EGFR
EGFR (epidermal growth factor receptor) inhibitors are compounds that block the signaling of EGFR, a receptor that is often overexpressed in various cancers and plays a critical role in angiogenesis. EGFR inhibitors are used to prevent tumor growth and metastasis by disrupting the pathways that promote blood vessel formation in tumors. These inhibitors are widely used in cancer research and therapy. At CymitQuimica, we offer a diverse selection of high-quality EGFR inhibitors to support your research in oncology and angiogenesis.
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Leptomycin B
CAS:87081-35-4
Leptomycin B: potent CRM1 inhibitor, blocks protein nuclear export and cell cycle, antifungal, modifies cysteine.
Formula:
C33H48O6
Purity:
99.04% - 99.71%
Color and Shape:
White Crystalline Solid
Molecular weight:
540.73
Ref: TM-T15735
| 1mg | 202.00 € | ||
| 2mg | 341.00 € | ||
| 5mg | 620.00 € | ||
| 10mg | 882.00 € | ||
| 25mg | 1,320.00 € | ||
| 50mg | 1,776.00 € | ||
| 100mg | 2,403.00 € | ||
| 1mL*10mM (DMSO) | 283.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Genistein
CAS:446-72-0
Genistein (NPI 031L) is a natural soy isoflavone, a multi-targeted tyrosine kinase inhibitor. Genistein has …
Formula:
C15H10O5
Purity:
98.22% - 99.69%
Color and Shape:
Rectangular Or Six-Sided Rods From 60% Alcohol Dendritic Needles From Ether Solid
Molecular weight:
270.24
Ref: TM-T1737
| 50mg | 46.00 € | ||
| 100mg | 59.00 € | ||
| 500mg | 95.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Rostafuroxin
CAS:156722-18-8
Rostafuroxin (PST 2238) has been used in trials studying the treatment of Essential Hypertension.
Formula:
C23H34O4
Purity:
100% - 99.08%
Color and Shape:
Solid
Molecular weight:
374.51
Ref: TM-T2621
| 2mg | 44.00 € | ||
| 5mg | 65.00 € | ||
| 10mg | 107.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 350.00 € | ||
| 100mg | 522.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Almonertinib mesylate
CAS:2134096-06-1
Almonertinib mesylate: EGFR tyrosine kinase inhibitor, targets EGFR-mutant non-small cell lung cancer.
Formula:
C31H39N7O5S
Purity:
98.85%
Color and Shape:
Solid
Molecular weight:
621.75
Ref: TM-T9865
| 1mg | 55.00 € | ||
| 5mg | 116.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 319.00 € | ||
| 50mg | 449.00 € | ||
| 100mg | 638.00 € | ||
| 200mg | 840.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
(Rac)-JBJ-04-125-02
CAS:2140807-05-0
(Rac)-JBJ-04-125-02 (JBJ-04-125-02) is effective as a single agent in both in vitro and in vivo …
Formula:
C29H26FN5O3S
Purity:
95.85%
Color and Shape:
Solid
Molecular weight:
543.61
Ref: TM-T8872
| 1mg | 105.00 € | ||
| 5mg | 216.00 € | ||
| 10mg | 354.00 € | ||
| 25mg | 597.00 € | ||
| 50mg | 852.00 € | ||
| 100mg | 1,159.00 € | ||
| 1mL*10mM (DMSO) | 263.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Mobocertinib
CAS:1847461-43-1
Mobocertinib (tak788) is a potent inhibitor of epidermal growth factor receptor (EGFR) and an antineoplastic …
Formula:
C32H39N7O4
Purity:
98.66% - 99.47%
Color and Shape:
Solid
Molecular weight:
585.7
Ref: TM-T8151
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 119.00 € | ||
| 100mg | 188.00 € | ||
| 500mg | 490.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
CUDC-101
CAS:1012054-59-9
CUDC-101 is a potent inhibitor of HDAC, EGFR and HER2 with IC50s of 4.4, 2.4 …
Formula:
C24H26N4O4
Purity:
95.76% - 99.12%
Color and Shape:
Solid
Molecular weight:
434.49
Ref: TM-T3108
| 5mg | 50.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 197.00 € | ||
| 100mg | 350.00 € | ||
| 200mg | 520.00 € | ||
| 500mg | 840.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Afatinib
CAS:850140-72-6
Afatinib (BIBW 2992) is an irreversible and orally EGFR family inhibitor that inhibits EGFR and …
Formula:
C24H25ClFN5O3
Purity:
97.56% - 99.9%
Color and Shape:
Off-White Solid
Molecular weight:
485.94
Ref: TM-T21312
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 86.00 € | ||
| 50mg | 115.00 € | ||
| 100mg | 144.00 € | ||
| 200mg | 177.00 € | ||
| 500mg | 300.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
PD153035
CAS:153436-54-5
PD153035 (NSC-669364) hydrochloride is an effective and selective inhibitor of EGFR (Ki/IC50: 5.2/29 pM, in …
Formula:
C16H14BrN3O2
Purity:
98.92% - 99.31%
Color and Shape:
Solid
Molecular weight:
360.21
Ref: TM-T2041
| 10mg | 42.00 € | ||
| 25mg | 80.00 € | ||
| 50mg | 133.00 € | ||
| 100mg | 225.00 € | ||
| 200mg | 335.00 € | ||
| 1mL*10mM (DMSO) | 40.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Nazartinib
CAS:1508250-71-2
Nazartinib (EGF816) (EGF816, NVS-816) is a covalent, irreversible, mutant-selective EGFR inhibitor that has nanomolar inhibitory …
Formula:
C26H31ClN6O2
Purity:
98.31% - ≥95%
Color and Shape:
Solid Powder
Molecular weight:
495.02
Ref: TM-T3506
| 1mg | 37.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 528.00 € | ||
| 500mg | 1,159.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
PD-089828
CAS:179343-17-0
PD 089828 inhibits FGFR1, PDGFRβ, EGFR (IC50s: 0.15-5.47 μM), and c-Src (IC50: 0.18 μM).
