CAS 83688-84-0

Tertatolol

Description:

Tertatolol, identified by its CAS number 83688-84-0, is a chemical compound that belongs to the class of beta-blockers, which are primarily used in the treatment of cardiovascular conditions. It is characterized by its ability to selectively block beta-adrenergic receptors, leading to a decrease in heart rate and blood pressure. Tertatolol exhibits a moderate lipophilicity, which influences its pharmacokinetic properties, including absorption and distribution in the body. The compound is typically administered in oral form and has a relatively long half-life, allowing for once-daily dosing in clinical settings. Its efficacy in managing conditions such as hypertension and arrhythmias is well-documented, although potential side effects may include fatigue, dizziness, and gastrointestinal disturbances. As with other beta-blockers, caution is advised in patients with asthma or certain heart conditions due to the risk of bronchoconstriction and bradycardia. Overall, Tertatolol represents a valuable therapeutic option in the management of various cardiovascular disorders.

Formula: C₁₆H₂₅NO₂S

InChI: InChI=1S/C16H25NO2S/c1-16(2,3)17-10-13(18)11-19-14-8-4-6-12-7-5-9-20-15(12)14/h4,6,8,13,17-18H,5,7,9-11H2,1-3H3

InChI key: InChIKey=HTWFXPCUFWKXOP-UHFFFAOYSA-N

SMILES: O(CC(CNC(C)(C)C)O)C1=C2C(=CC=C1)CCCS2

Synonyms:

• (±)-Tertatolol
• 1-((3,4-Dihydro-2H-1-benzothiopyran-8-yl)oxy)-3-((1,1-dimethylethyl)amino)-2-propanol
• 1-(tert-Butylamino)-3-(3,4-dihydro-2H-thiochromen-8-yloxy)propan-2-ol
• 2-Propanol, 1-[(3,4-dihydro-2H-1-benzothiopyran-8-yl)oxy]-3-[(1,1-dimethylethyl)amino]-
• 2H-1-Benzothiopyran, 2-propanol deriv.
• Racemic Tertatolol
• Racemic teraterol
• Tertatolol [BAN:INN]
• Tertatolol [INN:BAN]
• dl-Tertatolol
• 1-(tert-Butylamino)-3-((3,4-dihydro-2H-1-benzothiopyran-8-yl)oxy)propan-2-ol

rac Tertatolol

CAS: 83688-84-0

rac Tertatolol

Formula: C₁₆H₂₅NO₂S

Purity: 98%

Molecular weight: 295.44

Ref: 54-OR1129370

Tertatolol

CAS: 83688-84-0

Formula: C₁₆H₂₅NO₂S

Molecular weight: 295.44

Ref: 7W-GP4903

rac Tertatolol

CAS: 83688-84-0

Formula: C₁₆H₂₅NO₂S

Purity: 98%

Molecular weight: 295.4402

Ref: IN-DA00G4SR

rac Tertatolol

Controlled Product

CAS: 83688-84-0

Formula: C₁₆H₂₅NO₂S

Color and Shape: Neat

Molecular weight: 295.44

Ref: TR-T548800

Tertatolol

CAS: 83688-84-0

Tertatolol is a selective, non-specific inhibitor of cyclase. It has been used to study the role of cyclase in various aspects of the cardiovascular system and in infectious diseases. Tertatolol has also been found to reduce locomotor activity, glomerular filtration rate, and the toxicity of experimental models. In addition, it has been shown to be effective against inflammatory bowel disease. This drug binds to 2-adrenergic receptors with high affinity, inhibiting the binding of catecholamines and thereby decreasing the effects of noradrenaline on cardiac cells.

Formula: C₁₆H₂₅NO₂S

Purity: Min. 95%

Molecular weight: 295.4 g/mol

Ref: 3D-IDA68884

Tertatolol

CAS: 83688-84-0

Tertatolol is a highly active antagonist of beta-adrenoceptors and 5-HT receptors, and possesses the pharmacological effect of vasodilation.

Formula: C₁₆H₂₅NO₂S

Purity: 99.85%

Color and Shape: White Solid

Molecular weight: 295.44

Ref: TM-T17041