Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
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Subcategories of "Chromatin/Epigenetics"
Products of "Chromatin/Epigenetics"
CPI-1205
CAS:1621862-70-1
CPI-1205 is a highly potent and selective inhibitor of EZH2(IC50 : 0.002 μM, EC50 : …
Formula:
C27H33F3N4O3
Purity:
98.71% - 99.7%
Color and Shape:
Solid
Molecular weight:
518.57
Ref: TM-T8510
| 1mg | 92.00 € | ||
| 2mg | 119.00 € | ||
| 5mg | 208.00 € | ||
| 10mg | 307.00 € | ||
| 25mg | 519.00 € | ||
| 50mg | 731.00 € | ||
| 1mL*10mM (DMSO) | 447.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
DCLX069
CAS:792946-69-1
DCLX069: PRMT1 inhibitor, IC50=17.9µM, targets SAM pocket, inhibits breast/liver cancer, and AML cell growth.
Formula:
C20H25N3O2
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
339.43
Ref: TM-T27133
| 5mg | 50.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 113.00 € | ||
| 50mg | 179.00 € | ||
| 100mg | 285.00 € | ||
| 200mg | 400.00 € | ||
| 1mL*10mM (DMSO) | 54.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
AZD5305
CAS:2589531-76-8
AZD5305 is a potent, selective and oral active PARP inhibitor.
Formula:
C22H26N6O2
Purity:
98.68% - 99.19%
Color and Shape:
Solid
Molecular weight:
406.48
Ref: TM-T9165
| 1mg | 111.00 € | ||
| 5mg | 230.00 € | ||
| 10mg | 369.00 € | ||
| 25mg | 617.00 € | ||
| 50mg | 879.00 € | ||
| 100mg | 1,190.00 € | ||
| 1mL*10mM (DMSO) | 257.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
Peficitinib
CAS:944118-01-8
Peficitinib (ASP015K) (ASP015K, JNJ-54781532) is an orally bioavailable JAK inhibitor. Phase 3.
Formula:
C18H22N4O2
Purity:
98.67% - 99.4%
Color and Shape:
Solid
Molecular weight:
326.39
Ref: TM-T6933
| 2mg | 44.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 176.00 € | ||
| 50mg | 272.00 € | ||
| 100mg | 424.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
E-7386
CAS:1799824-08-0
E-7386 is an oral active CBP/ -catenin modulator.
Formula:
C39H48FN9O4
Purity:
98.92% - 99%
Color and Shape:
Solid
Molecular weight:
725.85
Ref: TM-T11136
| 1mg | 96.00 € | ||
| 5mg | 252.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 638.00 € | ||
| 50mg | 906.00 € | ||
| 100mg | 1,196.00 € | ||
| 1mL*10mM (DMSO) | 396.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
Olaparib
CAS:763113-22-0
View and buy Olaparib from TargetMol.Olaparib is a small molecule inhibitor of PARP1/PARP2.Cited in 10 …
Formula:
C24H23FN4O3
Purity:
100% - 99.90%
Color and Shape:
Solid
Molecular weight:
434.46
Ref: TM-T3015
| 1g | 234.00 € | ||
| 5mg | 37.00 € | ||
| 10mg | 53.00 € | ||
| 50mg | 75.00 € | ||
| 100mg | 90.00 € | ||
| 200mg | 118.00 € | ||
| 500mg | 170.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
TP-3654
CAS:1361951-15-6
TP-3654 is a second-generation Pim kinase inhibitor (Ki values against Pim-1/3: 5/42 nM).
Formula:
C22H25F3N4O
Purity:
97.72% - 99.95%
Color and Shape:
Solid
Molecular weight:
418.46
Ref: TM-T4523
| 5mg | 56.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 148.00 € | ||
| 50mg | 231.00 € | ||
| 100mg | 345.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
E7449
CAS:1140964-99-3
E7449 is a potent inhibitor of PARP1, PARP2, TNKS1, and TNKS2 with IC50s of 2, …
Formula:
C18H15N5O
Purity:
97.13%
Color and Shape:
Solid
Molecular weight:
317.34
Ref: TM-T4471
| 1mg | 45.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 537.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
Protosappanin A
CAS:102036-28-2
Protosappanin A combats brain inflammation, suppresses rat heart transplant rejection, fights MRSA, and inhibits HIV …
Formula:
C15H12O5
Purity:
100% - 99.42%
Color and Shape:
Solid
Molecular weight:
272.25
Ref: TM-TJS1779
| 1mg | 96.00 € | ||
| 5mg | 212.00 € | ||
| 10mg | 346.00 € | ||
| 25mg | 569.00 € | ||
| 50mg | 807.00 € | ||
| 100mg | 1,086.00 € | ||
| 1mL*10mM (DMSO) | 193.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
Molibresib
CAS:1260907-17-2
Molibresib (GSK525762) is an inhibitor of BET proteins (IC50: about 35 nM).