Formula:
C18H18Cl2N6O
Purity:
96.78%
Color and Shape:
Solid
Molecular weight:
405.28
Ref: TM-T8976
| 1mg | 37.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 374.00 € | ||
| 100mg | 547.00 € | ||
| 500mg | 1,159.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Naquotinib mesylate
CAS:1448237-05-5
Naquotinib mesylate (ASP8273 (mesylate)) is an orally available, mutant-selective and irreversible inhibitor of EGFR(iC50s of …
Formula:
C31H46N8O6S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
658.81
Ref: TM-T12175
| 2mg | 64.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Almonertinib hydrochloride
CAS:2134096-03-8
Almonertinib hydrochloride (HS-10296 hydrochloride) is a small molecule inhibitor of EGFR-activating mutations and T790M-resistant mutation.
Formula:
C30H36ClN7O2
Purity:
98.01% - 98.12%
Color and Shape:
Solid
Molecular weight:
562.1
Ref: TM-T5675
| 1mg | 92.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 311.00 € | ||
| 25mg | 537.00 € | ||
| 50mg | 753.00 € | ||
| 100mg | 1,026.00 € | ||
| 500mg | 2,080.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
BMS-690514
CAS:859853-30-8
BMS-690514 is a potent and orally active inhibitor of EGFR and VEGFR. It has IC50s …
Formula:
C19H24N6O2
Purity:
99.08%
Color and Shape:
Solid
Molecular weight:
368.43
Ref: TM-T14677
| 2mg | 139.00 € | ||
| 5mg | 225.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
MAPK-IN-2
MAPK-IN-2 (compound 3h) is an efficacious MAPK inhibitor with antineoplastic properties that significantly hinders proliferation …
Formula:
C20H11Cl2N3O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
380.23
Ref: TM-T79572
| 5mg | 922.00 € | ||
| 25mg | 1,539.00 € | ||
| 50mg | 2,303.00 € |
Estimated delivery in United States, on Friday 2 May 2025
ZM323881 hydrochloride
CAS:193000-39-4
ZM323881 hydrochloride (ZM 323881 HCl) is a potent and selective VEGFR2 inhibitor.
Formula:
C22H19ClFN3O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
411.86
Ref: TM-T1991
| 5mg | 72.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 404.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Friday 2 May 2025
Icotinib
CAS:610798-31-7
Icotinib (Conmana) is an orally available quinazoline-based inhibitor of epidermal growth factor receptor (EGFR), with …
Formula:
C22H21N3O4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
391.42
Ref: TM-T6153
| 1mg | 48.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 155.00 € | ||
| 25mg | 283.00 € | ||
| 50mg | 527.00 € | ||
| 100mg | 712.00 € | ||
| 1mL*10mM (DMSO) | 97.00 € |
Estimated delivery in United States, on Friday 2 May 2025
lavendustin A
CAS:125697-92-9
lavendustin A (RG-14355) is a potent, cell-permeable inhibitor of epidermal growth factor receptor (EGFR) tyrosine …
Formula:
C21H19NO6
Purity:
98%
Color and Shape:
Off-White Solid
Molecular weight:
381.38
Ref: TM-T4183
| 1mg | 74.00 € | ||
| 5mg | 143.00 € |
Estimated delivery in United States, on Friday 2 May 2025
Icotinib Hydrochloride
CAS:1204313-51-8
Icotinib Hydrochloride, an oral EGFR inhibitor (BPI-2009H), may halt cancer growth by blocking EGFR signaling.
Formula:
C22H22ClN3O4
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
427.88
Ref: TM-T2307
| 5mg | 60.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 140.00 € | ||
| 50mg | 227.00 € | ||
| 100mg | 338.00 € | ||
| 200mg | 500.00 € | ||
| 1mL*10mM (DMSO) | 66.00 € |
Estimated delivery in United States, on Friday 2 May 2025
TAK-285
CAS:871026-44-7
TAK-285 is a novel dual HER2 and EGFR(HER1) inhibitor, >10-fold selectivity for HER1/2 than HER4, …
Formula:
C26H25ClF3N5O3
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
547.96
Ref: TM-T6039
| 1mg | 40.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 378.00 € | ||
| 100mg | 563.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Friday 2 May 2025
