Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
Subcategories of "Chromatin/Epigenetics"
Found 2612 products of "Chromatin/Epigenetics"
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AMPK activator 1
CAS:AMPK activator 1 is an AMPK activator(compound No.1-75, EC50: <0.1μM).Formula:C32H33F3N4O3Purity:98%Color and Shape:SolidMolecular weight:578.62NV03
CAS:NV03 is a selective antagonist of the UHRF1-H3K9me3 interaction (Kd=2.4 μM) for cancer research. a ligand for E3 ligases in PROTAC synthesis.Formula:C19H27N5O2SPurity:99.88%Color and Shape:SolidMolecular weight:389.52M122
CAS:M122 is a selective histone deacetylase HDAC1 and HDAC2 inhibitor and potent antitumor agent.Formula:C24H25N5OS2Color and Shape:SolidMolecular weight:463.62CTK7A
CAS:CTK7A is a water-soluble inhibitor of p300. CTK7A inhibits tumor growth in xenografted mice.Formula:C28H24N2NaO6Purity:98%Color and Shape:SolidMolecular weight:507.498HDAC6-IN-6
CAS:HDAC6-IN-6: Potent HDAC6 blocker, BBB-permeable, IC50: 0.025μM; inhibits AChE, Aβ 1-42 aggregation; promotes neurite growth, low neurotoxicity.Formula:C20H15N3O2Color and Shape:SolidMolecular weight:329.35MAT2A inhibitor 1
CAS:MAT2A inhibitor 1 is an inhibitor of methionine adenosyltransferase 2A (MATA2) (IC50 < l00 nM).Formula:C31H22N6OSColor and Shape:SolidMolecular weight:526.61HDAC-IN-5
CAS:HDAC-IN-5 is a histone deacetylase (HDAC) inhibitor.Formula:C26H24F3N5O2SPurity:98%Color and Shape:SolidMolecular weight:527.56CTPB
CAS:CTPB is a potent p300 histone acetyltransferase (HAT) activator that can be used in the preparation of hair growth promoters and/or hair loss treatments.Formula:C31H43ClF3NO2Purity:99.51%Color and Shape:SolidMolecular weight:554.13JAK3-IN-12
CAS:JAK3-IN-12 (compound 15k) is a potent inhibitor of JAK3 (IC50: 9.5 nM) and can be used in the study of rheumatoid arthritis.Formula:C19H19N5O4SColor and Shape:SolidMolecular weight:413.45SB-429201
CAS:SB-429201 is an effective, selective inhibitor of HDAC1.Formula:C28H24N2O3Purity:98%Color and Shape:SolidMolecular weight:436.5JAK3-IN-9
CAS:JAK3-IN-9, potent JAK3 inhibitor, IC50 of 1.7 nM, highly selective, low toxicity, orally bioavailable, shows anti-arthritis activity.Formula:C17H23N5O4SColor and Shape:SolidMolecular weight:393.46CPI-455 HCl
CAS:CPI-455: specific KDM5A inhibitor, IC50=10±1nM, increases H3K4me3, reduces DTPs in cancer cells.Formula:C16H15ClN4OPurity:98%Color and Shape:SolidMolecular weight:314.77LB-205
CAS:LB-205 is a Zn 2+ dependent pan-inhibitor of class I and class II HDACs. It also has a long half-life in vivo.Formula:C18H21N3O2SColor and Shape:SolidMolecular weight:343.44INCB16562
CAS:INCB16562: oral JAK1/2 inhibitor, halts IL-6/STAT3 in myeloma cells, boosts drug efficacy, stunts myeloma in mice.Formula:C19H11Cl2N5Color and Shape:SolidMolecular weight:380.23Guadecitabine
