CAS 61197-73-7
:Loprazolam
Description:
Loprazolam is a benzodiazepine derivative primarily used for its anxiolytic and hypnotic properties. It is characterized by its ability to enhance the effects of the neurotransmitter gamma-aminobutyric acid (GABA) at the GABA-A receptor, leading to sedative, anxiolytic, muscle relaxant, and anticonvulsant effects. Loprazolam is typically administered in tablet form and is known for its relatively rapid onset of action and moderate duration of effects. The substance is often prescribed for the short-term management of insomnia and anxiety disorders. Its pharmacokinetics indicate that it is metabolized in the liver, with metabolites that may also exhibit pharmacological activity. Common side effects can include drowsiness, dizziness, and potential dependence with prolonged use. Due to its sedative properties, caution is advised when operating machinery or driving after consumption. As with other benzodiazepines, it is important to use Loprazolam under medical supervision to mitigate risks of tolerance and withdrawal symptoms.
Formula:C23H21ClN6O3
InChI:InChI=1S/C23H21ClN6O3/c1-27-8-10-28(11-9-27)14-19-23(31)29-20-7-6-15(30(32)33)12-17(20)22(25-13-21(29)26-19)16-4-2-3-5-18(16)24/h2-7,12,14H,8-11,13H2,1H3/b19-14-
InChI key:InChIKey=UTEFBSAVJNEPTR-RGEXLXHISA-N
SMILES:O=C\1N2C=3C(C(=NCC2=N/C1=C\N4CCN(C)CC4)C5=C(Cl)C=CC=C5)=CC(N(=O)=O)=CC3
Synonyms:- (2Z)-6-(2-Chlorophenyl)-2,4-dihydro-2-[(4-methyl-1-piperazinyl)methylene]-8-nitro-1H-imidazo[1,2-a][1,4]benzodiazepin-1-one
- (2Z)-6-(2-chlorophenyl)-2-[(4-methylpiperazin-1-yl)methylidene]-8-nitro-2,4-dihydro-1H-imidazo[1,2-a][1,4]benzodiazepin-1-one
- (Z)-6-(o-Chlorophenyl)-2,4-dihydro-2-((4-methyl-1-piperazinyl)methylene)-8-nitro-1H-imidazo(1,2-a)(1,4)benzodiazepin-1-one
- 1H-Imidazo(1,2-a)(1,4)benzodiazepin-1-one, 2,4-dihydro-6-(2-chlorophenyl)-2-((4-methyl-1-piperazinyl)methylene)-8-nitro-
- 1H-Imidazo[1,2-a][1,4]benzodiazepin-1-one, 6-(2-chlorophenyl)-2,4-dihydro-2-[(4-methyl-1-piperazinyl)methylene]-8-nitro-, (2Z)-
- 1H-Imidazo[1,2-a][1,4]benzodiazepin-1-one, 6-(2-chlorophenyl)-2,4-dihydro-2-[(4-methyl-1-piperazinyl)methylene]-8-nitro-, (Z)-
- 6-(2-Chlorophenyl)-2,4-dihydro-2-((4-methyl-1-piperazinyl)methylene)-8-nitro-1H-imidazo(1,2-a) (1,4)benzodiazepin-1-one
- DEA No. 2773
- Loprazolam [INN:BAN]
- Loprazolamum
- Loprazolamum [INN-Latin]
- Ru 31158
- Triazulenone
- Unii-759N8462G8
- Loprazolam
- (2Z)-6-(2-chlorophenyl)-2-[(4-methylpiperazin-1-yl)methylidene]-8-nitro-4H-imidazo[1,2-a][1,4]benzodiazepin-1-one
- Loprazolam USP/EP/BP
- Loprazolam (1mg/mL in Acetonitrile)
- (Z)-6-(2-Chlorophenyl)-2,4-dihydro-2-[(4-methyl-1-piperazinyl)methylene]-8-nitro-1H-imidazo[1,2-a][1,4]benzodiazepin-1-one
- Loprazolam solution
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Found 8 products.
Loprazolam
CAS:Controlled ProductApplications Sedative, hypnotic. Controlled substance (depressant).
References Agar, J.R., et al.: J. Med. Chem., 20, 1035 (1977), Clark, B.G., et al.: Drugs, 31, 500 (1986),Formula:C23H21ClN6O3Color and Shape:YellowMolecular weight:464.9Loprazolam (1mg/mL in Acetonitrile)
CAS:Controlled ProductFormula:C23H21ClN6O3Color and Shape:Single SolutionMolecular weight:464.9Loprazolam (100 μg/mL in Acetonitrile)
CAS:Controlled ProductFormula:C23H21ClN6O3Color and Shape:Single SolutionMolecular weight:464.9
