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Serine/threonin kinase

Serine/threonin kinase

Serine/threonine kinase inhibitors are compounds that target enzymes responsible for phosphorylating serine and threonine residues on proteins, which play a pivotal role in regulating apoptosis and other cellular processes. These kinases are involved in signaling pathways that control cell growth, division, and programmed cell death. Inhibiting specific serine/threonine kinases can alter the balance between cell survival and apoptosis, making these inhibitors essential tools in cancer research and other areas of cell biology. At CymitQuimica, we provide a comprehensive selection of high-quality serine/threonine kinase inhibitors to support your research in apoptosis, signal transduction, and disease mechanisms.

Found 15 products of "Serine/threonin kinase"

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  • BMT-124110 Formate


    <p>BMT-124110 Formate is a selective AAK1 inhibitor (IC50: 0.9 nM) with anti-injury sensory activity.BMT-124110 Formate inhibits the BMP-2-inducible protein kinase</p>
    Formula:C22H20N2O2
    Purity:99.52%
    Color and Shape:Soild
    Molecular weight:344.41
  • CID755673

    CAS:
    <p>CID755673 inhibits PKD (IC50: 182 nM), with selectivity over PLK1, AKT, CAMKIIα, CAK, PKC.</p>
    Formula:C12H11NO3
    Purity:97.68% - 99.84%
    Color and Shape:Solid
    Molecular weight:217.22
  • 1-Naphthyl PP1

    CAS:
    <p>1-Naphthyl PP1 (1-NA-PP 1) is a selective src inhibitor(v-Src and c-Fyn, c-Abl, CDK2 and CAMK II with IC50s of 1.0, 0.6, 0.6, 18 and 22 μM, respectively)</p>
    Formula:C19H19N5
    Purity:99.85%
    Color and Shape:White Cyrstalline Solid
    Molecular weight:317.39
  • PKD-IN-1

    CAS:
    <p>CRT0066101 is an inhibitor of PKD.</p>
    Formula:C18H19ClN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:342.82
  • kb NB 142-70

    CAS:
    <p>kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively).</p>
    Formula:C11H9NO2S2
    Purity:98.15% - ≥95%
    Color and Shape:Solid
    Molecular weight:251.32
  • 1-NM-PP1

    CAS:
    <p>1-NM-PP1 (PP1 Analog II) is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.</p>
    Formula:C20H21N5
    Purity:98% - 98.93%
    Color and Shape:White Cyrstalline Solid
    Molecular weight:331.41
  • N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine

    CAS:
    <p>Novel 2,6-naphthyridine inhibits PKC/PKD, identified by HTS.</p>
    Formula:C23H28N6
    Purity:98.35%
    Color and Shape:Solid
    Molecular weight:388.51
  • ML-7 hydrochloride

    CAS:
    <p>ML-7 hydrochloride (ML-7 HCl) is a cell-permeable, reversible, effective, ATP-competitive, and specific inhibitor of myosin light chain kinase (Ki: 300 nM);</p>
    Formula:C15H18ClIN2O2S
    Purity:99% - 99.26%
    Color and Shape:White Powder
    Molecular weight:452.74
  • CID 2011756

    CAS:
    <p>CID 2011756 is an ATP-competitive and specific PKD1 inhibitor.</p>
    Formula:C22H21ClN2O3
    Purity:98.15% - ≥95%
    Color and Shape:Solid
    Molecular weight:396.87
  • Benzamidine hydrochloride

    CAS:
    <p>Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin.</p>
    Formula:C7H9ClN2
    Purity:99.25% - 99.97%
    Color and Shape:White To Off-White Powder
    Molecular weight:156.61
  • SPHINX31

    CAS:
    <p>SPHINX31 is a potent inhibitor of serine/arginine-rich protein kinase 1 (SRPK1; IC50: 5.9 nM).</p>
    Formula:C27H24F3N5O2
    Purity:98.81% - 99.3%
    Color and Shape:Solid
    Molecular weight:507.51
  • GAK inhibitor 49

    CAS:
    <p>GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).</p>
    Formula:C20H22N2O5
    Purity:98.71%
    Color and Shape:Solid
    Molecular weight:370.4
  • SGC-GAK-1

    CAS:
    <p>SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).</p>
    Formula:C18H17BrN2O3
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:389.24
  • SRPKIN-1

    CAS:
    <p>SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).</p>
    Formula:C27H21FN2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:472.53
  • MS-444

    CAS:
    <p>MS-444 (BE-34776) is an MLCK and HuR inhibitor with antitumor activity that can be used to study triple-negative breast cancer and colorectal cancer.</p>
    Formula:C13H10O4
    Purity:99.45% - 99.45%
    Color and Shape:Solid
    Molecular weight:230.22