CAS:Guadecitabine is a second-generation DNA methyltransferases inhibitor. It is used for research on acute myeloid leukemia and myelodysplastic syndromes.Formula:C18H24N9O10PPurity:98%Color and Shape:SolidMolecular weight:557.41PB131
CAS:PB131, a selective and brain-permeable HDAC6 inhibitor, exhibits high binding affinity (IC50: 1.8 nM) and potent anti-inflammatory activity, making it suitableFormula:C16H16FN3O2Purity:98%Color and Shape:SolidMolecular weight:301.32ZL0454
CAS:ZL0454 is an effective and selective Bromodomain-containing protein 4 inhibitors (IC50: 49 and 32 nM for BD1 and BD2).Formula:C18H22N4O3SPurity:98%Color and Shape:SolidMolecular weight:374.46MPT0G211
CAS:MPT0G211: oral HDAC6 inhibitor with IC50=0.291 nM, 1000x selectivity, neuroprotective, anti-metastatic, crosses blood-brain barrier for Alzheimer's.Formula:C17H15N3O2Purity:99.93% - 99.98%Color and Shape:SolidMolecular weight:293.32Ref: TM-T60616
1mg92.00€5mg222.00€10mg356.00€25mg560.00€50mg782.00€100mg1,063.00€200mg1,459.00€1mL*10mM (DMSO)245.00€Bromodomain inhibitor-8
CAS:Bromodomain inhibitor-8 is an inhibitor of BET bromodomain used to treat autoimmune and inflammatory diseases.Formula:C26H25ClN2O3Color and Shape:SolidMolecular weight:448.94Exifone
CAS:Exifone (NSC-680919) is a mixed, nonessential activator of HDAC1 that is capable of binding to both free and substrate-bound enzyme, resulting in an increasedFormula:C13H10O7Purity:99.77% - 99.95%Color and Shape:Yellow SolidMolecular weight:278.21Bromodomain inhibitor-9
CAS:Bromodomain inhibitor-9 selectively targets BRD4-1 (Kd 12 nM), used in metabolic, inflammatory, fibrotic, and autoimmune disease studies.Formula:C24H28N4O5SColor and Shape:SolidMolecular weight:484.571,2,3,4,5,6-Hexabromocyclohexane
CAS:Inhibits JAK2 autophosphorylation; non-cytotoxic at 100μM; 1μM reduces activity by 50%, 50μM nearly abolishes it.Formula:C6H6Br6Purity:98%Color and Shape:SolidMolecular weight:557.54Tankyrase-IN-2
CAS:Tankyrase-IN-2 is a selective, potent and orally active inhibitor of tankyrase with IC50s of 10, 7, and 710 nM for TNKS1, TNKS2 as well as PARP1, respectivelyFormula:C17H14F2N2O2Purity:98%Color and Shape:SolidMolecular weight:316.36(5H)-Phenanthridinone
CAS:6(5H)-Phenanthridinone suppresses PARP1/2, reduces RDM4 cell growth, downregulates pro-inflammatory genes, and alleviates EAE symptoms in rats.Formula:C13H9NOColor and Shape:SolidMolecular weight:195.22NCC-149
CAS:NCC-149 is a HDAC8 inhibitor.Formula:C16H14N4O2SColor and Shape:SolidMolecular weight:326.37MS-1020
CAS:MS-1020 inhibits JAK3/STAT3, blocks active JAK3, suppresses JAK3/STAT5 signaling, and targets STAT3 in certain cells.Formula:C21H18N2O3Purity:98%Color and Shape:SolidMolecular weight:346.38AC-93253 iodide
CAS:AC-93253 iodide is a selective inhibitor of SIRT2. It significantly enhances the acetylation of tubulin p53 and histone H4.Formula:C23H25IN2SPurity:98%Color and Shape:SolidMolecular weight:488.43GNE-272
