-Dab-Arg-Phe-Phe-D-Trp-Lys-Thr-Phe) is a cyclic peptide, characterized by its unique sequence of amino acids and a cyclization that enhances its stability and bioactivity. The presence of both D- and L-amino acids in its structure contributes to its resistance to enzymatic degradation, making it a candidate for therapeutic applications. The sequence includes aromatic residues, such as phenylalanine and tryptophan, which can facilitate interactions with biological targets, potentially enhancing its affinity and specificity. The cyclic nature of the peptide often results in a conformational rigidity that can be advantageous for receptor binding. Additionally, the presence of various functional groups, such as the hydroxyl group from tyrosine and the amine group from lysine, may influence its solubility and interaction with other biomolecules. Overall, this compound's structural features suggest potential utility in drug design, particularly in the development of peptide-based therapeutics targeting specific biological pathways.
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Found 2 products.
  • Tyr-(D-Dab 4,Arg5,D-Trp8)-cyclo-Somatostatin-14 (4-11) trifluoroacetate salt
    Biosynth
    + Info

    Tyr-(D-Dab 4,Arg5,D-Trp8)-cyclo-Somatostatin-14 (4-11) trifluoroacetate salt

    CAS:
    <p>Please enquire for more information about Tyr-(D-Dab 4,Arg5,D-Trp8)-cyclo-Somatostatin-14 (4-11) trifluoroacetate salt including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>
    Formula:C67H85N15O11
    Purity:Min. 95%
    Molecular weight:1,276.49 g/mol

    Ref: 3D-FT109780

    1mg
    860.00€
    2mg
    1,042.00€
    5mg
    2,078.00€
  • Tyr-(D-Dab⁴,Arg⁵,D-Trp⁸)-cyclo-Somatostatin-14 (4-11)
    Bachem
    + Info

    Tyr-(D-Dab⁴,Arg⁵,D-Trp⁸)-cyclo-Somatostatin-14 (4-11)

    CAS:
    <p>High affinity ligand for all five somatostatin receptors (sst1-sst5). In AtT-20 mouse anterior pituitary tumor cells which mainly express sst2 and sst5 receptors the binding affinity of this somatostatin analog was found to be higher than that of somatostatin-14 and octreotide. In a model of epileptogenesis, however, KE 108 did not exhibit antiepileptic activity suggesting that the high potency and efficacy of a synthetic ligand to all known somatostatin receptors may not reproduce entirely the effects of the natural ligand.</p>
    Formula:C67H85N15O11
    Purity:98.6%
    Color and Shape:White Powder
    Molecular weight:1276.51

    Ref: 01-4041674

    1mg
    Discontinued
    5mg
    Discontinued
    Discontinued product