CAS 75507-68-5
:Flupirtine maleate
Description:
Flupirtine maleate is a pharmaceutical compound primarily recognized for its analgesic and muscle relaxant properties. It is classified as a non-opioid analgesic and is often used in the management of pain, particularly in conditions such as neuropathic pain and musculoskeletal disorders. The substance acts as a selective neuronal potassium channel opener, which contributes to its pain-relieving effects by stabilizing neuronal excitability. Flupirtine maleate is typically administered in its maleate salt form, enhancing its solubility and bioavailability. The compound has a favorable safety profile compared to traditional analgesics, with a lower risk of dependence and fewer gastrointestinal side effects. However, it is essential to monitor liver function during treatment, as there have been reports of hepatotoxicity associated with its use. Flupirtine maleate is not widely available in all countries, and its use may be subject to regulatory restrictions. Overall, it represents a unique approach to pain management, particularly for patients who may not respond well to conventional analgesics.
Formula:C19H21FN4O6
InChI:InChI=1/C15H17FN4O2.C4H4O4/c1-2-22-15(21)19-12-7-8-13(20-14(12)17)18-9-10-3-5-11(16)6-4-10;5-3(6)1-2-4(7)8/h3-8H,2,9H2,1H3,(H,19,21)(H3,17,18,20);1-2H,(H,5,6)(H,7,8)/b;2-1-
InChI key:InChIKey=DPYIXBFZUMCMJM-BTJKTKAUSA-N
SMILES:N(C(OCC)=O)C1=C(N)N=C(NCC2=CC=C(F)C=C2)C=C1.C(=C\C(O)=O)\C(O)=O
Synonyms:- Carbamic acid, N-[2-amino-6-[[(4-fluorophenyl)methyl]amino]-3-pyridinyl]-, ethyl ester, (2Z)-2-butenedioate (1:1)
- Carbamic acid, [2-amino-6-[[(4-fluorophenyl)methyl]amino]-3-pyridinyl]-, ethyl ester, (2Z)-2-butenedioate (1:1)
- Carbamic acid, [2-amino-6-[[(4-fluorophenyl)methyl]amino]-3-pyridinyl]-, ethyl ester, (Z)-2-butenedioate (1:1)
- Efiret
- Ethyl 2-Amino-6-[(4-Fluorobenzyl)Amino]Pyridine-3-Carbamate, Compound With Maleic Acid (1:1)
- W 2964M
- ethyl {2-amino-6-[(4-fluorobenzyl)amino]pyridin-3-yl}carbamate (2Z)-but-2-enedioate
- Flupirtine maleate
- Flupirtinemaleatelupirtine
- Fluoxetine Maleate
- Ketadolon
- 2-Amino-6-[[(4-fluorophenyl)methyl]amino]-3-pyridinyl]-carbamic acid ethyl ester maleate salt
- Flupirtine Maleate Salt
- Carbamic acid, N-[2-amino-6-[[(4-fluorophenyl)methyl]amino]-3-pyridinyl]-, ethyl ester, (2Z)-2-butenedioate
- Flupirtine Maleate Impurity
- N-[2-AMino-6-(4-fluorobenzylaMino)pyridin-3-yl]carbaMic acid ethyl ester Maleate
- 2-AMINO-6-[[(4-FLUOROPHENYL)METHYL]AMINO]-3-PYRIDINYL]-CARBAMIC ACID, ETHYL ESTER MALEATE
- 2-Amino-3-(ethoxycarbonylamino)-6-(4-fluorobenzylamino)pyridine Maleate Salt
- N-[2-Amino-6-[[4-fluorophenyl)methyl]amino]-3-pyridinyl]carbamicacidethylestermaleate
- Flupirtine maleate, >=99%
- N-[2-AMino-6-[[(4-fluorophenyl)Methyl]aMino]-3-pyridinyl]carbaMic Acid Ethyl Ester (2Z)-2-Butenedioate
- Keiton
- Ethyl-2-amino-6-[(4-fluorbenzyl)amino]pyridin-3-carbamat, Verbindung mit Maleinsure (1:1)
- Flupirtine Maleat
- See more synonyms
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Flupirtine Maleate Salt
CAS:Formula:C15H17FN4O2·C4H4O4Purity:>98.0%(HPLC)(T)Color and Shape:White to Almost white powder to crystalMolecular weight:420.40Flupirtine maleate
CAS:Flupirtine maleateFormula:C15H17FN4O2·C4H4O4Purity:99.5%Molecular weight:420.39Flupirtine Maleate
CAS:Formula:C15H17FN4O2·C4H4O4Color and Shape:White To Off-White SolidMolecular weight:304.33 116.07Carbamic acid, [2-amino-6-[[(4-fluorophenyl)methyl]amino]-3-pyridinyl]-, ethyl ester, (Z)-2-butenedioate (1:1)
CAS:Formula:C19H21FN4O6Purity:98%Color and Shape:SolidMolecular weight:420.3916Ethyl (2-amino-6-((4-fluorobenzyl)amino)pyridin-3-yl)carbamate maleate
CAS:Formula:C19H21FN4O6Purity:98%Molecular weight:420.39Flupirtine maleate
CAS:Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.Formula:C19H21FN4O6Purity:99.5% - 99.9%Color and Shape:Yellow SolidMolecular weight:420.39Flupirtine maleate salt
CAS:Formula:C15H17FN4O2·C4H4O4Purity:≥ 98.0%Color and Shape:White to off-white powderMolecular weight:420.39Flupirtine maleate - Bio-X ™
CAS:Flupirtine is a pyridine derivative that is used as a non-opioid analgesic. Flupirtine promotes Bcl-2, raises glutathione levels, activates an inward rectifying potassium channel, and reverses the effect of calcium on neuronal cell death by inhibiting its release from intracellular stores. Although it doesn't attach to the receptor, flupirtine functions as an NMDA receptor antagonist. It is used for the treatment of fibromyalgia.Formula:C15H17FN4O2•C4H4O4Purity:Min. 95%Color and Shape:PowderMolecular weight:420.39 g/molFlupirtine maleate
CAS:Voltage-gated potassium channel openerFormula:C19H21FN4O6Purity:Min. 95%Color and Shape:PowderMolecular weight:420.39 g/molFlupirtine Maleate
CAS:Controlled ProductApplications Analgesic. Substituted pyridine with central analgesic properties. A potassium channel opener.
References Vaupel, D., et al.: Eur. J. Pharmacol., 162, 447 (1989), Nickel, B., et al.: Arzneim.-Forsch., 40, 909 (1990), Lunemann, J., et al.: J. Immunol., 168, 4881 (2002).Formula:C15H17FN4O2·C4H4O4Color and Shape:NeatMolecular weight:420.39
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