Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
Read more
Subcategories of "Chromatin/Epigenetics"
Products of "Chromatin/Epigenetics"
Picolinamide
CAS:1452-77-3
Picolinamide (Picolinoylamide) is found to be a strong inhibitor of poly (ADP-ribose) synthetase of nuclei …
Formula:
C6H6N2O
Purity:
99.60%
Color and Shape:
Solid
Molecular weight:
122.12
Ref: TM-T6942
| 1g | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MS049
CAS:1502816-23-0
MS 049 is a potent, selective, and cell-active dual inhibitor of PRMT4 and PRMT6 with …
Formula:
C15H24N2O
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
248.36
Ref: TM-T4378
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 157.00 € | ||
| 50mg | 235.00 € | ||
| 100mg | 353.00 € | ||
| 200mg | 520.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TCS-PIM-1-4a
CAS:327033-36-3
SMI-4a, a Pim inhibitor, activates AMPK, halts mTORC1, and kills various myeloid/lymphoid cells (IC50=0.8-40μM).
Formula:
C11H6F3NO2S
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
273.23
Ref: TM-T4215
| 5mg | 51.00 € | ||
| 10mg | 75.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 210.00 € | ||
| 100mg | 315.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MS023
CAS:1831110-54-3
MS023 is a potent, selective, and cell-active Type I PRMT inhibitor with IC50 of 30 …
Formula:
C17H25N3O
Purity:
98.31% - 99.28%
Color and Shape:
Solid
Molecular weight:
287.4
Ref: TM-T6900
| 1mg | 39.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 238.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 550.00 € | ||
| 500mg | 1,194.00 € | ||
| 1mL*10mM (DMSO) | 83.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GSK121
CAS:1652591-80-4
GSK121 is an inhibitor of selective PAD4.
Formula:
C25H26F3N5O3
Purity:
98.92%
Color and Shape:
Solid
Molecular weight:
501.51
Ref: TM-T24105
| 1mg | 54.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 199.00 € | ||
| 25mg | 423.00 € | ||
| 50mg | 610.00 € | ||
| 100mg | 853.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PJ34
CAS:344458-19-1
PJ34 HCl is the hydrochloride salt of PJ34, which is a PARP inhibitor with EC50 …
Formula:
C17H17N3O2
Purity:
95.05% - 99.85%
Color and Shape:
Solid
Molecular weight:
295.34
Ref: TM-T6197
| 10mg | 52.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 144.00 € | ||
| 100mg | 225.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
HIF-2α-IN-4
CAS:882268-69-1
HIF-2a translation inhibitor is a compound used as a molecular building block.
Formula:
C9H9N3O4S2
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
287.32
Ref: TM-T50099
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 186.00 € | ||
| 50mg | 349.00 € | ||
| 100mg | 522.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
SP-146
SP-146 is a selective, potent and non-ATP-competitive Aurora B inhibitor(IC50 : 0.316 nM).
Formula:
C25H20FN7O
Purity:
97.82%
Color and Shape:
Solid
Molecular weight:
453.47
Ref: TM-T8685
| 1mg | 85.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € | ||
| 1mL*10mM (DMSO) | 172.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
dBET1
CAS:1799711-21-9
dBET1 fuses (+)-JQ1 with thalidomide, degrades BET proteins via cereblon (EC50: 430 nM), and triggers …
Formula:
C38H37ClN8O7S
Purity:
98.14% - 99.3%
Color and Shape:
Solid
Molecular weight:
785.27
Ref: TM-T4495
| 1mg | 52.00 € | ||
| 5mg | 103.00 € | ||
| 10mg | 168.00 € | ||
| 25mg | 279.00 € | ||
| 50mg | 446.00 € | ||
| 100mg | 678.00 € | ||
| 500mg | 1,397.00 € | ||
| 1mL*10mM (DMSO) | 167.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ZM39923 hydrochloride
CAS:1021868-92-7
ZM39923 hydrochloride (JAK3 Inhibitor IV) is an JAK1/3 inhibitor, almost no activity to JAK2 and …
Formula:
C23H25NO·HCl
Purity:
98.05%
Color and Shape:
Solid
Molecular weight:
367.91
Ref: TM-T6145
| 5mg | 58.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 304.00 € | ||
| 100mg | 455.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MK-8745
CAS:885325-71-3
MK-8745 is a potent and selective Aurora A inhibitor.
Formula:
C20H19ClFN5OS
Purity:
98.94% - 99.31%
Color and Shape:
Solid
Molecular weight:
431.91
Ref: TM-T2471
| 5mg | 45.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 146.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
JANEX-1
CAS:202475-60-3
JANEX-1: cell-permeable, reversible Jak3 inhibitor (IC50: 78 μM), ATP-competitive, selective; weak on JAK1/2, Zap/Syk, SRC.
