Serine/threonin kinase
Serine/threonine kinase inhibitors are compounds that target enzymes responsible for phosphorylating serine and threonine residues on proteins, which play a pivotal role in regulating apoptosis and other cellular processes. These kinases are involved in signaling pathways that control cell growth, division, and programmed cell death. Inhibiting specific serine/threonine kinases can alter the balance between cell survival and apoptosis, making these inhibitors essential tools in cancer research and other areas of cell biology. At CymitQuimica, we provide a comprehensive selection of high-quality serine/threonine kinase inhibitors to support your research in apoptosis, signal transduction, and disease mechanisms.
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![N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine](https://static.cymitquimica.com/products/TM/thumb/T9256.jpg)
N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine
CAS:1071135-06-2
Novel 2,6-naphthyridine inhibits PKC/PKD, identified by HTS.
Formula:
C23H28N6
Purity:
98.35%
Color and Shape:
Solid
Molecular weight:
388.51
Ref: TM-T9256
| 1mg | 143.00 € | ||
| 5mg | 312.00 € | ||
| 50mg | 1,053.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PKD-IN-1 dihydrochloride (956121-30-5 free base)
CAS:2308510-39-4
CRT0066101 dihydrochloride is an inhibitor of PKD.
Formula:
C18H21Cl3N4O
Purity:
99.50%
Color and Shape:
Solid
Molecular weight:
415.75
Ref: TM-T8957L
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 136.00 € | ||
| 50mg | 214.00 € | ||
| 100mg | 324.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
ML-7 hydrochloride
CAS:110448-33-4
ML-7 hydrochloride (ML-7 HCl) is a cell-permeable, reversible, effective, ATP-competitive, and specific inhibitor of myosin …
Formula:
C15H18ClIN2O2S
Purity:
99% - 99.61%
Color and Shape:
White Powder
Molecular weight:
452.74
Ref: TM-T3050
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 146.00 € | ||
| 50mg | 236.00 € | ||
| 100mg | 347.00 € | ||
| 200mg | 448.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
LP-935509
CAS:1454555-29-3
LP-935509 is a selective, brain-permeable, small molecule competitive inhibitor of articulin-2-associated kinase 1 (AAK1).Cost-effective and …
Formula:
C20H24N6O3
Purity:
98.82% - 99.64%
Color and Shape:
Solid
Molecular weight:
396.44
Ref: TM-T15781
| 1mg | 39.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 247.00 € | ||
| 50mg | 461.00 € | ||
| 100mg | 670.00 € | ||
| 1mL*10mM (DMSO) | 91.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PCSK9-IN-10
CAS:368434-98-4
PCSK9-IN-10: potent oral PCSK9 inhibitor (IC50 = 6.4 µM), upregulates LDLR, curbs atherosclerosis, for hyperlipidemia …
Formula:
C18H23N5O4
Purity:
98.85%
Color and Shape:
Soild
Molecular weight:
373.41
Ref: TM-T72025
| 1mg | 48.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 149.00 € | ||
| 25mg | 291.00 € | ||
| 50mg | 458.00 € | ||
| 100mg | 674.00 € | ||
| 500mg | 1,411.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
HA-1004
CAS:91742-10-8
HA-1004 is a inhibitor of PKG, PKA, PKC and MLC.
Formula:
C12H15N5O2S
Purity:
98.91% - 99.03%
Color and Shape:
Solid
Molecular weight:
293.34
Ref: TM-T27525
| 1mg | 183.00 € | ||
| 5mg | 406.00 € | ||
| 10mg | 600.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,281.00 € | ||
| 100mg | 1,726.00 € | ||
| 500mg | 3,468.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
SRPKIN-1
CAS:2089226-94-6
SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).
Formula:
C27H21FN2O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
472.53
Ref: TM-T16931
| 5mg | 1,062.00 € | ||
| 25mg | 1,787.00 € | ||
| 50mg | 2,160.00 € | ||
| 100mg | 2,813.00 € | ||
| 1mL*10mM (DMSO) | 1,170.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
BioE-1115
CAS:1268863-35-9
BioE-1115 is a selective and potent inhibitor of serine-threonine protein kinase (PASK, IC50 = 4 …
Formula:
C19H18FN3O2
Purity:
97.38%
Color and Shape:
Solid
Molecular weight:
339.36
Ref: TM-T10547
| 5mg | 35.00 € | ||
| 10mg | 46.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
HTH-01-091
CAS:2000209-42-5
HTH-01-091 is a potent and selective maternal embryonic leucine zipper kinase (MELK) inhibitor (IC50: 10.5 …
Formula:
C26H28Cl2N4O2
Purity:
98.40%
Color and Shape:
Solid
Molecular weight:
499.43
Ref: TM-T24152
| 1mg | 280.00 € | ||
| 5mg | 687.00 € | ||
| 10mg | 916.00 € | ||
| 25mg | 1,420.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,322.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
IPR-803
CAS:892243-35-5
IPR-803 is an effective inhibitor of the uPAR·uPA protein-protein interaction (PPI) with anti-tumor activity.
Formula:
C27H23N3O4
Purity:
95%
Color and Shape:
Solid
Molecular weight:
453.49
Ref: TM-T11666
| 1mg | 91.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 305.00 € | ||
| 25mg | 518.00 € | ||
| 50mg | 732.00 € | ||
| 1mL*10mM (DMSO) | 214.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
MS-444
CAS:150045-18-4
MS-444 (BE-34776) is an MLCK and HuR inhibitor with antitumor activity that can be used …
Formula:
C13H10O4
Purity:
99.45% - 99.45%
Color and Shape:
Solid
Molecular weight:
230.22
Ref: TM-T16145
| 1mg | 571.00 € | ||
| 2mg | 791.00 € | ||
| 25mg | 1,688.00 € | ||
| 50mg | 2,225.00 € | ||
| 100mg | 2,897.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
