CAS 5638-76-6: Betahistine (base and/or unspecified salts)
Description:Betahistine, with the CAS number 5638-76-6, is a histamine analog primarily used in the treatment of vestibular disorders, such as Ménière's disease. It functions as a vasodilator, improving blood flow to the inner ear, which can help alleviate symptoms like vertigo and tinnitus. Betahistine acts as a selective agonist for the H1 receptor and an antagonist for the H3 receptor, influencing neurotransmitter release and promoting vestibular compensation. The substance is typically administered in its dihydrochloride salt form, which enhances its solubility and bioavailability. Betahistine is generally well-tolerated, with common side effects including gastrointestinal disturbances and headaches. Its pharmacokinetics indicate rapid absorption and a relatively short half-life, necessitating multiple daily doses for effective symptom management. Overall, Betahistine is recognized for its therapeutic role in improving balance and reducing dizziness associated with inner ear disorders.
Formula:C8H12N2
InChI:InChI=1S/C8H12N2/c1-9-7-5-8-4-2-3-6-10-8/h2-4,6,9H,5,7H2,1H3
InChI key:InChIKey=UUQMNUMQCIQDMZ-UHFFFAOYSA-N
SMILES:N=1C=CC=CC1CCNC
- Synonyms:
- (2-(2-Pyridyl)ethyl)methylamine
- 2-(2-(Methylamino)ethyl)pyridine
- 2-(2-Methylaminoethyl)Pyridine
- 2-(β-Methylaminoethyl)pyridine
- 2-Pyridineethanamine, N-methyl-
- Betahistina
- Betahistina [INN-Spanish]
- Betahistine
- Betahistine [INN:BAN]
- Betahistinum
- See more synonyms
- Betahistinum [INN-Latin]
- Betaistina
- Betaistina [DCIT]
- Brn 0112294
- Methyl(2-pyridin-2-ylethyl)amine
- N-Methyl-2-(2-pyridinyl)ethanamine
- N-Methyl-2-(2-pyridyl)ethylamine
- N-Methyl-2-pyridineethanamine
- N-Methyl-2-pyridineethylamine
- N-Methyl-N-[2-(2-pyridinyl)ethyl]amine
- N-Methyl-N-[2-(pyridin-2-yl)ethyl]amine
- N-Methyl-N-beta-(2-pyridyl)ethylamine
- N-Methyl[2-(pyridin-2-yl)ethyl]amine
- N-[2-(2-Pyridyl)ethyl]-N-methylamine
- Nsc 42617
- Obe 101
- PT 9 base
- Pyridine, 2-(2-(methylamino)ethyl)-
- Pyridine, 2-(2-methylaminoethyl)-
- Serc base
- Sinmenier (free base)
- Unii-X32Kk4201D
- Vasomotal
- Y-G 14
- beta-Histine
- β-Histine

Betahistine Methanesulfonate
Ref: 3B-B1424
25g | 77.00 € |

N-Methyl-2-(pyridin-2-yl)ethanamine
Ref: IN-DA003T69
1g | 51.00 € | ||
5g | 133.00 € | ||
25g | 265.00 € | ||
100g | To inquire | ||
100mg | 30.00 € | ||
250mg | 27.00 € |

Betahistine-13C-d3 DiHCl
Ref: 4Z-B-364
5mg | To inquire | ||
10mg | To inquire | ||
25mg | To inquire | ||
50mg | To inquire | ||
100mg | To inquire |

2-[2-(Methylamino)ethyl]pyridine
Ref: 54-OR22222
1g | 51.00 € | ||
5g | 107.00 € | ||
250mg | 38.00 € |

Betahistine
Ref: 3B-B6621
5g | 82.00 € | ||
25g | 296.00 € |

Betahistine
Ref: TM-T4195
100mg | 35.00 € | ||
1mL*10mM (DMSO) | 35.00 € |

N-Methyl-N-(2-pyridin-2-ylethyl)amine
Ref: 10-F065480
1g | 40.00 € | ||
5g | To inquire | ||
25g | To inquire |

Betahistine
Controlled ProductRef: TR-B324005
500mg | 178.00 € |

2-(2-Methylaminoethyl)Pyridine
Ref: 3D-FM52866
1g | Discontinued | Request information | |
2g | Discontinued | Request information | |
5g | Discontinued | Request information | |
10g | Discontinued | Request information | |
25g | Discontinued | Request information |