Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
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Subcategories of "Chromatin/Epigenetics"
Products of "Chromatin/Epigenetics"
BI-9564
CAS:1883429-22-8
BI-9564, a specific cell-permeable BRD9 BD inhibitor. The Kd for BRD9 is 5.9 nM, and …
Formula:
C20H23N3O3
Purity:
98.77%
Color and Shape:
Solid
Molecular weight:
353.41
Ref: TM-T6786
| 5mg | 51.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 175.00 € | ||
| 50mg | 333.00 € | ||
| 100mg | 490.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
CEP-33779
CAS:1257704-57-6
CEP-33779 is a novel and selective inhibitor of JAK2 with an IC50 of 1.8±0.6 nM.
Formula:
C24H26N6O2S
Purity:
98.81% - ≥95%
Color and Shape:
Solid
Molecular weight:
462.57
Ref: TM-T6122
| 1mg | 45.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 241.00 € | ||
| 50mg | 372.00 € | ||
| 100mg | 553.00 € | ||
| 500mg | 1,194.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
UNC926
CAS:1184136-10-4
UNC926 inhibits L3MBTL1 (IC50: 3.9 μM), has affinity for L3MBTL3, blocks 3xMBT-H4K20me1 interactions, doesn't affect …
Formula:
C16H21BrN2O
Purity:
96.97%
Color and Shape:
Solid
Molecular weight:
337.25
Ref: TM-T4012
| 2mg | 37.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 261.00 € | ||
| 100mg | 421.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Baricitinib phosphate
CAS:1187595-84-1
Baricitinib phosphate (INCB028050) is a selective orally bioavailable JAK1/JAK2 inhibitor.
Formula:
C16H20N7O6PS
Purity:
98.87% - 99.68%
Color and Shape:
Solid
Molecular weight:
469.41
Ref: TM-T2360
| 5mg | 47.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 91.00 € | ||
| 50mg | 113.00 € | ||
| 100mg | 142.00 € | ||
| 500mg | 343.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Gandotinib
CAS:1229236-86-5
LY2784544(Gandotinib (LY2784544)) is a potent JAK2 inhibitor (IC50: 3 nM), effective in JAK2V617F(Ki: 0.245 nM).
Formula:
C23H25ClFN7O
Purity:
99.16% - 99.86%
Color and Shape:
Solid
Molecular weight:
469.94
Ref: TM-T2638
| 5mg | 51.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 290.00 € | ||
| 100mg | 460.00 € | ||
| 500mg | 1,012.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
ML367
CAS:381168-77-0
ML367 inhibits ATAD5 stabilization with low micromolar activity, serving as a probe molecule.
Formula:
C19H12F2N4
Purity:
99.39%
Color and Shape:
Solid
Molecular weight:
334.32
Ref: TM-T5425
| 5mg | 47.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 184.00 € | ||
| 100mg | 304.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
BYK204165
CAS:1104546-89-5
BYK204165 (RT-017290) is a potent PARP inhibitor (PARP1; IC50 = 44.67 nM for human recombinant …
Formula:
C15H12N2O2
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
252.27
Ref: TM-T7896
| 1mg | 46.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 198.00 € | ||
| 50mg | 297.00 € | ||
| 100mg | 442.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
XAV-939
CAS:284028-89-3
XAV-939 (NVP-XAV939) shows the selective inhibition against Wnt/β-catenin-mediated transcription by tankyrase1/2 inhibition (IC50: 11/4 nM …
Formula:
C14H11F3N2OS
Purity:
97.47% - 99.04%
Color and Shape:
Solid
Molecular weight:
312.31
Ref: TM-T1878
| 5mg | 57.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 113.00 € | ||
| 50mg | 172.00 € | ||
| 100mg | 262.00 € | ||
| 200mg | 460.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Reversine
CAS:656820-32-5
Reversine, a small synthetic purine analogue (2, 6-disubstituted purine), is a potent inhibitior of Aurora …
Formula:
C21H27N7O
Purity:
98% - 99.75%
Color and Shape:
Solid
Molecular weight:
393.49
Ref: TM-T1825
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 161.00 € | ||
| 50mg | 219.00 € | ||
| 100mg | 384.00 € | ||
| 1mL*10mM (DMSO) | 70.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
MRTX-1719
CAS:2630904-45-7
MRTX-1719 is a potent and selective inhibitor of the PRMT5/MTA complex with an IC50 value …
Formula:
C23H18ClFN6O2
Purity:
98.27% - 99.18%
Color and Shape:
Solid
Molecular weight:
464.88
Ref: TM-T40254
| 1mg | 369.00 € | ||
| 5mg | 720.00 € | ||
| 10mg | 979.00 € | ||
| 25mg | 1,636.00 € | ||
| 50mg | 2,292.00 € | ||
| 100mg | 3,347.00 € | ||
| 1mL*10mM (DMSO) | 739.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
I-BRD9
CAS:1714146-59-4
I-BRD9 (GSK602) is the first selective cellular inhibitor for BRD9 with pIC50 of 7.3.
