CAS 73168-24-8

(B-mercapto-B,B-cyclopentamethyl-*enepropionyl1,O

Formula: C₅₂H₇₄N₁₄O₁₂S₂

InChI: InChI=1/C52H74N14O12S2/c1-78-32-16-14-31(15-17-32)25-35-46(73)63-36(24-30-10-4-2-5-11-30)47(74)61-34(18-19-40(53)67)45(72)64-37(26-41(54)68)48(75)65-38(29-79-80-52(27-43(70)60-35)20-6-3-7-21-52)50(77)66-23-9-13-39(66)49(76)62-33(12-8-22-58-51(56)57)44(71)59-28-42(55)69/h2,4-5,10-11,14-17,33-39H,3,6-9,12-13,18-29H2,1H3,(H2,53,67)(H2,54,68)(H2,55,69)(H,59,71)(H,60,70)(H,61,74)(H,62,76)(H,63,73)(H,64,72)(H,65,75)(H4,56,57,58)/t33?,34-,35-,36+,37-,38+,39-/m0/s1

Synonyms:

• 3-Mercapto-3-Methyl-Butyryl-Tyr(Me)-Phe-Gln-Asn-Cys-Pro-Arg-Gly-Nh2
• Vasopressin, 1-(1-mercaptocyclohexaneacetic acid)-2-(O- methyl-L-tyrosine)-8-L-arginine-
• (beta-Mercapto-beta,beta-cyclopentamethylene-propionyl(sup 1),O-Me-Tyr(sup 2),Arg(sup 8))-vasopressin
• (d(CH2)5(1)-O-Me-Tyr(2)-arg(8))vasopressin
• 1-(beta-Mercapto-beta,beta-cyclopentamethylenepropionic acid)-2-(O-methyl-tyr)-argipressin
• 1-(beta-Mercapto-beta,beta-cyclopentamethylenepropionic acid)-2-O-methyltyrosyl-8-arginine vasopressin
• Aavp
• Avpa
• Arginine vasopressin, beta-mercapto-(beta,beta-cyclopentamethylenepropionic acid)(1)-methyl-tyr(2)-
• Argipressin, (beta-mercapto)beta,beta-cyclopentamethylenepropionic acid(1)-O-methyl-tyr(2)-
• Cgp 25838
• Cpg 25838E
• Manning compound
• Mcppa-avp
• Sk&F 100273
• Skf 100273
• d(CH2)5(Tyr(Me)(2))AVP
• d(CH2)5-Tyr(Me)argipressin
• d(CH2)5Tyr(Me)AVP
• Glycinamide, N-((1-mercaptocyclohexyl)acetyl)-O-methyl-L-tyrosyl-L-phenylalanyl-L-glutaminyl-L-asparaginyl-L-cysteinyl-L-prolyl-L-arginyl-, cyclic (1-5)-disulfide

(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin

CAS: 73168-24-8

V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.

Formula: C₅₂H₇₄N₁₄O₁₂S₂

Purity: 98%

Color and Shape: Solid

Molecular weight: 1151.38

Ref: TM-TP2136

[β-Mercapto-β,β-cyclopentamethylenepropionyl1, O-me-Tyr2, Arg8]-Vasopressin

CAS: 73168-24-8

Formula: C₅₂H₇₄N₁₄O₁₂S₂

Molecular weight: 1151.36

Ref: 7W-GL5689

[Pmp1, Tyr(Me)2]-Arg8-Vasopressin

CAS: 73168-24-8

[Pmp1, Tyr(Me)2]-Arg8-vasopressin is a peptide that has been shown to activate the V2 receptor and inhibit vasopressin-induced water retention. It has also been shown to inhibit the binding of vasopressin to its receptor. The peptide is an excellent research tool for studying the interaction between the V2 receptor and vasopressin. The peptide is supplied at high purity in lyophilized form and can be reconstituted with water or buffer before use.

Formula: C₅₂H₇₅N₁₄O₁₂S₂

Purity: Min. 95%

Molecular weight: 1,152.4 g/mol

Ref: 3D-PVP-4203-V

(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin trifluoroacetate salt

CAS: 73168-24-8

The monoclonal antibody (mAb) is a recombinant protein that binds to the extracellular region of the vasopressin receptor. It is used in pharmacological research to study the physiological function and pharmacological effects of vasopressin. The mAb has been shown to be minimally toxic, with an LD50 value of greater than 10 mg/kg in mice. It has also been shown to inhibit viruses and inhibit drug-sensitive enzymes. This antibody can be used as a diagnostic tool for congestive heart disease, as well as in experimental models for studying the minimal toxicity and tumor treatment properties of various drugs.

Formula: C₅₂H₇₄N₁₄O₁₂S₂

Purity: Min. 95%

Molecular weight: 1,151.36 g/mol

Ref: 3D-FT109486

(d(CH₂)₅¹,Tyr(Me)²,Arg⁸)-Vasopressin

CAS: 73168-24-8

A very potent V₁ receptor antagonist (antivasopressor) with almost no antidiuretic activity.

Formula: C₅₂H₇₄N₁₄O₁₂S₂

Purity: > 99%

Color and Shape: White

Molecular weight: 1151.38

Ref: 01-4031349