CAS:GNE-272 is a selective inhibitor of CBP/EP300 (IC50: 0.02, 0.03, and 13 μM for CBP, EP300, and BRD4, respectively) and a selective in vivo probe for CBP/EP300.Formula:C22H25FN6O2Color and Shape:SolidMolecular weight:424.47Ac-Lys-AMC
CAS:Ac-Lys-AMC (Hexanamide) is a fluorescent substrate for histone deacetylase HDACs.Formula:C18H23N3O4Purity:98%Color and Shape:SolidMolecular weight:345.39PS315
CAS:PS315, a PS48 derivative, allosterically inhibits PKCζ/η (IC50: 10/30 μM), targeting aPKC's PIF-pocket, with anti-cancer properties.Formula:C23H19ClO2Purity:98%Color and Shape:SolidMolecular weight:362.85ZYJ-34v
CAS:ZYJ-34v is an oral histone deacetylase inhibitor (HDACi) with potent antitumor activities.Formula:C27H35N3O6Purity:98%Color and Shape:SolidMolecular weight:497.58SD-1029
CAS:SD-1029 is a JAK2 inhibitor and a novel Stat3 activation inhibitor that inhibits Stat3 phosphorylation and JAK-STAT signaling.Formula:C25H32Br2Cl2N2O3Color and Shape:SolidMolecular weight:639.25Jaspamycin
CAS:Jaspamycin (7-CN-7-C-Ino) does not bind with purified human PKARIα.Formula:C12H12N4O5Color and Shape:SolidMolecular weight:292.25(R)-UT-155
CAS:(R)-UT-155 is a selective androgen receptor degrader (SARD) ligand.Formula:C20H15F4N3O2Color and Shape:SolidMolecular weight:405.35ARTD10/PARP10-IN-1
CAS:ARTD10/PARP10-IN-1 is a PARP inhibitor that inhibits ARTD8/PARP14 and has anticancer and antitumour activity for the study of prostate cancer.Formula:C12H12N2O4Purity:99.14%Color and Shape:SolidMolecular weight:248.233-Deazaneplanocin A
CAS:3-Deazaneplanocin A (DZNep) is an EZH2 and AHCY inhibitor with antipoxigenic activity that inhibits fibrosis in the liver, kidneys, peritoneum, and airways.Formula:C12H14N4O3Purity:99.03% - 99.68%Color and Shape:SolidMolecular weight:262.27GS-626510
CAS:GS-626510 is an orally bioavailable inhibitor of BET family bromodomains (Kd: 0.59-3.2 nM for BRD2/3/4; IC50: 83 nM and 78 nM for BD1 and BD2).Formula:C25H22N4OColor and Shape:SolidMolecular weight:394.47AMPK activator
CAS:AMPK activatorFormula:C22H21FO4Purity:98%Color and Shape:SolidMolecular weight:368.4LW479
CAS:LW479 is a novel inhibitor of HDAC and is a promising candidate for the prevention of breast cancer.Formula:C21H23BrN2O4SColor and Shape:SolidMolecular weight:479.39KDM5A-IN-1
CAS:KDM5A-IN-1 is a pan-histidine lysine demethylase 5 KDM5 inhibitor that inhibits KDM5A, KDM5B, and KDM5C.Can be used in the study of cancer.Formula:C15H22N4O2Purity:>99.99%Color and Shape:SolidMolecular weight:290.36DC_517
CAS:DC_517 is an inhibitor of DNA methyltransferase 1 (DNMT1) ( IC50: 1.7 μM; Kd: 0.91 μM).Formula:C33H35N3O2Color and Shape:SolidMolecular weight:505.65Sirt2-IN-1
CAS:Sirt2-IN-1 is an inhibitor of sirtuin 2 (IC50 = 163 nM).Formula:C28H27N7O2S2Purity:99.57% - 99.84%Color and Shape:SolidMolecular weight:557.69Ref: TM-T12920
1mg100.00€5mg203.00€10mg323.00€25mg513.00€50mg697.00€100mg888.00€500mg1,783.00€1mL*10mM (DMSO)253.00€L 888607 Racemate
