Thyroid hormone receptor(THR)
Thyroid hormone receptors (THRs) are nuclear receptors that mediate the effects of thyroid hormones, which are critical for regulating metabolism, growth, and development. Modulation of THR activity is important in the treatment of thyroid disorders, metabolic syndromes, and certain cancers. THR agonists and antagonists are used in research to study the physiological and pathological roles of thyroid hormones. At CymitQuimica, we offer a wide range of high-quality thyroid hormone receptor modulators to support your research in endocrinology, metabolism, and hormone regulation.
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Taltirelin acetate
CAS:1549593-23-8
Taltirelin acetate (TA-0910 acetate) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM …
Formula:
C19H27N7O7
Purity:
99.44%
Color and Shape:
Solid
Molecular weight:
465.46
Ref: TM-T13072
| 2mg | 36.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 149.00 € | ||
| 50mg | 241.00 € | ||
| 100mg | 375.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
3,5-Diiodothyropropionic acid
CAS:1158-10-7
3,5-Diiodothyropropionic acid: thyroid hormone analog, boosts α-myosin mRNA, binds TRα1 & TRβ1 (Ka: 2.40/M, 4.06/M).
Formula:
C15H12I2O4
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
510.06
Ref: TM-T13492
| 5mg | 46.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 115.00 € | ||
| 50mg | 170.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Carbimazole
CAS:22232-54-8
Carbimazole, an imidazolium-based thyroid blocker, turns to MMI in the body. Used in Graves' disease …
Formula:
C7H10N2O2S
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
186.23
Ref: TM-T0952
| 500mg | 50.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Methimazole
CAS:60-56-0
Methimazole (Thiamazole) is an antithyroid compound with significant hepatotoxicity and is often used in the …
Formula:
C4H6N2S
Purity:
99.94%
Color and Shape:
White Solid
Molecular weight:
114.17
Ref: TM-T0840
| 500mg | 49.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Tiratricol
CAS:51-24-1
Tiratricol, a thyroid hormone metabolite for hyperlipidemia and obesity, studied in Allan-Herndon-Dudley Syndrome treatment.
Formula:
C14H9I3O4
Purity:
99.16% - 99.6%
Color and Shape:
Solid
Molecular weight:
621.93
Ref: TM-T1604
| 1g | 133.00 € | ||
| 50mg | 39.00 € | ||
| 100mg | 52.00 € | ||
| 200mg | 65.00 € | ||
| 500mg | 93.00 € | ||
| 1mL*10mM (DMSO) | 44.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Propylthiouracil
CAS:51-52-5
Propylthiouracil (6-n-Propylthiouracil) is a thyroid peroxidase inhibitor and also a 5' -deiodinase inhibitor.
Formula:
C7H10N2OS
Purity:
99.94%
Color and Shape:
White Crystalline Powder Of Starch-Like Appearance To Eye And To Touch Saturated Solution Is Neutral Or Slightly Acid To Litmus (Ntp 1992)
Molecular weight:
170.23
Ref: TM-T1309
| 25mg | 39.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 63.00 € | ||
| 200mg | 78.00 € | ||
| 500mg | 94.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
L-Thyroxine sodium salt pentahydrate
CAS:6106-07-6
L-Thyroxine sodium salt pentahydrate is a thyroid hormone that inhibits the release of thyroid hormones …
Formula:
C15H20I4NNaO9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
888.93
Ref: TM-T15699
| 100mg | 36.00 € | ||
| 500mg | 55.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
NH-3
CAS:447415-26-1
NH-3, an orally active THR antagonist with a 55 nM IC50, blocks thyroid hormone binding …
Formula:
C28H27NO6
Purity:
97.09%
Color and Shape:
Solid
Molecular weight:
473.52
Ref: TM-T40548
| 1mg | 214.00 € | ||
| 5mg | 539.00 € | ||
| 10mg | 774.00 € | ||
| 25mg | 1,179.00 € | ||
| 50mg | 1,576.00 € | ||
| 100mg | 2,140.00 € | ||
| 500mg | 4,291.00 € | ||
| 1mL*10mM (DMSO) | 485.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Taltirelin
CAS:103300-74-9
Taltirelin (TA-0910) is at thyrotropin-releasing hormone receptor (TRH-R) superagonist (IC50 of 910 nM and EC50 …
Formula:
C17H23N7O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
405.41
Ref: TM-T7590
| 2mg | 63.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AH-3960
CAS:862907-48-0
AH-3960 is an thyroid hormone receptor-1 (PTHR1) agonist.