Formula:
C22H22ClN5O2
Purity:
98% - 99.08%
Color and Shape:
Solid
Molecular weight:
423.9
Ref: TM-T1906
| 1mg | 42.00 € | ||
| 2mg | 56.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 213.00 € | ||
| 50mg | 352.00 € | ||
| 100mg | 526.00 € | ||
| 200mg | 736.00 € | ||
| 500mg | 1,149.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
(+)-JQ1 PA
CAS:2115701-93-2
(+)-JQ1 PA is a derivative of the Bromodomain and extra-terminal (BET) inhibitor JQ1(IC50 of 10.4 …
Formula:
C22H20ClN5OS
Purity:
98.36%
Color and Shape:
Solid
Molecular weight:
437.95
Ref: TM-T17311
| 1mg | 49.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 147.00 € | ||
| 25mg | 259.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 555.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
C-82
CAS:1422253-37-9
C-82 is a specific CBP/β-catenin antagonist. It inhibits the binding between β-catenin and CBP and …
Formula:
C33H34N6O4
Purity:
98.86% - 99.66%
Color and Shape:
Solid
Molecular weight:
578.66
Ref: TM-T10641
| 1mg | 423.00 € | ||
| 5mg | 848.00 € | ||
| 10mg | 1,225.00 € | ||
| 25mg | 1,953.00 € | ||
| 1mL*10mM (DMSO) | 1,123.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
Itacitinib
CAS:1334298-90-6
Itacitinib (INCB039110) is an orally bioavailable inhibitor of Janus-associated kinase 1 (JAK1) with potential antineoplastic …
Formula:
C26H23F4N9O
Purity:
96.4% - 99.01%
Color and Shape:
Solid
Molecular weight:
553.51
Ref: TM-T3998
| 1mg | 49.00 € | ||
| 2mg | 70.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 177.00 € | ||
| 25mg | 320.00 € | ||
| 50mg | 534.00 € | ||
| 100mg | 763.00 € | ||
| 500mg | 1,523.00 € | ||
| 1mL*10mM (DMSO) | 136.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
A-966492
CAS:934162-61-5
A-96649 is a new-type and effective inhibitor. The Ki of A-966492 for PARP1 and PARP2 …
Formula:
C18H17FN4O
Purity:
98.53% - 99.25%
Color and Shape:
Solid
Molecular weight:
324.35
Ref: TM-T6366
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 266.00 € | ||
| 100mg | 381.00 € | ||
| 200mg | 540.00 € | ||
| 1mL*10mM (DMSO) | 54.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
GSK503
CAS:1346572-63-1
GSK-503, a potent EZH2 inhibitor, has potential antitumor activity.
Formula:
C31H38N6O2
Purity:
98% - 99.74%
Color and Shape:
Solid
Molecular weight:
526.67
Ref: TM-T1775
| 1mg | 36.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 204.00 € | ||
| 50mg | 368.00 € | ||
| 100mg | 551.00 € | ||
| 500mg | 1,188.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
PFI-4
CAS:900305-37-5
PFI-4 is a potent and selective and cell-permeable BRPF1 bromodomain inhibitor.
Formula:
C21H24N4O3
Purity:
99.53% - ≥95%
Color and Shape:
Solid
Molecular weight:
380.44
Ref: TM-T1973
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 118.00 € | ||
| 50mg | 185.00 € | ||
| 100mg | 305.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
NI-57
CAS:1883548-89-7
NI-57 inhibits BRPF family proteins: BRPF1 (IC50=3.1nM), BRPF2 (IC50=46nM), BRPF3 (IC50=140nM).
Formula:
C19H17N3O4S
Purity:
100% - 98%
Color and Shape:
Solid
Molecular weight:
383.42
Ref: TM-TQ0083
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 165.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
Menin-MLL inhibitor MI-2
CAS:1271738-62-5
Menin-MLL inhibitor MI-2 (MI2) is a potent menin-MLL interaction inhibitor with IC50 of 446 nM.
Formula:
C18H25N5S2
Purity:
97.46%
Color and Shape:
Solid
Molecular weight:
375.55
Ref: TM-T2649
| 2mg | 41.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 237.00 € | ||
| 100mg | 368.00 € | ||
| 200mg | 538.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
Molibresib besylate
CAS:1895049-20-3
Molibresib besylate (GSK 525762C) is a BET protein family inhibitor used in the study of …
Formula:
C28H28ClN5O5S
Purity:
99.64% - 99.64%
Color and Shape:
Solid
Molecular weight:
582.07
Ref: TM-T11472L
| 2mg | 144.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
Oroxylin A
CAS:480-11-5
Oroxylin A fights tumors, aids RAS therapy, promotes CaCo-2 cell apoptosis, blocks MCF-7 cell invasion …
Formula:
C16H12O5
Purity:
98.72% - 99.55%
Color and Shape:
Solid
Molecular weight:
284.26
Ref: TM-T6S1315
| 20mg | 135.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
