CAS 956906-93-7

PF 04217903 mesylate

Description:

PF 04217903 mesylate, with the CAS number 956906-93-7, is a chemical compound that belongs to a class of substances known for their potential therapeutic applications, particularly in the field of pharmacology. This compound is characterized by its mesylate salt form, which enhances its solubility and stability, making it suitable for various formulations. Typically, compounds like PF 04217903 mesylate are evaluated for their efficacy and safety in clinical settings, often targeting specific biological pathways or receptors. The mesylate group contributes to its pharmacokinetic properties, influencing absorption, distribution, metabolism, and excretion. Additionally, the compound may exhibit specific interactions with biological molecules, which can be crucial for its intended therapeutic effects. As with many pharmaceutical agents, understanding its mechanism of action, potential side effects, and interactions with other drugs is essential for its application in medical treatments. Further research and clinical trials are often necessary to fully elucidate its characteristics and therapeutic potential.

Formula: C₂₀H₂₀N₈O₄S

Synonyms:

• PF-04217903.MsOH
• 4-[1-(6-QuinolinylMethyl)-1H-1,2,3-triazolo[4,5-b]pyrazin-6-yl]-1H-pyrazole-1-ethanol Methanesulfonate
• 4-[1-(6-Quinolinylmethyl)-1H-1,2,3-triazolo[4,5-b]pyrazin-6-yl]-1H-pyrazole-1-ethanol mesylate
• PF-04217903 Methanesulfonate
• 2-(4-(1-(Quinolin-6-ylmethyl)-1H-[1,2,3]triazolo[4,5-b]pyrazin-6-yl)-1H-pyrazol-1-yl)ethan-1-ol methanesulfonate
• PF04217903 METHANESULFONATE;PF 04217903 METHANESULFONATE
• HBEMHKVWZJTVOC-UHFFFAOYSA-N
• PF 04217903 mesylate
• 4-[1-(6-Quinolinylmethyl)-1H-1,2,3-triazolo[4,5-b]pyrazin-6-yl]-1H-pyrazole-1-ethanol methanesulfonate (1:1)

PF-04217903 methanesulfonate

CAS: 956906-93-7

Formula: C₂₀H₂₀N₈O₄S

Purity: 99.82%

Color and Shape: Solid

Molecular weight: 468.4890

Ref: IN-DA01DOMZ

2-(4-(1-(Quinolin-6-Ylmethyl)-1H-[1,2,3]Triazolo[4,5-B]Pyrazin-6-Yl)-1H-Pyrazol-1-Yl)Ethan-1-Ol Methanesulfonate

CAS: 956906-93-7

2-(4-(1-(Quinolin-6-Ylmethyl)-1H-[1,2,3]Triazolo[4,5-B]Pyrazin-6-Yl)-1H-Pyrazol-1-Yl)Ethan-1-Ol Methanesulfonate

Purity: 98%

Molecular weight: 468.49g/mol

Ref: 54-OR1024319

PF-04217903 methanesulfonate

CAS: 956906-93-7

PF-04217903 methanesulfonate is a potent ATP-competitive inhibitor of c-Met kinase (Ki of 4.8 nM for human c-Met).

Formula: C₂₀H₂₀N₈O₄S

Purity: 98%

Color and Shape: Solid

Molecular weight: 468.49

Ref: TM-T12417

PF 04217903 mesylate

CAS: 956906-93-7

PF 04217903 mesylate is a factor receptor inhibitor that inhibits the transcription of insulin-like growth factor and epidermal growth factor. It is used in the treatment of neoplastic disease, such as breast cancer, ovarian cancer, and prostate cancer. PF 04217903 mesylate also inhibits angiogenesis by inhibiting the expression of transcription factors that are involved in this process. These effects may be due to its ability to inhibit the production of erythropoietin and other proangiogenic molecules. PF 04217903 mesylate has been shown to inhibit the proliferation of vascular endothelial cells in vitro and in vivo.

Formula: C₁₉H₁₆N₈O·CH₃SO₃H

Purity: Min. 95%

Molecular weight: 468.49 g/mol

Ref: 3D-GNB90693