CAS:L 888607 Racemate blocks DP1 and TP receptors with 132 nM and 17 nM affinity.Formula:C19H15ClFNO2SColor and Shape:SolidMolecular weight:375.84Ilorasertib hydrochloride
CAS:Ilorasertib hydrochloride (ABT-348 hydrochloride) is an ATP-competitive multitargeted kinase inhibitor, which inhibits Aurora C, Aurora B, and Aurora A (IC50s:Formula:C25H22ClFN6O2SPurity:98.45%Color and Shape:SolidMolecular weight:525Tetrahydrouridine
CAS:Tetrahydrouridine (NSC-112907; THU) is a multidrug resistance modulator.Formula:C9H16N2O6Purity:98%Color and Shape:SolidMolecular weight:248.23ITF3756
CAS:ITF3756 is a selective HDAC6 inhibitor.Formula:C13H11N5O2SPurity:97.74%Color and Shape:SolidMolecular weight:301.32Tyk2-IN-7
CAS:Tyk2-IN-7 is an inhibitor of TYK2 JH2, binds to the TYK2 JH2 domain (IC50: 0.00053 μM; Ki.app: 0.00007 μM).Formula:C18H15D3N6O3SPurity:98%Color and Shape:SolidMolecular weight:401.46Givinostat hydrochloride monohydrate
CAS:Givinostat hydrochloride monohydrate (ITF2357) is an HDAC inhibitor.Formula:C24H27N3O4·HCl·H2OPurity:97.97% - 99.51%Color and Shape:SolidMolecular weight:475.97Pulrodemstat Methylbenzenesulfonate
CAS:LSD1-IN-7 Methylbenzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.Formula:C31H31F2N5O5SPurity:98%Color and Shape:SolidMolecular weight:623.67HDAC3-IN-T247
CAS:HDAC3-IN-T247 (HDAC3 inhibitor T247) is a histone deacetylase 3 (HDAC3) inhibitor with antiviral activity that inhibits the proliferation of cancer cells.Formula:C21H19N5OSPurity:98.11% - 98.94%Color and Shape:SolidMolecular weight:389.47Ref: TM-T24131
1mg87.00€5mg178.00€10mg295.00€25mg610.00€50mg867.00€100mg1,153.00€1mL*10mM (DMSO)203.00€YM-53601 free base
CAS:YM-53601 free base is an inhibitor of squalene synthetase which suppresses lipogenic biosynthesis and lipid secretion in rodents.Formula:C21H21FN2OPurity:98%Color and Shape:SolidMolecular weight:336.4EP009
CAS:EP009, a novel, selective, and orally active inhibitor of JAK3, induces therapeutic response in T-cell malignancies.Formula:C14H24O2Color and Shape:SolidMolecular weight:224.34MDK8228
CAS:MDK8228 is an inhibitor of CBP/p300 and BRD4 bromodomain. MDK8228 downregulates IL-6, IL-ß and IFN-ß in macrophages.Formula:C31H41N5O3Color and Shape:SolidMolecular weight:531.69AJH-836
CAS:AJH-836 is a compound that activates Munc13-1 and PKC ε/α, demonstrating a dissociation constant (Kd) of 4.5 nM for PKCα, and facilitates the translocation ofFormula:C22H38O5Purity:98%Color and Shape:SolidMolecular weight:382.53SIRT2-IN-9
CAS:SIRT2-IN-9: selective SIRT2 inhibitor; IC50=1.3μM; halts MCF-7 cell growth; for cancer study.Formula:C21H22N6OS2Purity:97.6%Color and Shape:SolidMolecular weight:438.57RM65
CAS:RM65 is an arginine methyltransferase inhibitor.Formula:C34H32N2O4S2Purity:98%Color and Shape:SolidMolecular weight:596.76HDAC-IN-58
CAS:HDAC-IN-58, a selective HDAC6 inhibitor, exhibits potent inhibitory activity with an IC50 of 2.06 nM, rendering it suitable for research into chronicFormula:C16H13ClF2N4O3SPurity:98%Color and Shape:SolidMolecular weight:414.81JAK-IN-21