Formula:
C22H22F3N3O3S2
Purity:
98.16% - 99.28%
Color and Shape:
Solid
Molecular weight:
497.55
Ref: TM-T6859
| 1mg | 40.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 211.00 € | ||
| 50mg | 402.00 € | ||
| 100mg | 598.00 € | ||
| 1mL*10mM (DMSO) | 83.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Filgotinib
CAS:1206161-97-8
Filgotinib (GLPG0634) is a selective JAK1 inhibitor. The IC50 values against JAK1, JAK2, JAK3, and …
Formula:
C21H23N5O3S
Purity:
98.03% - ≥95%
Color and Shape:
Solid
Molecular weight:
425.5
Ref: TM-T1929
| 1mg | 38.00 € | ||
| 5mg | 77.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 161.00 € | ||
| 50mg | 241.00 € | ||
| 100mg | 318.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
UNC0642
CAS:1481677-78-4
UNC0642 is an effective and specific G9a/GLP inhibitor (IC50< 2.5 nM).
Formula:
C29H44F2N6O2
Purity:
98.75% - 99.5%
Color and Shape:
Solid
Molecular weight:
546.7
Ref: TM-T4166
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 226.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 557.00 € | ||
| 200mg | 806.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
TP0463518
CAS:1558021-37-6
TP-0463518 is a highly potent HIF prolyl hydroxylase (PHD) inhibitor (IC50s: 13 nM and 18 …
Formula:
C20H18ClN3O6
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
431.83
Ref: TM-T5392
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 118.00 € | ||
| 50mg | 184.00 € | ||
| 100mg | 348.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Rucaparib
CAS:283173-50-2
Rucaparib (PF-01367338) is a orally PARP inhibitor and a H6PD inhibitor. Rucaparib exhibits antitumor activity …
Formula:
C19H18FN3O
Purity:
98.37% - 99.89%
Color and Shape:
Solid
Molecular weight:
323.36
Ref: TM-T4463
| 2mg | 48.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 231.00 € | ||
| 100mg | 356.00 € | ||
| 200mg | 528.00 € | ||
| 500mg | 850.00 € | ||
| 1mL*10mM (DMSO) | 81.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
FG-2216
CAS:223387-75-5
FG-2216 (YM-311) is a HIF-prolyl hydroxylase inhibitor for the PDH2 enzyme; orally bioavailable and induced …
Formula:
C12H9ClN2O4
Purity:
100% - 99%
Color and Shape:
Solid
Molecular weight:
280.66
Ref: TM-T2445
| 2mg | 39.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 245.00 € | ||
| 100mg | 363.00 € | ||
| 500mg | 857.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
4'-Methoxychalcone
CAS:959-23-9
4'-Methoxychalcone with a variety of pharmacological activities, such as anti-tumor and anti-inflammatory activities.
Formula:
C16H14O2
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
238.28
Ref: TM-T7443
| 50mg | 50.00 € | ||
| 100mg | 72.00 € | ||
| 500mg | 161.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
PF 477736
CAS:952021-60-2
PF 477736 (PF-736,PF-00477736) is a specifc, effective and ATP-competitive Chk1 inhibitor (Ki: 0.49 nM ) …
Formula:
C22H25N7O2
Purity:
98% - 98.34%
Color and Shape:
Solid
Molecular weight:
419.48
Ref: TM-T6028
| 2mg | 49.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Senaparib
CAS:1401682-78-7
Senaparib (IMP4297) is a novel highly potent and selective oral PARP1/2 inhibitor with strong antitumor …
Formula:
C24H20F2N6O3
Purity:
99.41%
Color and Shape:
Solid
Molecular weight:
478.45
Ref: TM-T9593
| 1mg | 45.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 425.00 € | ||
| 100mg | 624.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Ritlecitinib
CAS:1792180-81-4
Ritlecitinib (PF-06651600) is an orally available, selective JAK3 inhibitor and does not affect the activity …
Formula:
C15H19N5O
Purity:
98.82% - 99.92%
Color and Shape:
Solid
Molecular weight:
285.34
Ref: TM-T5382
| 2mg | 46.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 325.00 € | ||
| 100mg | 485.00 € | ||
| 200mg | 690.00 € | ||
| 500mg | 1,047.00 € | ||
| 1mL*10mM (DMSO) | 76.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
