Inhibitor Enzymes
Inhibitor enzymes are molecules that decrease or block the activity of enzymes, preventing them from catalyzing their specific reactions. These inhibitors can be reversible or irreversible and are crucial tools in research and drug development for studying enzyme mechanisms, controlling metabolic pathways, and developing therapeutic agents. Inhibitor enzymes are widely used to modulate biological processes and to treat various diseases by targeting specific enzymes. At CymitQuimica, we offer a comprehensive range of high-quality enzyme inhibitors to support your research and pharmaceutical development needs.
Found 123 products of "Inhibitor Enzymes"
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Benzyl Methyl Carbonate
CAS:Controlled Product<p>Applications Benzyl Methyl Carbonate is used in designing of inhibitors for serine and thiol proteases.<br></p>Formula:C9H10O3Color and Shape:NeatMolecular weight:166.17(R)-Pinocembrin
CAS:Controlled Product<p>Applications (2R)-Pinocembrin is the (R)-enantiomer of Pinocembrin, a flavanoid with antioxidant activity found in damiana, honey, and propolis. (2R)-Pinocembrin is a potential inhibitor of PIM1 kinase, an oncogene that has been implicated in the development of leukemias, lymphomas, and prostate cancer.<br>References Zhao, J. et al.: J. Ethnopharmacol., 120, 387 (2008); Holder, S. et al.: Mol. Cancer Ther., 6, 163 (2007); Holder, S. et al.: Bioorg. Med. Chem., 15, 6463 (2007);<br></p>Formula:C15H12O4Color and Shape:WhiteMolecular weight:256.25Teneligliptin Hydrobromide (2:5)
CAS:Controlled Product<p>Applications Teneligliptin Hydrobromide (2:5) is a dipeptidyl peptidase-4 (DPP-4) inhibitor that is used to treat type 2 diabetes. It is eliminated via excretion, and has a half-life of 24.2 hours in the human body.<br>References Goda, M. & Kadowaki, T.: Drugs Today, 49, 615 (2013); Kishimoto, M.: Diabetes Metab. Syndr. Obes., 6, 187 (2012)<br></p>Formula:C22H32·5Br2·5N6OSColor and Shape:NeatMolecular weight:628.86Bis(2-butoxyethyl) 2-(3-Hydroxybutoxy)ethyl Phosphate Triester
CAS:Controlled Product<p>Applications Bis(2-butoxyethyl) 2-(3-Hydroxybutoxy)ethyl Phosphate Triester is derived from 2-Butoxyethanol (B692895), which is a reagent in the synthesis of 4-butoxyethoxy-N-octadecyl-1,8-naphthalimide as a new fluorescent probe for the determination of proteins. Also used as a reagent in the synthesis of 4-hydroxybenzaldehyde derivatives as tyrosinase inhibitors.<br>References Sun, Y., et al.: Bioorg. Med. Chem. Lett., 21, 3798 (2011); Yi, W., et al.: Eur. J. Med. Chem., 45, 639 (2010)<br></p>Formula:C18H39O8PColor and Shape:Colourless To Light YellowMolecular weight:414.47Daidzein Diglucuronide
CAS:Controlled ProductFormula:C27H26O16Color and Shape:White To Off-WhiteMolecular weight:606.49Nicotelline
CAS:Controlled Product<p>Applications Nicotelline is a Nicotine (N412420) related metabolite with potential as an inhibitor of human cytochrome P-450 2A6.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Denton, T. et al.: Biochem. Pharm., 67, 751 (2004); Gorrod, J. et al.: Anal. Det. Nic. Rel. Comp. Metab., 69, (1999);<br></p>Formula:C15H11N3Color and Shape:NeatMolecular weight:233.27(3S,5S)-Atorvastatin Calcium Salt
CAS:Controlled Product<p>Impurity Atorvastatin Related Compound E<br>Applications Impuritiy of Atorvaststin (A791750), a selective, competitive HMG-CoA reductase inhibitor. Atorvastatin is the only drug in its class specfically indicated for lowering both elevated LDL-cholesterol and triglycerides in patients with hypercholesterolemia. Atorvastatin Related Compound E<br>References Kearney, A.S., et al.: Pharm. Res., 10, 1461 (1993), Heinonen, T.M., et al.: Clin. Ther., 18, 853 (1996), Whitfield, L.R., et al.: Eur. J. Drug Metab. Pharmacokinet., 25, 97 (2000),<br></p>Formula:C33H34FN2O5·CaColor and Shape:NeatMolecular weight:1155.34N-(2-Hydroxyethyl)-1-deoxy-L-idonojirimycin Hydrochloride
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications α-Glycosidase inhibitor.<br>References van de Water, F., et al.: Drug Metab. Rev., 37, 443 (2005), Koepsell, H., et al.: Pharm. Res., 24, 1227 (2007), Jappar, D., et al.: Pharm. Res., 26, 172 (2009),<br></p>Formula:C8H18ClNO5Color and Shape:NeatMolecular weight:243.69N-(2-Hydroxyethyl)-1-deoxy-L-altronojirimycin Hydrochloride Salt
