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CAS 66981-73-5

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Tianeptine

Description:
Tianeptine is an atypical antidepressant primarily used in the treatment of major depressive disorder. It is classified as a selective serotonin reuptake enhancer (SSRE), which distinguishes it from traditional SSRIs that inhibit serotonin reuptake. Tianeptine's mechanism of action is believed to involve modulation of glutamate receptors and enhancement of neuroplasticity, contributing to its antidepressant effects. The substance is known for its unique pharmacological profile, which may also include anxiolytic and neuroprotective properties. Tianeptine is typically administered in oral form and has a relatively short half-life, necessitating multiple doses throughout the day for sustained effects. It is important to note that while tianeptine is approved for use in some countries, it is not universally recognized or available, and its use can be associated with potential for misuse and dependence. As with any medication, it is crucial to use tianeptine under medical supervision to monitor for efficacy and any adverse effects.
Formula:C21H25ClN2O4S
InChI:InChI=1/C21H25ClN2O4S/c1-24-18-9-6-5-8-16(18)21(23-13-7-3-2-4-10-20(25)26)17-12-11-15(22)14-19(17)29(24,27)28/h5-6,8-9,11-12,14,21,23H,2-4,7,10,13H2,1H3,(H,25,26)
InChI key:InChIKey=JICJBGPOMZQUBB-UHFFFAOYSA-N
SMILES:N(CCCCCCC(O)=O)C1C=2C(S(=O)(=O)N(C)C=3C1=CC=CC3)=CC(Cl)=CC2
Synonyms:
  • (1)-7-((3-Chloro-6,11-dihydro-6-methyldibenzo(c,f)(1,2)thiazepin-11-yl)amino)heptanoic acid S,S-dioxide
  • 7-[(3-Chloro-6,11-Dihydro-6-Methyldibenzo[C,F][1,2]Thiazepin-11-Yl)-Amino]Heptanoic Acid S,S-Dioxide
  • 7-[(3-Chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic acid
  • 7-[(3-Chloro-6-Methyl-5,5-Dioxido-6,11-Dihydrodibenzo[C,F][1,2]Thiazepin-11-Yl)Amino]Heptanoic Acid
  • Coaxil
  • Dibenzo[c,f][1,2]thiazepine, heptanoic acid deriv.
  • Heptanoic Acid, 7-[(3-Chloro-6,11-Dihydro-6-Methyl-5,5-Dioxidodibenzo[C,F][1,2]Thiazepin-11-Yl)Amino]-
  • Heptanoic acid, 7-[(3-chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]-, S,S-dioxide, (±)-
  • Tianeptine acid
  • Tianeptine
  • See more synonyms
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Found 1 products.
  • Tianeptine

    Controlled Product
    CAS:
    Tianeptine is a selective serotonin reuptake inhibitor that is used to treat depression. It has been demonstrated to have antidepressant effects in animals, and has been shown to increase the extracellular levels of glutamate in the hippocampus. Tianeptine may be effective in treating diseases such as infectious disease, bowel disease, and toll-like receptor (TLR) activation. The mechanism of action for tianeptine is not fully understood; however, it is believed that it acts by inhibiting glutamate uptake into presynaptic neurons and increasing serotonin levels in the brain. This drug also has an effect on receptors, which may be due to its ability to inhibit the binding of certain drugs to their receptors or block the activity of certain receptors.
    Formula:C21H25ClN2O4S
    Purity:Min. 95%
    Molecular weight:436.96 g/mol

    Ref: 3D-RCA98173

    100mg
    1,021.00€
    250mg
    1,388.00€