CAS:JAK-IN-21 is a selective and potent JAK inhibitor that inhibits JAK1, JAK2, J2V617F and TYK2 with IC50 values of 1.73, 2.04, 109 and 62.9 nM, respectively.Formula:C19H16N8OPurity:99.87%Color and Shape:SolidMolecular weight:372.38JAK-IN-14
CAS:JAK-IN-14 (compound 16) is a specific JAK1 inhibitor. It prevents JAK1 phosphorylation by binding to the active site of JAK in immune, inflammation and cancer.Formula:C19H15FN4OPurity:98.27%Color and Shape:SolidMolecular weight:334.35Ref: TM-T9764
1mg81.00€5mg170.00€10mg268.00€25mg555.00€50mg888.00€100mg1,414.00€200mg1,882.00€1mL*10mM (DMSO)178.00€LSD1-IN-6
CAS:LSD1-IN-6, a potent LSD1 inhibitor (IC50: 123 nM), enhances H3K4me2 without altering LSD1 expression. Reversible.Formula:C15H13BrN2O3Purity:98%Color and Shape:SolidMolecular weight:349.18IDO1 and HDAC1 Inhibitor
CAS:IDO1 and HDAC1 Inhibitor is a dual IDO1 and HDAC1 inhibitor (IC50s: 69.0 nM and 66.5 nM).Formula:C25H22BrFN8O4Purity:98%Color and Shape:SolidMolecular weight:597.4HDAC-IN-49
HDAC-IN-49: potent, broad HDAC inhibitor; IC50s: 10-1880 nM for HDAC1-6; strong anti-leukemic, low toxicity to healthy cells.Formula:C26H27FN4O4Color and Shape:SolidMolecular weight:478.52Sirt1/2-IN-1
CAS:Sirt1/2-IN-1 inhibits SIRT1 (IC50: 1.81 μg/mL) and SIRT2 (2.10 μg/mL), less on SIRT3 (20.5 μg/mL), with anticancer properties.Formula:C22H13ClN2OS2Color and Shape:SolidMolecular weight:420.93PIM-1 Inhibitor 2
CAS:PIM-1 Inhibitor 2 (PIM1-IN-2) is a potent Pim-1 inhibitor with potential anti-cancer activity, used in cancer research.Formula:C17H11ClN4OPurity:98.81%Color and Shape:SolidMolecular weight:322.752′-Deoxy-5-nitrocytidine
CAS:2′-Deoxy-5-nitrocytidine is a DNA Methyltransferase inhibitor that can be used for cancer research[1].Formula:C9H12N4O6Color and Shape:SolidMolecular weight:272.21SB-284851-BT
CAS:SB-284851-BT: BRD4/p38α/BRDT inhibitor; IC50: BRD4-BD1 1.7µM, BRDT 18µM, BRD4 3.7µM; Kd p38α 0.47nM; reduces IL-8, affects c-Myc/NF-κB.Formula:C26H26FN5OColor and Shape:SolidMolecular weight:443.52PKC-IN-4
CAS:PKC-IN-4 (compound 7l) is a highly potent and orally active inhibitor of atypical protein kinase C (aPKC), exhibiting an IC 50 value of 0.52 μM.Formula:C21H25N5SColor and Shape:SolidMolecular weight:379.52CD161
CAS:CD161: powerful, selective oral BET inhibitor; IC50: 28.2 nM (BRD4 BD1), 7.2 nM (BRD4 BD2); strong anticancer properties.Formula:C26H21N5O2Purity:98%Color and Shape:SolidMolecular weight:435.48YF479
CAS:YF479 is an inhibitor of histone deacetylase that acts by inhibiting breast tumor growth, metastasis, and recurrence.Formula:C22H27BrN2O5Purity:98%Color and Shape:SolidMolecular weight:479.36DC-CPin7
CAS:DC-CPin7, a powerful inhibitor of the bromodomain of CREB-binding protein (CBP), exhibits an IC50 value of 2.5 μM [1].Formula:C19H22N2O5Color and Shape:SolidMolecular weight:358.39OICR-0547
