EGFR
EGFR (epidermal growth factor receptor) inhibitors are compounds that block the signaling of EGFR, a receptor that is often overexpressed in various cancers and plays a critical role in angiogenesis. EGFR inhibitors are used to prevent tumor growth and metastasis by disrupting the pathways that promote blood vessel formation in tumors. These inhibitors are widely used in cancer research and therapy. At CymitQuimica, we offer a diverse selection of high-quality EGFR inhibitors to support your research in oncology and angiogenesis.
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Tucatinib
CAS:937263-43-9
Tucatinib (ONT-380) is a potent and selective HER2 inhibitor (IC50: 8 nM).
Formula:
C26H24N8O2
Purity:
99.05% - 99.96%
Color and Shape:
Solid
Molecular weight:
480.52
Ref: TM-T2364
| 1g | 1,110.00 € | ||
| 2mg | 40.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 127.00 € | ||
| 50mg | 189.00 € | ||
| 100mg | 343.00 € | ||
| 500mg | 812.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Methyl 2,5-dihydroxycinnamate
CAS:63177-57-1
Methyl 2,5-dihydroxycinnamate is an EGF receptor-associated tyrosine kinases inhibitor.
Formula:
C10H10O4
Purity:
98.98%
Color and Shape:
Crystalline
Molecular weight:
194.18
Ref: TM-T22974
| 5mg | 60.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 349.00 € | ||
| 100mg | 522.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
ZD-4190
CAS:413599-62-9
ZD-4190 blocks VEGFR2 and EGFR, aiding cancer treatment.
Formula:
C19H16BrFN6O2
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
459.27
Ref: TM-T5475
| 1mg | 82.00 € | ||
| 5mg | 177.00 € | ||
| 10mg | 266.00 € | ||
| 25mg | 422.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € | ||
| 1mL*10mM (DMSO) | 179.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Mutant EGFR inhibitor
CAS:1421373-62-7
Selective, potent inhibitor for mutated EGFR: L858R, Exon19 deletion, T790M resistance mutants.
Formula:
C27H30ClN7O2
Purity:
96.21% - 98%
Color and Shape:
Solid
Molecular weight:
520.03
Ref: TM-T2705
| 1mg | 36.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 258.00 € | ||
| 100mg | 371.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 104.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
HG-14-10-04
CAS:1356962-34-9
HG-14-10-04 is a potent and specific ALK inhibitor.
Formula:
C29H34ClN7O
Purity:
100% - 99.75%
Color and Shape:
Solid
Molecular weight:
532.08
Ref: TM-T4015
| 1mg | 59.00 € | ||
| 2mg | 87.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 194.00 € | ||
| 25mg | 274.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | 493.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
TX1-85-1
CAS:1603845-32-4
TX1-85-1: irreversible Her3 inhibitor (IC50: 23 nM), degrades Her3 protein, disrupts signaling, binds Cys721 covalently.
Formula:
C32H36N8O3
Purity:
98.12% - 98.12%
Color and Shape:
Solid
Molecular weight:
580.68
Ref: TM-T17182
| 1mg | 69.00 € | ||
| 5mg | 125.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 362.00 € | ||
| 50mg | 532.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Alflutinib
CAS:1869057-83-9
Alflutinib (ASK120067) is an inhibitor of EGFR, and its targets including EGFR activating mutations and …
Formula:
C28H31F3N8O2
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
568.59
Ref: TM-T22254
| 1mg | 210.00 € | ||
| 5mg | 428.00 € | ||
| 10mg | 610.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,295.00 € | ||
| 100mg | 1,755.00 € | ||
| 1mL*10mM (DMSO) | 556.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
(±)-Norcantharidin
CAS:29745-04-8
(±)-Norcantharidin (Endothall anhydride) is a synthetic anticancer compound which is a dual inhibitor for c-Met …
Formula:
C8H8O4
Purity:
99.43% - ≥98%
Color and Shape:
Solid
Molecular weight:
168.15
Ref: TM-T5656
| 1g | 530.00 € | ||
| 5mg | 44.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 77.00 € | ||
| 50mg | 103.00 € | ||
| 100mg | 151.00 € | ||
| 500mg | 357.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Saracatinib
CAS:379231-04-6
Saracatinib (AZD0530) (AZD0530) is an effective Src inhibitor (IC50: 2.7 nM), and effective to Lck, …
Formula:
C27H32ClN5O5
Purity:
98% - 99.63%
Color and Shape:
Solid
Molecular weight:
542.03
Ref: TM-T6078
| 10mg | 64.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 143.00 € | ||
| 100mg | 224.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
WS6
CAS:1421227-53-3
