EGFR
EGFR (epidermal growth factor receptor) inhibitors are compounds that block the signaling of EGFR, a receptor that is often overexpressed in various cancers and plays a critical role in angiogenesis. EGFR inhibitors are used to prevent tumor growth and metastasis by disrupting the pathways that promote blood vessel formation in tumors. These inhibitors are widely used in cancer research and therapy. At CymitQuimica, we offer a diverse selection of high-quality EGFR inhibitors to support your research in oncology and angiogenesis.
Read more
Epertinib
CAS:908305-13-5
Epertinib is a reversible and selective tyrosine kinase inhibitor of EGFR, HER2, and HER4 (IC50s: …
Formula:
C30H27ClFN5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
560.02
Ref: TM-T11213L
| 25mg | 1,262.00 € | ||
| 50mg | 1,644.00 € | ||
| 100mg | 2,336.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Larotinib
CAS:1438072-11-7
Larotinib is an orally active, potent, and broad-spectrum tyrosine kinase inhibitor (TKI) with an IC50 …
Formula:
C24H26ClFN4O4
Purity:
98.45%
Color and Shape:
Liquid
Molecular weight:
488.94
Ref: TM-T73334
| 1mg | 80.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 253.00 € | ||
| 25mg | 430.00 € | ||
| 50mg | 615.00 € | ||
| 100mg | 861.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
H-9 dihydrochloride
CAS:116700-36-8
H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.
Formula:
C11H15Cl2N3O2S
Purity:
96.57%
Color and Shape:
Solid
Molecular weight:
324.23
Ref: TM-T22833
| 1mg | 35.00 € | ||
| 5mg | 71.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 152.00 € | ||
| 50mg | 219.00 € | ||
| 100mg | 324.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
RTC-5
CAS:1423077-49-9
RTC-5 (TRC-382) is a phenothiazine compound that has been specifically enhanced for its potent anti-cancer …
Formula:
C24H22ClF3N2O3S
Purity:
98.14%
Color and Shape:
Solid
Molecular weight:
510.96
Ref: TM-T12777
| 5mg | 52.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 278.00 € | ||
| 100mg | 403.00 € | ||
| 500mg | 849.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Tyrphostin A25
CAS:118409-58-8
Tyrphostin A25 (Tyrphostin AG 82) is a specific EGFR tyrosine kinase inhibitor and GPR35 agonist …
Formula:
C10H6N2O3
Purity:
98.76%
Color and Shape:
Yellow Green Powder /Off-White Solid
Molecular weight:
202.17
Ref: TM-T21622
| 2mg | 38.00 € | ||
| 5mg | 55.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 117.00 € | ||
| 50mg | 173.00 € | ||
| 100mg | 246.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
EGFR-IN-11
CAS:2463200-44-2
EGFR-IN-11 selectively blocks EGFR-tyrosine kinase and promotes apoptosis; targets EGFRL858R/T790M/C797S, IC50=18 nM; halts cell cycle …
Formula:
C29H35N9O2S
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
573.71
Ref: TM-T11158
| 1mg | 85.00 € | ||
| 5mg | 182.00 € | ||
| 10mg | 313.00 € | ||
| 25mg | 496.00 € | ||
| 50mg | 686.00 € | ||
| 100mg | 911.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 236.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
SDZ281-977
CAS:150779-71-8
SDZ 281-977 is a derivative of Lavendustin A which is the EGF receptor tyrosine kinase …
Formula:
C18H20O5
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
316.35
Ref: TM-T16866
| 1mg | 97.00 € | ||
| 5mg | 231.00 € | ||
| 10mg | 369.00 € | ||
| 25mg | 739.00 € | ||
| 50mg | 1,146.00 € | ||
| 1mL*10mM (DMSO) | 257.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
EGFR-IN-99
CAS:2068806-31-3
EGFR-IN-99 (JBJ-03-142-02) is an EGFR and HER2 Exon 20 insertion mutation inhibitor for the study …
Formula:
C25H22FN7O3
Purity:
97.75%
Color and Shape:
Liquid
Molecular weight:
487.49
Ref: TM-T35901
| 1mg | 125.00 € | ||
| 5mg | 297.00 € | ||
| 10mg | 441.00 € | ||
| 25mg | 714.00 € | ||
| 50mg | 979.00 € | ||
| 100mg | 1,324.00 € | ||
| 500mg | 2,639.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Falnidamol
CAS:196612-93-8
Falnidamol (BIBX 1382), an oral selective EGFR inhibitor, IC50 3 nM, weak on ErbB2 and …
Formula:
C18H19ClFN7
Purity:
96.46%
Color and Shape:
Solid
Molecular weight:
387.84
Ref: TM-TQ0271
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 98.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 446.00 € | ||
| 200mg | 622.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Nimotuzumab
CAS:828933-51-3
Nimotuzumab is a humanized therapeutic monoclonal antibody against epidermal growth factor receptor EGFR).
