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CAS 61197-73-7

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Loprazolam

Description:
Loprazolam is a benzodiazepine derivative primarily used for its anxiolytic and hypnotic properties. It is characterized by its ability to enhance the effects of the neurotransmitter gamma-aminobutyric acid (GABA) at the GABA-A receptor, leading to sedative, anxiolytic, muscle relaxant, and anticonvulsant effects. Loprazolam is typically administered in tablet form and is known for its relatively rapid onset of action and moderate duration of effects. The substance is often prescribed for the short-term management of insomnia and anxiety disorders. Its pharmacokinetics indicate that it is metabolized in the liver, with metabolites that may also exhibit pharmacological activity. Common side effects can include drowsiness, dizziness, and potential dependence with prolonged use. Due to its sedative properties, caution is advised when operating machinery or driving after consumption. As with other benzodiazepines, it is important to use Loprazolam under medical supervision to mitigate risks of tolerance and withdrawal symptoms.
Formula:C23H21ClN6O3
InChI:InChI=1S/C23H21ClN6O3/c1-27-8-10-28(11-9-27)14-19-23(31)29-20-7-6-15(30(32)33)12-17(20)22(25-13-21(29)26-19)16-4-2-3-5-18(16)24/h2-7,12,14H,8-11,13H2,1H3/b19-14-
InChI key:InChIKey=UTEFBSAVJNEPTR-RGEXLXHISA-N
SMILES:O=C\1N2C=3C(C(=NCC2=N/C1=C\N4CCN(C)CC4)C5=C(Cl)C=CC=C5)=CC(N(=O)=O)=CC3
Synonyms:
  • (2Z)-6-(2-Chlorophenyl)-2,4-dihydro-2-[(4-methyl-1-piperazinyl)methylene]-8-nitro-1H-imidazo[1,2-a][1,4]benzodiazepin-1-one
  • (2Z)-6-(2-chlorophenyl)-2-[(4-methylpiperazin-1-yl)methylidene]-8-nitro-2,4-dihydro-1H-imidazo[1,2-a][1,4]benzodiazepin-1-one
  • (Z)-6-(o-Chlorophenyl)-2,4-dihydro-2-((4-methyl-1-piperazinyl)methylene)-8-nitro-1H-imidazo(1,2-a)(1,4)benzodiazepin-1-one
  • 1H-Imidazo(1,2-a)(1,4)benzodiazepin-1-one, 2,4-dihydro-6-(2-chlorophenyl)-2-((4-methyl-1-piperazinyl)methylene)-8-nitro-
  • 1H-Imidazo[1,2-a][1,4]benzodiazepin-1-one, 6-(2-chlorophenyl)-2,4-dihydro-2-[(4-methyl-1-piperazinyl)methylene]-8-nitro-, (2Z)-
  • 1H-Imidazo[1,2-a][1,4]benzodiazepin-1-one, 6-(2-chlorophenyl)-2,4-dihydro-2-[(4-methyl-1-piperazinyl)methylene]-8-nitro-, (Z)-
  • 6-(2-Chlorophenyl)-2,4-dihydro-2-((4-methyl-1-piperazinyl)methylene)-8-nitro-1H-imidazo(1,2-a) (1,4)benzodiazepin-1-one
  • DEA No. 2773
  • Loprazolam [INN:BAN]
  • Loprazolamum
  • See more synonyms
Found 7 products.
  • Loprazolam, 1mg/ml in Methanol

    Controlled Product
    CAS:
    Formula:C23H21ClN6O3
    Color and Shape:Single Solution
    Molecular weight:464.9

    Ref: LP-LPR-1281-FB-1LM

    1ml
    118.00€
  • Loprazolam

    Controlled Product
    CAS:
    Formula:C23H21ClN6O3
    Color and Shape:Neat
    Molecular weight:464.9

    Ref: LP-LPR-1281-FB

    10mg
    192.00€
    50mg
    617.00€
    100mg
    925.00€
  • Loprazolam

    Controlled Product
    CAS:

    Applications Sedative, hypnotic. Controlled substance (depressant).
    References Agar, J.R., et al.: J. Med. Chem., 20, 1035 (1977), Clark, B.G., et al.: Drugs, 31, 500 (1986),

    Formula:C23H21ClN6O3
    Color and Shape:Neat
    Molecular weight:464.9

    Ref: TR-L469510

    1mg
    235.00€
    2500µg
    328.00€
    25mg
    2,095.00€
  • Loprazolam (100 μg/mL in Acetonitrile)

    Controlled Product
    CAS:
    Formula:C23H21ClN6O3
    Color and Shape:Single Solution
    Molecular weight:464.9

    Ref: TR-KIT2128

    10x1ml
    323.00€
  • Loprazolam (1mg/mL in Acetonitrile)

    Controlled Product
    CAS:
    Formula:C23H21ClN6O3

    Ref: TR-KIT2125-1ML

    1x1ml
    946.00€
  • Loprazolam (100 μg/mL in Acetonitrile)

    Controlled Product
    CAS:
    Formula:C23H21ClN6O3

    Ref: TR-KIT2128-1ML

    10x1ml
    240.00€
  • Loprazolam (1mg/mL in Acetonitrile)

    Controlled Product
    CAS:
    Formula:C23H21ClN6O3
    Color and Shape:Single Solution
    Molecular weight:464.9

    Ref: TR-KIT2125

    1x1ml
    122.00€