Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
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Subcategories of "Chromatin/Epigenetics"
Products of "Chromatin/Epigenetics"
E7449
CAS:1140964-99-3
E7449 is a potent inhibitor of PARP1, PARP2, TNKS1, and TNKS2 with IC50s of 2, …
Formula:
C18H15N5O
Purity:
97.13%
Color and Shape:
Solid
Molecular weight:
317.34
Ref: TM-T4471
| 1mg | 36.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 186.00 € | ||
| 50mg | 280.00 € | ||
| 100mg | 416.00 € | ||
| 200mg | 615.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Protosappanin A
CAS:102036-28-2
Protosappanin A combats brain inflammation, suppresses rat heart transplant rejection, fights MRSA, and inhibits HIV …
Formula:
C15H12O5
Purity:
100% - 99.42%
Color and Shape:
Solid
Molecular weight:
272.25
Ref: TM-TJS1779
| 1mg | 96.00 € | ||
| 5mg | 212.00 € | ||
| 10mg | 346.00 € | ||
| 25mg | 569.00 € | ||
| 50mg | 807.00 € | ||
| 100mg | 1,086.00 € | ||
| 1mL*10mM (DMSO) | 193.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Molibresib
CAS:1260907-17-2
Molibresib (GSK525762) is an inhibitor of BET proteins (IC50: about 35 nM).
Formula:
C22H22ClN5O2
Purity:
98% - 99.08%
Color and Shape:
Solid
Molecular weight:
423.9
Ref: TM-T1906
| 1mg | 42.00 € | ||
| 2mg | 56.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 213.00 € | ||
| 50mg | 352.00 € | ||
| 100mg | 526.00 € | ||
| 200mg | 736.00 € | ||
| 500mg | 1,149.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
(+)-JQ1 PA
CAS:2115701-93-2
(+)-JQ1 PA is a derivative of the Bromodomain and extra-terminal (BET) inhibitor JQ1(IC50 of 10.4 …
Formula:
C22H20ClN5OS
Purity:
98.36%
Color and Shape:
Solid
Molecular weight:
437.95
Ref: TM-T17311
| 1mg | 49.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 147.00 € | ||
| 25mg | 259.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 555.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
WM-1119
CAS:2055397-28-7
WM-1119 is a highly potent, selective KAT6A/B inhibitor
Formula:
C18H13F2N3O3S
Purity:
96.59% - 98.18%
Color and Shape:
Solid
Molecular weight:
389.38
Ref: TM-T4679
| 5mg | 51.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 150.00 € | ||
| 100mg | 215.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
XD14
CAS:1370888-71-3
XD14 inhibits BET bromodomains with Kd: BRD4(1) 160nM, BRD2(1) 170nM, BRD3(1) 380nM, BRD3(2) 490nM, BRD2(2) …
Formula:
C20H27N3O5S
Purity:
98.4%
Color and Shape:
Solid
Molecular weight:
421.51
Ref: TM-T19935
| 1mg | 51.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 324.00 € | ||
| 50mg | 515.00 € | ||
| 100mg | 728.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
FL-411
CAS:2118944-88-8
FL-411 (BRD4-IN-1) is a potent and selective BRD4 inhibitor with an IC50 of 0.43±0.09 μM …
Formula:
C18H19N3O2S
Purity:
96.23%
Color and Shape:
Solid
Molecular weight:
341.43
Ref: TM-T4365
| 2mg | 35.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 272.00 € | ||
| 100mg | 453.00 € | ||
| 200mg | 627.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
GSK3685032
CAS:2170137-61-6
GSK3685032 is a non-covalent and selective DNMT1 inhibitor(IC50 = 36 nM).
Formula:
C22H24N6OS
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
420.53
Ref: TM-T9573
| 1mg | 91.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 296.00 € | ||
| 25mg | 555.00 € | ||
| 50mg | 795.00 € | ||
| 100mg | 1,087.00 € | ||
| 1mL*10mM (DMSO) | 200.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Daminozide
CAS:1596-84-5
Daminozide (Succinic Acid) is a plant growth regulator, selectively inhibits the KDM2/7 JmjC subfamily.
Formula:
C6H12N2O3
Purity:
99.88%
Color and Shape:
White Crystalline Solid Physical Description Odorless White Crystals Or Powder (Ntp 1992)
Molecular weight:
160.17
Ref: TM-T3719
| 1g | 59.00 € | ||
| 5g | 85.00 € | ||
| 500mg | 54.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
GSK-5959
CAS:901245-65-6
GSK-5959 is a selective BRPF1 inhibitor with IC50 ~80 nM, 100-fold more specific than 35 …
Formula:
C22H26N4O3
Purity:
98.35% - 98.65%
Color and Shape:
Solid
Molecular weight:
394.47
Ref: TM-T1972
| 5mg | 57.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 155.00 € | ||
| 50mg | 247.00 € | ||
| 100mg | 368.00 € | ||
| 200mg | 538.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Deucravacitinib
CAS:1609392-27-9
Deucravacitinib (BMS-986165) is a highly selective, orally bioavailable, allosteric TYK2 inhibitor.Cost-effective and quality-assured.