CAS:OICR-0547 is an inactive derivative of OICR-9429 and is commonly used as a negative control for OICR-9429.Formula:C28H29F3N4O4Purity:98%Color and Shape:SolidMolecular weight:542.55HIF-1α inhibitor-1
CAS:HIF-1α inhibitor-1 is a HIF-1 alpha inhibitor.Formula:C15H11N3O4Color and Shape:SolidMolecular weight:297.27SMYD2-IN-1
CAS:SMYD2-IN-1 is an inhibitor of SMYD2 (IC50 of 4.45 nM).Formula:C25H25Cl2F2N7O2Purity:98%Color and Shape:SolidMolecular weight:564.41Bisindolylmaleimide II
CAS:protein kinase C (PKC) inhibitorFormula:C27H26N4O2Purity:98%Color and Shape:SolidMolecular weight:438.52LSD1-IN-12
CAS:LSD1-IN-12 (compound 2) is an effective inhibitor of LSD1, demonstrating inhibitory Ki values of 1.1 μM (LSD1), 61 μM (LSD2), 2.3 μM (MAO-A), and 3.5 μM (MAO-BFormula:C16H16N2OColor and Shape:SolidMolecular weight:252.31SRTCX1002
CAS:SRTCX1002 is a SIRT1 Activator Suppressing Inflammatory Responses through Promotion of p65 Deacetylation and NF-κB Activity inhibitor.Formula:C21H19N5O2SPurity:98%Color and Shape:SolidMolecular weight:405.47PU141
CAS:PU141 is a novel inhibitor of histone acetyltransferase (HAT).Formula:C14H9F3N2OSPurity:98%Color and Shape:SolidMolecular weight:310.29CHIC35
CAS:CHIC-35 is a selective deacetylase SIRT1 inhibitor.Formula:C14H15ClN2OColor and Shape:SolidMolecular weight:262.73OTS186935 trihydrochloride
CAS:OTS186935 trihydrochloride is a protein methyltransferase inhibitor of SUV39H2(IC50 of 6.49 nM).Formula:C25H29Cl4N5O2Purity:98%Color and Shape:SolidMolecular weight:573.34HDAC-IN-45
CAS:HDAC-IN-45, a small HDAC blocker, forms H-bonds with Y303 and shows anticancer properties; IC50 for HDAC1/2/3: 0.108/0.585/0.563 μM.Formula:C25H20ClFN8OColor and Shape:SolidMolecular weight:502.93dBRD9-A
CAS:Potent BRD9 degrader that binds selectively, fully degrades BRD9 at low doses, and hinders synovial sarcoma growth in vitro and in mice.Formula:C42H49N7O8Color and Shape:SolidMolecular weight:779.88ET-JQ1-OH
CAS:ET-JQ1-OH is an allele-specific BET inhibitor.Formula:C21H21ClN4O2SColor and Shape:SolidMolecular weight:428.93Y02224
CAS:Y02224 is a BET inhibitor. It shows the reasonable antiproliferative effect on leukemia cells.Formula:C20H17BrN2O4SPurity:98%Color and Shape:SolidMolecular weight:461.33PB118
PB118 clears Aβ, boosts phagocytosis, enhances tubulin networks, reduces p-tau & inflammation in AD; HDAC6 IC50: 5.6 nM.Formula:C18H19FN2O2Color and Shape:SoildMolecular weight:314.35HDAC3-IN-T326
CAS:HDAC3-IN-T326: potent, selective HDAC3 inhibitor, boosts NF-κB acetylation, activates latent HIV gene expression.Formula:C21H18N6O3SPurity:98%Color and Shape:SolidMolecular weight:434.47Dot1L-IN-5
CAS:Dot1L-IN-5 is a potent inhibitor of the disruptor of telomeric silencing 1-like protein ( DOT1L ) with an IC 50 SPA DOT1L of 0.17 nM [1].Formula:C23H19ClF2N8O5SColor and Shape:SolidMolecular weight:592.96Helenalin Acetate