WS6, a β cell proliferation inducer, regulates Erb3 binding protein-1 (EBP1) and the IκB kinase …
Formula:
C29H31F3N6O3
Purity:
97.23% - 99.83%
Color and Shape:
Solid
Molecular weight:
568.59
Ref: TM-T2106
| 1mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 220.00 € | ||
| 100mg | 327.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Tuxobertinib
CAS:2414572-47-5
Tuxobertinib (BDTX-189) is a potent and selective inhibitor of allosteric EGFR and HER2 oncogenic mutations. …
Formula:
C29H29ClN6O4
Purity:
98.86%
Color and Shape:
Solid
Molecular weight:
561.03
Ref: TM-T9072
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 186.00 € | ||
| 50mg | 349.00 € | ||
| 100mg | 519.00 € | ||
| 200mg | 743.00 € | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Naquotinib
CAS:1448232-80-1
Naquotinib (ASP8273) (ASP8273) is an orally available, mutant-selective and irreversible EGFR inhibitor; (IC50s: 8-33 nM …
Formula:
C30H42N8O3
Purity:
97.49%
Color and Shape:
Solid
Molecular weight:
562.71
Ref: TM-TQ0092
| 1mg | 51.00 € | ||
| 2mg | 66.00 € | ||
| 5mg | 95.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 132.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Olafertinib
CAS:1660963-42-7
Olafertinib (RX-518) is a novel mutant-selective, irreversible, orally available EGFR inhibitor. It can overcome T790M-mediated …
Formula:
C29H28F2N6O2
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
530.57
Ref: TM-TQ0255
| 1mg | 48.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 299.00 € | ||
| 50mg | 441.00 € | ||
| 100mg | 644.00 € | ||
| 1mL*10mM (DMSO) | 111.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
AZD3759 hydrochloride
CAS:1626387-81-2
AZD3759 hydrochloride is an oral, CNS-penetrant EGFR inhibitor with IC50s of 0.2/0.3/0.2 nM.
Formula:
C22H24Cl2FN5O3
Purity:
99.41%
Color and Shape:
Solid
Molecular weight:
496.36
Ref: TM-T4249
| 2mg | 35.00 € | ||
| 5mg | 48.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 171.00 € | ||
| 100mg | 273.00 € | ||
| 200mg | 396.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
KI8751
CAS:228559-41-9
KI8751 is a potent and selective inhibitor of VEGFR2 with IC50 of 0.9 nM.
Formula:
C24H18F3N3O4
Purity:
99.73% - 99.9%
Color and Shape:
Solid
Molecular weight:
469.41
Ref: TM-T2446
| 2mg | 36.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 153.00 € | ||
| 50mg | 289.00 € | ||
| 100mg | 508.00 € | ||
| 200mg | 660.00 € | ||
| 500mg | 1,003.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
FIIN-3
CAS:1637735-84-2
FIIN-3 is an irreversible inhibitor of FGFR.
Formula:
C34H36Cl2N8O4
Purity:
97.63% - 98.92%
Color and Shape:
Solid
Molecular weight:
691.61
Ref: TM-T3466
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 244.00 € | ||
| 50mg | 360.00 € | ||
| 100mg | 513.00 € | ||
| 200mg | 699.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
WZ8040
CAS:1214265-57-2
WZ8040 is a novel mutant-selective irreversible EGFRT790M inhibitor, does not inhibit ERBB2 phosphorylation (T798I).
Formula:
C24H25ClN6OS
Purity:
97.42%
Color and Shape:
Solid
Molecular weight:
481.01
Ref: TM-T6734
| 1mg | 47.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 147.00 € | ||
| 25mg | 241.00 € | ||
| 50mg | 358.00 € | ||
| 100mg | 527.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
ZM39923 hydrochloride
CAS:1021868-92-7
ZM39923 hydrochloride (JAK3 Inhibitor IV) is an JAK1/3 inhibitor, almost no activity to JAK2 and …
Formula:
C23H25NO·HCl
Purity:
98.05%
Color and Shape:
Solid
Molecular weight:
367.91
Ref: TM-T6145
| 5mg | 58.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 304.00 € | ||
| 100mg | 455.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
SU5214
CAS:186611-04-1
SU5214 is a modulator of tyrosine kinase signal transduction.
Formula:
C16H13NO2
Purity:
99.52% - 99.55%
Color and Shape:
Solid
Molecular weight:
251.28
Ref: TM-T3569
| 5mg | 38.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 107.00 € | ||
| 50mg | 169.00 € | ||
| 100mg | 269.00 € | ||
| 200mg | 391.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Canertinib dihydrochloride
CAS:289499-45-2
Canertinib dihydrochloride (PD-183805 dihydrochloride) is the hydrochloride salt of an orally bio-available quinazoline with potential …
Formula:
C24H27Cl3FN5O3
Purity:
99.23%
Color and Shape:
Solid
Molecular weight:
558.86
Ref: TM-T2501
| 5mg | 38.00 € | ||
| 10mg | 52.00 € | ||
| 50mg | 74.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
