
Serine/threonin kinase
Serine/threonine kinase inhibitors are compounds that target enzymes responsible for phosphorylating serine and threonine residues on proteins, which play a pivotal role in regulating apoptosis and other cellular processes. These kinases are involved in signaling pathways that control cell growth, division, and programmed cell death. Inhibiting specific serine/threonine kinases can alter the balance between cell survival and apoptosis, making these inhibitors essential tools in cancer research and other areas of cell biology. At CymitQuimica, we provide a comprehensive selection of high-quality serine/threonine kinase inhibitors to support your research in apoptosis, signal transduction, and disease mechanisms.
Found 15 products of "Serine/threonin kinase"
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BMT-124110 Formate
<p>BMT-124110 Formate is a selective AAK1 inhibitor (IC50: 0.9 nM) with anti-injury sensory activity.BMT-124110 Formate inhibits the BMP-2-inducible protein kinase</p>Formula:C22H20N2O2Purity:99.52%Color and Shape:SoildMolecular weight:344.41CID755673
CAS:<p>CID755673 inhibits PKD (IC50: 182 nM), with selectivity over PLK1, AKT, CAMKIIα, CAK, PKC.</p>Formula:C12H11NO3Purity:97.68% - 99.84%Color and Shape:SolidMolecular weight:217.221-Naphthyl PP1
CAS:<p>1-Naphthyl PP1 (1-NA-PP 1) is a selective src inhibitor(v-Src and c-Fyn, c-Abl, CDK2 and CAMK II with IC50s of 1.0, 0.6, 0.6, 18 and 22 μM, respectively)</p>Formula:C19H19N5Purity:99.85%Color and Shape:White Cyrstalline SolidMolecular weight:317.39PKD-IN-1
CAS:<p>CRT0066101 is an inhibitor of PKD.</p>Formula:C18H19ClN4OPurity:98%Color and Shape:SolidMolecular weight:342.82kb NB 142-70
CAS:<p>kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively).</p>Formula:C11H9NO2S2Purity:98.15% - ≥95%Color and Shape:SolidMolecular weight:251.321-NM-PP1
CAS:<p>1-NM-PP1 (PP1 Analog II) is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.</p>Formula:C20H21N5Purity:98% - 98.93%Color and Shape:White Cyrstalline SolidMolecular weight:331.41N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine
CAS:<p>Novel 2,6-naphthyridine inhibits PKC/PKD, identified by HTS.</p>Formula:C23H28N6Purity:98.35%Color and Shape:SolidMolecular weight:388.51ML-7 hydrochloride
CAS:<p>ML-7 hydrochloride (ML-7 HCl) is a cell-permeable, reversible, effective, ATP-competitive, and specific inhibitor of myosin light chain kinase (Ki: 300 nM);</p>Formula:C15H18ClIN2O2SPurity:99% - 99.26%Color and Shape:White PowderMolecular weight:452.74CID 2011756
CAS:<p>CID 2011756 is an ATP-competitive and specific PKD1 inhibitor.</p>Formula:C22H21ClN2O3Purity:98.15% - ≥95%Color and Shape:SolidMolecular weight:396.87Benzamidine hydrochloride
CAS:<p>Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin.</p>Formula:C7H9ClN2Purity:99.25% - 99.97%Color and Shape:White To Off-White PowderMolecular weight:156.61SPHINX31
CAS:<p>SPHINX31 is a potent inhibitor of serine/arginine-rich protein kinase 1 (SRPK1; IC50: 5.9 nM).</p>Formula:C27H24F3N5O2Purity:98.81% - 99.3%Color and Shape:SolidMolecular weight:507.51GAK inhibitor 49
CAS:<p>GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).</p>Formula:C20H22N2O5Purity:98.71%Color and Shape:SolidMolecular weight:370.4SGC-GAK-1
CAS:<p>SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).</p>Formula:C18H17BrN2O3Purity:99.85%Color and Shape:SolidMolecular weight:389.24SRPKIN-1
CAS:<p>SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).</p>Formula:C27H21FN2O3SPurity:98%Color and Shape:SolidMolecular weight:472.53MS-444
CAS:<p>MS-444 (BE-34776) is an MLCK and HuR inhibitor with antitumor activity that can be used to study triple-negative breast cancer and colorectal cancer.</p>Formula:C13H10O4Purity:99.45% - 99.45%Color and Shape:SolidMolecular weight:230.22