CAS:Helenalin Acetate: anti-inflammatory, anti-cancer, hinders C/EBPß and p300 cooperation.Formula:C17H20O5Purity:98%Color and Shape:SolidMolecular weight:304.34PS432
CAS:PS432 inhibits atypical PKCs, targets PIF-pocket, reduces tumors in mice sans side effects.Formula:C25H19ClN2O5SPurity:98%Color and Shape:SolidMolecular weight:494.95DM-01
CAS:DM-01 is a potent and selective inhibitor of EZH2.Formula:C23H24F3N3O2Color and Shape:SolidMolecular weight:431.45Kgp-IN-1
CAS:Kgp-IN-1 is an arginine-specific gingipain (Rgp) inhibitor.Formula:C19H24F4N4O3Purity:98%Color and Shape:SolidMolecular weight:432.41(1S,2R)-Tranylcypromine hydrochloride
CAS:(1S,2R)-Tranylcypromine hydrochloride ((1S,2R)-SKF 385), a potent antidepressant, functions by inhibiting both MAO and LSD1.Formula:C9H12ClNColor and Shape:SolidMolecular weight:169.651Gue1654
CAS:Gue1654 is an OXE-R inhibitor and cardiomyocyte apoptosis.Gue1654 can be used for the study of cardiovascular diseases.Formula:C23H17N3OS3Purity:98.02% - 98.04%Color and Shape:SolidMolecular weight:447.6CID-4785700
CAS:CID-4785700 is a potent pan-GTPase inhibitor that inhibits Rab7 and inhibits the fungal histone acetyltransferase Rtt109 that binds to Asf1 and Vps75Formula:C22H23ClFN3O3Purity:98.16%Color and Shape:SolidMolecular weight:431.89Ref: TM-T71740
1mg315.00€5mg873.00€10mg1,080.00€25mg1,431.00€50mg1,783.00€100mg2,250.00€500mg4,419.00€PARP-1/2-IN-1
CAS:PARP-1-/2-IN-1 is a potent inhibitor of PARP-1 (IC50: 0.51 nM) and PARP-2 (IC50: 23.11 nM).Formula:C24H27FN4O3Color and Shape:SolidMolecular weight:438.49Akt Inhibitor X
CAS:Akt Inhibitor X is a cell-permeable and reversible inhibitor of Akt phosphorylation.Formula:C20H25ClN2OPurity:98%Color and Shape:SolidMolecular weight:344.88Resminostat
CAS:Resminostat (4SC-201) is an orally bioavailable inhibitor of histone deacetylases (HDACs) with potential antineoplastic activity.Formula:C16H19N3O4SPurity:99.46%Color and Shape:SolidMolecular weight:349.4NSC-636819
CAS:NSC-636819 is a novel inhibitor of KDM4A/KDM4B.Formula:C22H12Cl4N2O4Purity:98%Color and Shape:SolidMolecular weight:510.15PNZ5
CAS:PNZ5, an isoxazole-based pan-BET inhibitor, demonstrates potent activity and high selectivity comparable to the established (+)-JQ1, exhibiting a dissociationFormula:C20H18N2O2Purity:99.51% - 99.61%Color and Shape:SolidMolecular weight:318.37Ref: TM-T12513
1mg109.00€5mg243.00€10mg355.00€25mg532.00€50mg750.00€100mg1,009.00€200mg1,369.00€1mL*10mM (DMSO)240.00€JAK-IN-10
CAS:JAK-IN-10 is a JAK inhibitor. JAK-IN-10 can be used for the research of dry eye disorders.Formula:C20H18FN5O3SPurity:99.53%Color and Shape:SolidMolecular weight:427.45Ref: TM-T13571
1mg82.00€5mg167.00€10mg246.00€25mg405.00€50mg572.00€100mg772.00€500mg1,539.00€1mL*10mM (DMSO)178.00€SW155246
CAS:SW155246 is a potent and selective inhibitor of DNMT1 (DNA methyltransferase 1; IC50 of 1.2 μM).Formula:C16H11ClN2O5SPurity:98.99%Color and Shape:SolidMolecular weight:378.79