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications α-Glycosidase inhibitor.<br>References Jefferies, I., et al.: Bioorg. Med. Chem. Lett., 7, 1171 (1997), Hassan, A., et al.: Carbohydr. Res., 339, 1565 (2004),<br></p>Formula:C8H18ClNO5Color and Shape:NeatMolecular weight:243.68523'-Deoxyadenosine 5’-Diphosphate Triethylamine Salt (>90%)
CAS:<p>Stability Hygroscopic<br>Applications 3'-Deoxyadenosine 5’-Diphosphate Triethylamine Salt, is a nucleotide and was proposed to be a possible inhibitor of DNA synthesis.<br>References Frederiksen, Sune.: Biochimica et Biophysica Acta, 76(3), 366-71 (1963)<br></p>Formula:C10H15N5O9P2•xC6H15NPurity:>90%Color and Shape:NeatMolecular weight:411.20 + x(101.19)Naringenin chalcone
CAS:Controlled ProductFormula:C15H12O5Color and Shape:NeatMolecular weight:272.25Nitromifene Citrate (E/Z mixture)
CAS:Controlled Product<p>Applications Nitromifene citrate is a non-steroidal estrogen antagonist. It is structurally similar to Tamoxifen (T006000) which is a selective estrogen response modifier (SERM).<br>References Rudick, C., et al.: Endorcrinol., 144, 179 (2003); Sutherland, R., et al.: Nature, 267, 434 (1977)<br></p>Formula:C33H36N2O11Color and Shape:Yellow To OrangeMolecular weight:636.65LCZ696
CAS:<p>Applications LCZ696 is a novel dual-acting inhibitor of angiotensin II receptor and neprilysin, which can be used for blood pressure reduction.<br>References Ruilope, L.M.; et al.: Lancet, 375, 1255 (2010)<br></p>Formula:C24H28NO5·C24H27N5O3·3Na·x(H2O)Color and Shape:MixtureMolecular weight:479.48 + (433.47) + x(18.02)2,5-Dideoxy-2,5-imino-D-mannitol
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications A glucosidase inhibitor.<br>References Fellows, L.E.: Pestic. Sci., 17, 602 (1986)<br></p>Formula:C6H13NO4Color and Shape:Off White SolidMolecular weight:163.17Vitamin B12 e-Monocarboxylic Acid
CAS:<p>Stability Hygroscopic<br>Applications Vitamin B12 Monocarboxylic Acid is an impurity of Vitamin B12 (V676005) which is a water-soluble vitamin with a key role in the normal functioning of the brain and nervous system, and for the formation of blood.<br>References Rickes, et al.: Science, 107, 396 (1948); Kirschbaum, J., et al.: Anal. Profiles Drug Subs., 10, 183 (1981); Grasbeck, R., et al.: Clin. Biochem., 17, 99 (1984)<br></p>Formula:C63H87CoN13O15PColor and Shape:Dark Red SolidMolecular weight:1356.35Abamine
CAS:Controlled Product<p>Applications Abamine is an inhibitor of 9-Cis-Epoxycarotenoid dioxygenase (NCED), the key regulatory enzyme in the plant hormone abscisic acid (ABA) biosynthesis pathway.<br>References Kitahata, N., et al.: Bioorg. Med. Chem., 14, 5555 (2006); Han, S., et al.: Bioorg. Med. Chem. Lett., 14, 3033 (2004)<br></p>Formula:C21H24FNO4Color and Shape:NeatMolecular weight:373.42tert-Butyl (2S,4S)-4-[4-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]-2-[(1,3-thiazolidin-3-yl)carbonyl]pyrrolidine-1-carboxylate
CAS:Controlled Product<p>Applications tert-Butyl (2S,4S)-4-[4-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]-2-[(1,3-thiazolidin-3-yl)carbonyl]pyrrolidine-1-carboxylate is an orally anti-diabetic agent as a inhibitors of dipeptidylpeptidase IV (DPP-4).<br>References Yoshida, T., et al.: Bioorg. Med. Chem., 20, 5705-5719 (2012);<br></p>Formula:C27H38N6O3SColor and Shape:NeatMolecular weight:526.69CP-10447
CAS:<p>Applications CP-10447 is an inhibitor apolipoprotein B (apoB) and triglyceride secretion in human hepatoma cells (HepG2) by inhibiting MTP activity and stimulating the early ER degradation of apoB. It is useful tool for further study of the mechanisms of apoB secretion and triglyceride-rich lipoprotein assembly.<br>References Haghpassand, M. et al.: J. Lipid. Res., 37, 1468 (1996); Pan, M. et al.: J. Biol. chem., 275, 27399 (2000);<br></p>Formula:C16H13BrN2OColor and Shape:NeatMolecular weight:329.19N-(10-Aminodecyl)-5-chloro-1-naphthalenesulfonamide Hydrochloride
CAS:Controlled Product<p>Applications Naphthalenesulfonamides derivatives are neoplasm inhibitors.<br>References Hidaka, H., et al.: Proc. Nat. Acad. Sci. USA, 78, 4354 (1981)<br></p>Formula:C20H29ClN2O2S·ClHColor and Shape:NeatMolecular weight:433.44
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