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CAS 98123-83-2

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Epsiprantel

Description:
Epsiprantel is a chemical compound primarily used as an anthelmintic agent, particularly effective against certain parasitic infections in veterinary medicine. It belongs to the class of compounds known as praziquantel derivatives, which are characterized by their ability to disrupt the integrity of the parasite's cell membranes, leading to paralysis and death of the organism. Epsiprantel is typically administered orally and is known for its relatively low toxicity to mammals, making it a safer option for treating infections in animals. The compound is soluble in organic solvents but has limited solubility in water, which influences its formulation and delivery methods. Its mechanism of action involves the alteration of calcium ion permeability in the parasite, resulting in muscle contraction and subsequent paralysis. Epsiprantel is often used in combination with other antiparasitic agents to enhance efficacy and broaden the spectrum of activity against various helminths. As with any pharmaceutical, proper dosage and administration are crucial to ensure effectiveness while minimizing potential side effects.
Formula:C20H26N2O2
InChI:InChI=1S/C20H26N2O2/c23-19-14-21(20(24)16-8-2-1-3-9-16)13-18-17-11-5-4-7-15(17)10-6-12-22(18)19/h4-5,7,11,16,18H,1-3,6,8-10,12-14H2
InChI key:InChIKey=LGUDKOQUWIHXOV-UHFFFAOYSA-N
SMILES:O=C1N2C(C=3C(CCC2)=CC=CC3)CN(C(=O)C4CCCCC4)C1
Synonyms:
  • Epsiprantel
  • BRL 38705
  • (+-)-2-(Cyclohexylcarbonyl)-2,3,6,7,8,12b-hexahydropyrazino(2,1-a)(2)benzazepin-4(1H)-one
  • Epsiprantelum
  • Pyrazino[2,1-a][2]benzazepin-4(1H)-one, 2-(cyclohexylcarbonyl)-2,3,6,7,8,12b-hexahydro-
  • Epsiprantelum [Latin]
  • Epsiprantel [INN:BAN]
  • BRL 38705
  • 2-(Cyclohexylcarbonyl)-2,3,6,7,8,12b-hexahydropyrazino[2,1-a][2]benzazepin-4(1H)-one
  • Epsiprantel
  • See more synonyms
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