Purity:
95.00%
Color and Shape:
Liquid
Ref: TM-T9923
| 1mg | 438.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
EGFR-IN-9
CAS:1226549-39-8
EGFR-IN-9 is a potent EGFR kinase inhibitor with IC50s of 7 nM, 28 nM for …
Formula:
C29H24N4O3
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
476.53
Ref: TM-T11163
| 1mg | 52.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 168.00 € | ||
| 25mg | 326.00 € | ||
| 50mg | 496.00 € | ||
| 1mL*10mM (DMSO) | 115.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
EGFR-IN-1 hydrochloride
CAS:2227455-78-7
EGFR-IN-1 HCl targets L858R/T790M EGFR mutants over wild-type; IC50: 4 nM in H1975, 28 nM …
Formula:
C28H31ClN6O4
Purity:
99.8%
Color and Shape:
Solid
Molecular weight:
551.04
Ref: TM-T11157L
| 1mg | 95.00 € | ||
| 5mg | 238.00 € | ||
| 10mg | 352.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 737.00 € | ||
| 100mg | 1,012.00 € | ||
| 500mg | 2,033.00 € | ||
| 1mL*10mM (DMSO) | 335.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
EGFR/ErbB-2 inhibitor-1
CAS:1135150-79-6
EGFR/ErbB-2 inhibitor-1 is a selective ErbB2/HER2 inhibitor that effectively blocks ErbB2 and HER2 signaling.
Formula:
C23H15ClFN3OS2
Purity:
97.55%
Color and Shape:
Liquid
Molecular weight:
467.97
Ref: TM-T79861
| 1mg | 182.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,004.00 € | ||
| 50mg | 1,385.00 € | ||
| 100mg | 1,831.00 € | ||
| 500mg | 3,652.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
PF-06459988
CAS:1428774-45-1
PF-06459988 is a novel, effective, orally active, irreversible, and selective epidermal growth factor receptor (EGFR) …
Formula:
C19H22ClN7O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
431.88
Ref: TM-T16492
| 1mg | 143.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
JGK-068S
CAS:2490431-16-6
Compound I (JGK-068S) is a potent inhibitor of the epidermal growth factor receptor (EGFR) [1].
Formula:
C22H23BrFN5O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
488.35
Ref: TM-T79124
| 5mg | 1,290.00 € | ||
| 50mg | 2,618.00 € | ||
| 100mg | 3,484.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Labuxtinib
CAS:1426449-01-5
Labutinib is a selective inhibitor of the c-kit tyrosine kinase [1].
Formula:
C20H16FN5O2
Purity:
99.77%
Color and Shape:
Liquid
Molecular weight:
377.37
Ref: TM-T79851
| 1mg | 138.00 € | ||
| 5mg | 333.00 € | ||
| 10mg | 533.00 € | ||
| 25mg | 1,059.00 € | ||
| 50mg | 1,523.00 € | ||
| 100mg | 2,046.00 € | ||
| 200mg | 2,763.00 € | ||
| 1mL*10mM (DMSO) | 369.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
YS-363
CAS:2470908-90-6
YS-363 is a potent, selective, and orally active inhibitor of the epidermal growth factor receptor …
Formula:
C30H30N4O3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
494.58
Ref: TM-T80748
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Feb 2025
DZD1516
CAS:2387570-00-3
DZD1516, a potent and selective HER2 inhibitor (IC50 = 0.56 nM), demonstrates good blood-brain barrier …
Formula:
C28H27F2N7O3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
547.56
Ref: TM-T79297
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
2′-Thioadenosine
CAS:136904-69-3
2'-Thioadenosine (PD157432) serves as a selective and irreversible inhibitor of ErbB-1 and ErbB-2 tyrosine kinases, …
Formula:
C10H13N5O3S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
283.31
Ref: TM-T78634
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Lifirafenib
CAS:1446090-79-4
Lifirafenib (Beigene-283) is a potent inhibitor of RAF family kinases and EGFR in biochemical assays …
Formula:
C25H17F3N4O3
Purity:
98% - 98.25%
Color and Shape:
Solid
Molecular weight:
478.42
Ref: TM-T22272
| 1mg | 35.00 € | ||
| 5mg | 68.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | To inquire | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