Formula:
C16H15N3O3
Purity:
98% - 99.73%
Color and Shape:
Solid
Molecular weight:
297.31
Ref: TM-T2045
| 1mg | 44.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 149.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 439.00 € | ||
| 100mg | 644.00 € | ||
| 500mg | 1,347.00 € | ||
| 1mL*10mM (DMSO) | 91.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
SGC2085
CAS:1821908-48-8
SGC2085 is an effective and selective coactivator-associated arginine methyltransferase 1 (CARM1) inhibitor (IC50: 50 nM).
Formula:
C19H24N2O2
Purity:
99.71% - 99.86%
Color and Shape:
Solid
Molecular weight:
312.41
Ref: TM-T7089
| 1mg | 87.00 € | ||
| 2mg | 118.00 € | ||
| 5mg | 225.00 € | ||
| 10mg | 337.00 € | ||
| 25mg | 557.00 € | ||
| 50mg | 810.00 € | ||
| 100mg | 1,116.00 € | ||
| 1mL*10mM (DMSO) | 159.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
CPI-1205
CAS:1621862-70-1
CPI-1205 is a highly potent and selective inhibitor of EZH2(IC50 : 0.002 μM, EC50 : …
Formula:
C27H33F3N4O3
Purity:
98.71% - 99.7%
Color and Shape:
Solid
Molecular weight:
518.57
Ref: TM-T8510
| 1mg | 92.00 € | ||
| 2mg | 119.00 € | ||
| 5mg | 208.00 € | ||
| 10mg | 307.00 € | ||
| 25mg | 519.00 € | ||
| 50mg | 731.00 € | ||
| 1mL*10mM (DMSO) | 447.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
DCLX069
CAS:792946-69-1
DCLX069: PRMT1 inhibitor, IC50=17.9µM, targets SAM pocket, inhibits breast/liver cancer, and AML cell growth.
Formula:
C20H25N3O2
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
339.43
Ref: TM-T27133
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 307.00 € | ||
| 100mg | 489.00 € | ||
| 500mg | 1,012.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
AZD5305
CAS:2589531-76-8
AZD5305 is a potent, selective and oral active PARP inhibitor.
Formula:
C22H26N6O2
Purity:
98.68% - 99.19%
Color and Shape:
Solid
Molecular weight:
406.48
Ref: TM-T9165
| 1mg | 111.00 € | ||
| 5mg | 230.00 € | ||
| 10mg | 369.00 € | ||
| 25mg | 617.00 € | ||
| 50mg | 879.00 € | ||
| 100mg | 1,190.00 € | ||
| 1mL*10mM (DMSO) | 257.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Peficitinib
CAS:944118-01-8
Peficitinib (ASP015K) (ASP015K, JNJ-54781532) is an orally bioavailable JAK inhibitor. Phase 3.
Formula:
C18H22N4O2
Purity:
98.67% - 99.4%
Color and Shape:
Solid
Molecular weight:
326.39
Ref: TM-T6933
| 2mg | 40.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 176.00 € | ||
| 50mg | 272.00 € | ||
| 100mg | 424.00 € | ||
| 200mg | 634.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
E-7386
CAS:1799824-08-0
E-7386 is an oral active CBP/ -catenin modulator.
Formula:
C39H48FN9O4
Purity:
98.92% - 99%
Color and Shape:
Solid
Molecular weight:
725.85
Ref: TM-T11136
| 1mg | 96.00 € | ||
| 5mg | 252.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 638.00 € | ||
| 50mg | 906.00 € | ||
| 100mg | 1,196.00 € | ||
| 1mL*10mM (DMSO) | 396.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Olaparib
CAS:763113-22-0
View and buy Olaparib from TargetMol.Olaparib is a small molecule inhibitor of PARP1/PARP2.Cited in 10 …
Formula:
C24H23FN4O3
Purity:
100% - 99.90%
Color and Shape:
Solid
Molecular weight:
434.46
Ref: TM-T3015
| 1g | 234.00 € | ||
| 5mg | 37.00 € | ||
| 10mg | 53.00 € | ||
| 50mg | 75.00 € | ||
| 100mg | 90.00 € | ||
| 200mg | 118.00 € | ||
| 500mg | 170.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TP-3654
CAS:1361951-15-6
TP-3654 is a second-generation Pim kinase inhibitor (Ki values against Pim-1/3: 5/42 nM).
Formula:
C22H25F3N4O
Purity:
97.72% - 99.95%
Color and Shape:
Solid
Molecular weight:
418.46
Ref: TM-T4523
| 5mg | 56.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 148.00 € | ||
| 50mg | 231.00 € | ||
| 100mg | 345.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
