CAS 83846-83-7
:Ketanserin tartrate
Description:
Ketanserin tartrate is a pharmaceutical compound primarily used as an antihypertensive agent and for the treatment of certain psychiatric conditions. It is a selective antagonist of the serotonin 5-HT2A receptor and also exhibits some alpha-1 adrenergic receptor blocking activity. This dual action contributes to its effectiveness in managing blood pressure and improving mood disorders. Ketanserin tartrate is typically administered in its tartrate salt form, which enhances its solubility and bioavailability. The compound is characterized by its relatively low toxicity profile, making it suitable for long-term use in patients. Its pharmacokinetics involve oral administration, with a moderate half-life that allows for once or twice daily dosing. Common side effects may include dizziness, fatigue, and gastrointestinal disturbances, reflecting its influence on neurotransmitter systems. Overall, Ketanserin tartrate is recognized for its therapeutic benefits in cardiovascular and psychiatric applications, although its use may be limited by the availability of newer agents with improved efficacy and safety profiles.
Formula:C26H28FN3O9
InChI:InChI=1/C22H22FN3O3.C4H6O6/c23-17-7-5-15(6-8-17)20(27)16-9-11-25(12-10-16)13-14-26-21(28)18-3-1-2-4-19(18)24-22(26)29;5-1(3(7)8)2(6)4(9)10/h1-8,16H,9-14H2,(H,24,29);1-2,5-6H,(H,7,8)(H,9,10)/t;1-,2+
InChI key:InChIKey=KMTLTEVOQLMYRS-LREBCSMRSA-N
SMILES:O=C1C=2C(NC(=O)N1CCN3CCC(C(=O)C4=CC=C(F)C=C4)CC3)=CC=CC2.[C@@H]([C@H](C(O)=O)O)(C(O)=O)O
Synonyms:- 2,4(1H,3H)-Quinazolinedione, 3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-, (2R,3R)-2,3-dihydroxybutanedioate (1:1)
- 2,4(1H,3H)-Quinazolinedione, 3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-, [R-(R*,R*)]-2,3-dihydroxybutanedioate (1:1)
- Ketanserine tartrate
- Kjk 945
- Perketan
- R 49945
- Serepress
- Sufrexal
- Ketanserin tartrate
- 3-[2-[4-(4-fluorobenzoyl)piperidino]ethyl]quinazoline-2,4(1H,3H)-dione [R-(R*,R*)]-tartrate
- KETANSERIN TARTRATE (R 41468) (SELECTIVE 5-HT2/5-HT1C SEROTONI
- r-(r*,r*))-2,3-dihydroxybutanedioate(1:1)
- 3-[2-[4-(4-FLUOROBENZOYL)-1-PIPERIDINYL]ETHYL]-2,4[1H,3H]-QUINAZOLINEDIONE TARTRATE
- 3-[2-[4-(4-Fluorobenzoyl)piperidino]ethyl]-2,4-(1H,3H)-quinazolinedione tartrate
- 3-[2-[4-(4-FLUOROBENZOYL)-1-PIPERDINYL]ETHYL]-2,4(1H,3H)-QUINAZOLINEDIONE
- 3-(2-[4-(4-FLUOROBENZOYL)-1-PIPERIDINYL]ETHYL)-2,4(1H,3H)-QUINAZOLINEDIONE TARTRATE SALT
- 3-[2-[4-(4-FLUOROBENZOYL)-1-PIPERDINYL]ETHYL]-2,4(1H,3H)-QUINAZOLINEDIONE TARTRATE
- R 41468
- KETANSERIN TARTRATE SALT
- 3-(2-(4-(p-fluorobenzoyl)-1-piperidinyl)ethyl)-2,4(1h,3h)-quinazolinedionel
- 3-[2-(4-FLUOROBENZOYL)-1-PIPERDINYL]-ETHYL]-2,4(1H,3H)-QUINAZOLINEDIONE TARTRATE
- 4(1h,3h)-quinazolinedione,3-(2-(4-(4-fluorobenzoyl)-1-piperidinyl)ethyl)-(
- R 41468 (+)-tartrate salt, 3-(2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl)-2,4(1H,3H)-quinazolinedione (+)-tartrate salt
- R 41468 TARTRATE SALT
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Ketanserin tartrate, 98+%
CAS:Selective 5-HT2A serotonin receptor antagonistFormula:C22H22FN3O3·C4H6O6Purity:98+%Color and Shape:powder, White to off-whiteMolecular weight:545.523-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2,4[1H,3H]-quinazolinedione tartrate
CAS:Formula:C26H28FN3O9Purity:97%Color and Shape:SolidMolecular weight:545.5136Ketanserin Tartrate
CAS:Controlled ProductApplications Ketanserin Tartrate is used in nutrient-sensitized screening for drugs that shift energy metabolism from mitochondrial respiration to glycolysis for preventing a variety of diseases ranging from cancer to ischemic injury.
Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package
References Gohil, V. M., et al.: Nat. Biotechnol, 28, 249 (2010)Formula:C22H22FN3O3·C4H6O6Color and Shape:NeatMolecular weight:545.513-(2-(4-(4-Fluorobenzoyl)piperidin-1-yl)ethyl)quinazoline-2,4(1H,3H)-dione (2R,3R)-2,3-dihydroxysuccinate
CAS:3-(2-(4-(4-Fluorobenzoyl)piperidin-1-yl)ethyl)quinazoline-2,4(1H,3H)-dione (2R,3R)-2,3-dihydroxysuccinateFormula:C26H28FN3O9Purity:97%Molecular weight:545.51Ketanserin tartrate
CAS:Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.Formula:C26H28FN3O9Purity:99.80%Color and Shape:SolidMolecular weight:545.51Ketanserin tartrate - Bio-X ™
CAS:Ketanserin is a 5-HT2A serotonin receptor antagonist that is used for the treatment of hypertension. This drug is also used in research to study the serotonergic system. Ketanserin has been found to also block the vesicular monoamine transporter 2.Formula:C22H22FN3O3•C4H6O6Purity:Min. 95%Color and Shape:PowderMolecular weight:545.51 g/molKetanserin Tartrate
CAS:M02041 - Ketanserin Tartrate
Formula:C26H28FN3O9Purity:97%Color and Shape:SolidMolecular weight:545.52
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