CAS 77614-16-5

dermorphin acetate

Description:

Dermorphin acetate is a synthetic peptide derived from the frog skin secretion of the Phyllomedusa genus, specifically known for its potent analgesic properties. It is classified as an opioid peptide, exhibiting a high affinity for mu-opioid receptors, which are primarily responsible for mediating pain relief and other effects associated with opioids. Dermorphin acetate is characterized by its relatively small molecular size and specific amino acid sequence, which contributes to its biological activity. The acetate form enhances its solubility and stability, making it suitable for various applications, including research in pain management and potential therapeutic uses. However, due to its strong opioid-like effects, dermorphin acetate also poses risks of addiction and side effects similar to other opioids. Its use is subject to regulatory scrutiny, and ongoing research aims to better understand its pharmacological profile and potential applications in medicine.

Formula: C₄₀H₅₀N₈O₁₀

InChI: InChI=1/C40H50N8O10/c1-23(44-37(55)29(41)18-25-9-13-27(50)14-10-25)36(54)46-30(19-24-6-3-2-4-7-24)38(56)43-21-34(52)45-31(20-26-11-15-28(51)16-12-26)40(58)48-17-5-8-33(48)39(57)47-32(22-49)35(42)53/h2-4,6-7,9-16,23,29-33,49-51H,5,8,17-22,41H2,1H3,(H2,42,53)(H,43,56)(H,44,55)(H,45,52)(H,46,54)(H,47,57)/t23-,29+,30+,31+,32+,33+/m1/s1

Synonyms:

• Tyrosyl-alanyl-phenylalanyl-glycyl-tyrosyl-prolyl-serinamide
• L-tyrosyl-D-alanyl-L-phenylalanylglycyl-L-tyrosyl-L-prolyl-L-serinamide
• Dermorphin
• Dermorphin trifluoroacetate salt
• (2S)-1-[(2S)-2-[[2-[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]-3-phenyl-propanoyl]amino]acetyl]amino]-3-(4-hydroxyphenyl)propanoyl]-N-[(1S)-1-carbamoyl-2-hydro
• Dermorphin Powder
• (2S)-N-[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]-1-[(2S)-2-[[2-[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]-3-phenylpropanoyl]amino]acetyl]amino]-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carboxamide
• Dermorphin HAc
• DERMORPHIN ACETATE
• L-Tyr-D-Ala-L-Phe-Gly-L-Tyr-L-Pro-L-Ser-NH2

Dermorphin

CAS: 77614-16-5

Dermorphin

Purity: ≥98%

Molecular weight: 802.87g/mol

Ref: 54-BUP21934

Dermorphin

CAS: 77614-16-5

Dermorphin is agonist of μ-opioid receptor (MOR) agonist.

Formula: C₄₀H₅₀N₈O₁₀

Purity: 98.82%

Color and Shape: Solid

Molecular weight: 802.87

Ref: TM-T7404

Dermorphin acetate

Controlled Product

CAS: 77614-16-5

The acetate salt of a hepta-peptide first isolated from the skin of  South American frogs.  It binds as an agonist with high potency and selectivity to mu opioid receptors.  Dermorphin is not found in humans or other mammals.  It appears to be made in mammals through an unusual posttranslational modification carried out by an amino acid isomerase.

Formula: C₄₀H₅₀N₈O₁₀C₂H₄O₂

Purity: Min. 95%

Color and Shape: Powder

Molecular weight: 862.92 g/mol

Ref: 3D-FD182310

Dermorphin

CAS: 77614-16-5

A hepta-peptide first isolated from the skin of  South American frogs.  It binds as an agonist with high potency and selectivity to mu opioid receptors.  Dermorphin is not found in humans or other mammals.  It appears to be made in mammals through an unusual posttranslational modification carried out by an amino acid isomerase.

Formula: C₄₀H₅₀N₈O₁₀

Purity: Min. 95%

Molecular weight: 802.87 g/mol

Ref: 3D-FD108711