CAS 716354-04-0

AWXQYTLSBPWDMJ-KUMHGWDASA-N

Formula: C₃₆H₄₀ClF₂N₅O₃S

Synonyms:

• Benzenesulfonamide, 4-chloro-2-fluoro-5-[[4-(3-fluorophenyl)-4-[2-[(3-endo)-3-(2-methyl-1H-benzimidazol-1-yl)-8-azabicyclo[3.2.1]oct-8-yl]ethyl]-1-piperidinyl]carbonyl]-N-methyl-
• AWXQYTLSBPWDMJ-KUMHGWDASA-N

GSK163929

CAS: 716354-04-0

GSK163929 (compound 122) is an orally active CCR5 antagonist with anti-HIV properties and demonstrates low inhibitory potency against hEGR. Administered at a dosage of 2000 mg/kg/day (i.v., 7 d), it shows no adverse effects in rats, and at 250 mg/kg/day (i.v., 7 d), it is similarly non-toxic in dogs.

Formula: C₃₆H₄₀ClF₂N₅O₃S

Color and Shape: Solid

Molecular weight: 696.25

Ref: TM-T203363