CAS 85650-56-2
:Asenapine maleate
Description:
Asenapine maleate is an atypical antipsychotic medication primarily used in the treatment of schizophrenia and bipolar disorder. It is a salt form of asenapine, which is a dibenzo-oxepine derivative. The compound exhibits a complex structure that allows it to interact with various neurotransmitter receptors in the brain, particularly serotonin and dopamine receptors, which are crucial in mood regulation and psychotic disorders. Asenapine maleate is typically administered sublingually, allowing for rapid absorption and onset of action. Its pharmacological profile includes antagonistic activity at multiple receptor sites, contributing to its efficacy in managing symptoms of psychosis and mood stabilization. The substance is characterized by its low solubility in water, which influences its formulation and delivery methods. Common side effects may include sedation, weight gain, and metabolic changes, necessitating careful monitoring during treatment. Overall, asenapine maleate represents a significant option in psychiatric pharmacotherapy, with a unique mechanism of action and a specific therapeutic application.
Formula:C17H16ClNO·C4H4O4
InChI:InChI=1/C17H16ClNO.C4H4O4/c1-19-9-14-12-4-2-3-5-16(12)20-17-7-6-11(18)8-13(17)15(14)10-19;5-3(6)1-2-4(7)8/h2-8,14-15H,9-10H2,1H3;1-2H,(H,5,6)(H,7,8)/b;2-1-/t14-,15-;/s2
InChI key:InChIKey=GMDCDXMAFMEDAG-UHGYJBHVNA-N
SMILES:CN1C[C@]2([C@@](C=3C(OC=4C2=CC(Cl)=CC4)=CC=CC3)(C1)[H])[H].C(=C\C(O)=O)\C(O)=O
Synonyms:- (3aR,12bR)-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1H-dibenzo[2,3:6,7]oxepino[4,5-c]pyrrole (2Z)-but-2-enedioate
- (3aS,12bS)-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1H-dibenzo[2,3:6,7]oxepino[4,5-c]pyrrole (2Z)-but-2-enedioate
- 1H-Dibenz[2,3:6,7]oxepino[4,5-c]pyrrole, 5-chloro-2,3,3a,12b-tetrahydro-2-methyl-, (3aR,12bR)-rel-, (2Z)-2-butenedioate (1:1)
- 1H-Dibenz[2,3:6,7]oxepino[4,5-c]pyrrole, 5-chloro-2,3,3a,12b-tetrahydro-2-methyl-, trans-, (Z)-2-butenedioate (1:1)
- Asenapine Maleate
- Org 5222
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Found 14 products.
Asenapine Maleate
CAS:Formula:C17H16ClNO·C4H4O4Purity:>98.0%(HPLC)Color and Shape:White to Light yellow powder to crystalMolecular weight:401.849-chloro-4-methyl-13-oxa-4-azatetracyclo[12.4.0.0^{2,6}.0^{7,12}]octadeca-1(18),7,9,11,14,16-hexaene; but-2-enedioic acid
CAS:Formula:C21H20ClNO5Purity:99%Color and Shape:SolidMolecular weight:401.8402Asenapine Maleate
CAS:Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.Formula:C21H20ClNO5Purity:99.28%Color and Shape:SolidMolecular weight:401.84Asenapine Maleate
CAS:Formula:C17H16ClNO·C4H4O4Color and Shape:White To Off-White SolidMolecular weight:285.78 116.07Asenapine Maleate
CAS:Controlled ProductFormula:C17H16ClNO·C4H4O4Color and Shape:NeatMolecular weight:401.84Asenapine maleate
CAS:Formula:C17H16ClNO·C4H4O4Purity:≥ 98.0%Color and Shape:White to off-white powderMolecular weight:401.84Asenapine-13C,d3 Maleate
CAS:Controlled Product<p>Applications Asenapine-13C,d3 maleate, is the labeled analogue of Asenapine-13C,d3 Maleate, a 5-HT receptor antagonist developed for the treatment of acute schizophrenia and bipolar mania.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Tarazi. F.I., et al.: Drugs. Today., 45, 865 (2009); Boboaca, S.D., et al.: Int. J. Molec. Sci., 12, 4348 (2011); Audinot, V., et al.: Neuropsycopharmacol., 25, 410 (2001);<br></p>Formula:CC16D3H13ClNO·C4H3O4Color and Shape:NeatMolecular weight:404.843Asenapine maleate
CAS:Controlled Product<p>Inhibits dopamine, serotonin and adrenergic receptors</p>Formula:C17H16ClNOC4H4O4Purity:Min. 95%Color and Shape:White PowderMolecular weight:401.84 g/molAsenapine Maleate
CAS:Controlled Product<p>Applications Asenapine Maleate, is a 5-HT receptor antagonist developed for the treatment of acute schizophrenia and bipolar mania. Antagonist of serotonin, norepinephrine, dopamine and histamine receptors.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Tarazi. F.I., et al.: Drugs. Today., 45, 865 (2009); Boboaca, S.D., et al.: Int. J. Molec. Sci., 12, 4348 (2011); Audinot, V., et al.: Neuropsycopharmacol., 25, 410 (2001);<br></p>Formula:C17H16ClNO·C4H4O4Color and Shape:NeatMolecular weight:401.84
![9-chloro-4-methyl-13-oxa-4-azatetracyclo[12.4.0.0^{2,6}.0^{7,12}]octadeca-1(18),7,9,11,14,16-hexae…](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FIN%2Fthumb%2FDA0036DT.jpg&w=3840&q=75)