Formula:
C13H22N4O3
Purity:
98.44%
Color and Shape:
Solid
Molecular weight:
282.34
Ref: TM-T23673
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 384.00 € | ||
| 50mg | 591.00 € | ||
| 100mg | 828.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Liothyronine sodium
CAS:55-06-1
Liothyronine Sodium is a synthetic T3 thyroid hormone, potent and faster-acting than T4, used for …
Formula:
C15H11I3NNaO4
Purity:
98%
Color and Shape:
Crystals White To Beige Powder
Molecular weight:
672.96
Ref: TM-T1669
| 100mg | 51.00 € | ||
| 200mg | 73.00 € | ||
| 500mg | 113.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Eprotirome
CAS:355129-15-6
Eprotirome (KB2115), a synthetic thyroid hormone mimetic, is a thyroid hormone receptor agonist.
Formula:
C18H17Br2NO5
Purity:
98.29% - 98.42%
Color and Shape:
Solid
Molecular weight:
487.14
Ref: TM-T5360
| 1mg | 90.00 € | ||
| 5mg | 218.00 € | ||
| 10mg | 324.00 € | ||
| 25mg | 516.00 € | ||
| 50mg | 693.00 € | ||
| 100mg | 916.00 € | ||
| 200mg | 1,246.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Glutaurine aceate
Glutaurine aceate containing glutamine and taurine residues is an orally active hormone of the parathyroid.
Formula:
C9H18N2O8S
Purity:
98%
Color and Shape:
Soild
Molecular weight:
314.31
Ref: TM-T25455L
| 5mg | 55.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 172.00 € | ||
| 100mg | 249.00 € | ||
| 200mg | 373.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
2,2-BIS(2-HYDROXY-5-BIPHENYLYL)PROPANE
CAS:24038-68-4
2,2-BIS(2-HYDROXY-5-BIPHENYLYL)PROPANE is targets the thyroid stimulating hormone receptor (human)
Formula:
C27H24O2
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
380.48
Ref: TM-T8672
| 500mg | 55.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
L-Thyroxine sodium
CAS:55-03-8
L-Thyroxine sodium (LT4 sodium), the major hormone derived from the thyroid gland, is the agonist …
Formula:
C15H10I4NO4·Na
Purity:
99.56%
Color and Shape:
Yellowish To Buff-Colored Amorphous Powder Solid
Molecular weight:
798.85
Ref: TM-T22355
| 1g | 67.00 € | ||
| 500mg | 51.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Sobetirome
CAS:211110-63-3
Sobetirome (IACS-010759) is a selective agonist of thyroid hormone receptor β (TRβ) and binds selectively …
Formula:
C20H24O4
Purity:
98.08% - 98.25%
Color and Shape:
Solid
Molecular weight:
328.4
Ref: TM-T5313
| 1mg | 48.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 278.00 € | ||
| 50mg | 551.00 € | ||
| 100mg | 782.00 € | ||
| 200mg | 1,054.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Liothyronine sodium hydrate
CAS:345957-19-9
Liothyronine sodium hydrate (Triiodothyronine sodium hydrate) is a TR伪 and TR尾 agonist and a thyroxine …
Formula:
C15H11NNaO4xH2O
Color and Shape:
Liquid
Molecular weight:
0
Ref: TM-T64268
| 10mg | 41.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 81.00 € | ||
| 100mg | 108.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
REVERSE T3
CAS:5817-39-0
Reverse T3 (3,3',5'-triiodo-L-thyronine) inhibits the increase of sodium current generated by other thyroid hormone analogs …
Formula:
C15H12I3NO4
Purity:
95.99% - 97.66%
Color and Shape:
Powder
Molecular weight:
650.97
Ref: TM-T7578
| 1mg | 49.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 621.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Resmetirom
CAS:920509-32-6
Resmetirom (VIA-3196) is a highly selective thyroid hormone receptor β (THR-β) agonist.
Formula:
C17H12Cl2N6O4
Purity:
100% - 99.91%
Color and Shape:
Solid
Molecular weight:
435.22
Ref: TM-T3595
| 1mg | 39.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 209.00 € | ||
| 50mg | 335.00 € | ||
| 100mg | 497.00 € | ||
| 500mg | 1,108.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
KAT681
CAS:373641-87-3
KAT681 is a liver selective thyromimetic.
Formula:
C24H22FNNaO6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
462.429
Ref: TM-T15644
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