Formula:
C20H19D3N8O3
Purity:
100% - 99.43%
Color and Shape:
Solid
Molecular weight:
425.46
Ref: TM-T14687
| 1mg | 69.00 € | ||
| 5mg | 149.00 € | ||
| 10mg | 269.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 625.00 € | ||
| 100mg | 892.00 € | ||
| 200mg | 1,205.00 € | ||
| 500mg | 1,784.00 € | ||
| 1mL*10mM (DMSO) | 165.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Momelotinib
CAS:1056634-68-4
Momelotinib (LM-1149), an oral JAK1/2 inhibitor with IC50s 11/18 nM, blocks ATP binding, disrupting JAK-STAT …
Formula:
C23H22N6O2
Purity:
97.47% - 99.56%
Color and Shape:
Solid
Molecular weight:
414.46
Ref: TM-T1849
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 163.00 € | ||
| 50mg | 254.00 € | ||
| 100mg | 399.00 € | ||
| 200mg | 612.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
MS436
CAS:1395084-25-9
MS436 is a selective, small-molecule inhibitor for the BRD4 bromodomains.
Formula:
C18H17N5O3S
Purity:
97.95% - 98.92%
Color and Shape:
Solid
Molecular weight:
383.42
Ref: TM-T1854
| 2mg | 43.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 191.00 € | ||
| 50mg | 341.00 € | ||
| 100mg | 498.00 € | ||
| 500mg | 1,068.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
SNS-314 Mesylate
CAS:1146618-41-8
SNS-314 Mesylate (SNS-314) is an effective and specific Aurora A/B/C inhibitor. SNS-314 is less inhibition …
Formula:
C18H15ClN6OS2·CH4O3S
Purity:
99.92% - 99.92%
Color and Shape:
Solid
Molecular weight:
527.04
Ref: TM-T2617
| 2mg | 39.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 244.00 € | ||
| 100mg | 384.00 € | ||
| 1mL*10mM (DMSO) | 70.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Niraparib
CAS:1038915-60-4
Niraparib (MK-4827) inhibits PARP1/PARP2 (IC50: 3.8/2.1 nM), effective on BRCA mutant cancers, 330x less effective …
Formula:
C19H20N4O
Purity:
98% - 99.91%
Color and Shape:
Solid
Molecular weight:
320.39
Ref: TM-T3231
| 5mg | 59.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 111.00 € | ||
| 50mg | 142.00 € | ||
| 100mg | 213.00 € | ||
| 200mg | 314.00 € | ||
| 500mg | 543.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
AKBA
CAS:67416-61-9
AKBA (3-O-Acetyl-11-keto-beta-boswellic acid), a natural component from frankincense, is a novel activator of Nrf2.
Formula:
C32H48O5
Purity:
97.85% - 99.77%
Color and Shape:
Solid
Molecular weight:
512.72
Ref: TM-T5S1569
| 1g | 1,822.00 € | ||
| 1mg | 42.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 273.00 € | ||
| 100mg | 431.00 € | ||
| 500mg | 1,162.00 € | ||
| 1mL*10mM (DMSO) | 143.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
MN-64
CAS:92831-11-3
MN-64 is a tankyrases inhibitor, showed 6 nM potency against tankyrase 1, isoenzyme selectivity, and …
Formula:
C18H16O2
Purity:
99.36% - 99.93%
Color and Shape:
Solid
Molecular weight:
264.32
Ref: TM-T3168
| 10mg | 44.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 122.00 € | ||
| 100mg | 182.00 € | ||
| 200mg | 272.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
SGC0946
CAS:1561178-17-3
SGC0946 is a highly effective and specific DOT1L methyltransferase inhibitor (IC50: 0.3 nM); selectively kill …
Formula:
C28H40BrN7O4
Purity:
98% - 99.82%
Color and Shape:
Solid
Molecular weight:
618.57
Ref: TM-T3082
| 2mg | 53.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 423.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
SMI-16a
CAS:587852-28-6
SMI-16a (PIM1/2 Kinase Inhibitor VI) , a cell-permeable thiazolidinedione compound, acts as an effective, ATP-competitive …
Formula:
C13H13NO3S
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
263.31
Ref: TM-T3989
| 1mg | 35.00 € | ||
| 2mg | 47.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 231.00 € | ||
| 100mg | 346.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
OF-1
CAS:919973-83-4
OF-1 is a potent inhibitor of BRPF1B and BRPF2 bromodomain.
Formula:
C17H18BrN3O4S
Purity:
98.55% - ≥95%
Color and Shape:
Solid
Molecular weight:
440.31
Ref: TM-T2127
| 1mg | 38.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 132.00 € | ||
| 25mg | 251.00 € | ||
| 50mg | 401.00 € | ||
| 100mg | 621.00 € | ||
| 200mg | 868.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
