Vasopressin Receptor
Vasopressin receptors are a family of G protein-coupled receptors that mediate the effects of vasopressin, a hormone involved in regulating water balance, blood pressure, and kidney function. Vasopressin receptor agonists and antagonists are studied for their roles in treating conditions such as diabetes insipidus, hyponatremia, and heart failure. These receptors are also important targets in research on fluid balance and cardiovascular health. At CymitQuimica, we provide a selection of high-quality vasopressin receptor modulators to support your research in endocrinology, nephrology, and cardiovascular biology.
Found 47 products for "Vasopressin Receptor".
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[Deamino-Pen1,Val4,D-Arg8]-vasopressin
CAS:[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an antagonist of arginine-vasopressin (AVP).Formula:C48H69N13O11S2Purity:98%Color and Shape:SolidMolecular weight:1068.27Val9-Oxytocin
CAS:Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor.Formula:C46H72N12O12S2Purity:98%Color and Shape:SolidMolecular weight:1049.27(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS:(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].Formula:C52H76N14O11S2Purity:98%Color and Shape:SolidMolecular weight:1137.38V1a/V2 antagonist 1
V1a/V2 antagonist 1 (Compound 18j) is an orally active dual-target antagonist of V1a and V2 receptors, exhibiting high binding affinity toward these receptors [Ki values are hV1a: 0.13 nM, hV2: 0.53 nM, and mV1a: 0.5 nM; IC50 for hV1a is 2.2 nM]. This compound can inhibit oxytocin-induced scratching behavior in mice.Formula:C25H26ClN5O3Color and Shape:SolidMolecular weight:479.96d[Leu4,Lys8]-VP
CAS:Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.Formula:C47H67N11O11S2Purity:98%Color and Shape:SolidMolecular weight:1026.2d[Cha4]-AVP TFA
d[Cha4]-AVP TFA: potent, selective V1b agonist, K i 1.2 nM, favors V1b over V1a, V2, oxytocin receptors.Formula:C52H72F3N13O13S2Color and Shape:SolidMolecular weight:1208.33Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
CAS:Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), acts as a weak agonist at the antidiuretic receptor but is a potentFormula:C45H63N15O11S2Color and Shape:SolidMolecular weight:1054.21[Asu1,6-Arg8]Vasopressin
CAS:[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.Formula:C48H68N14O12Color and Shape:SolidMolecular weight:1033.14(Phe2,Orn8)-Oxytocin acetate
(Phe2,Orn8)-Oxytocin acetate: V1 agonist with EC50 of 280 nM for rabbit epididymis contractility.Formula:C44H69N13O13S2Color and Shape:SolidMolecular weight:1052.23Fedovapagon
CAS:Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.Formula:C27H34N4O3Purity:99.46%Color and Shape:Yellow SolidMolecular weight:462.58Atosiban
CAS:Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions rapidly.Formula:C43H67N11O12S2Purity:98%Color and Shape:White SolidMolecular weight:994.19Argipressin
CAS:Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.Formula:C46H65N15O12S2Purity:98%Color and Shape:White SolidMolecular weight:1084.23Felypressin
CAS:Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.Formula:C46H65N13O11S2Purity:99.65%Color and Shape:SolidMolecular weight:1040.22RG7713
CAS:RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.Formula:C25H28ClN3O2Purity:99.74%Color and Shape:White SolidMolecular weight:437.96Desmopressin acetate (16679-58-6 free base)
CAS:Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine production.Formula:C48H68N14O14S2Purity:98.84% - >99.99%Color and Shape:White SolidMolecular weight:1129.26Fuscoside
CAS:Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.Formula:C26H31N3O4Purity:98.13% - 99.66%Color and Shape:White SolidMolecular weight:449.54Tolvaptan
CAS:Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.Formula:C26H25ClN2O3Purity:99.78% - >99.99%Color and Shape:SolidMolecular weight:448.94d[Cha4]-AVP acetate(500170-27-4 free base)
'd[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'Formula:C52H75N13O13S2Purity:99.86%Color and Shape:SolidMolecular weight:1154.37Atosiban acetate
CAS:Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin.Formula:C45H71N11O14S2Purity:97.08% - 99.92%Color and Shape:White SolidMolecular weight:1054.24Ref: TM-T5148
5mg70.00€10mg109.00€1mL*10mM (DMSO)127.00€25mg166.00€50mg195.00€100mg254.00€500mg625.00€Conivaptan hydrochloride
CAS:Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia andFormula:C32H26N4O2·HClPurity:98.33% - 99.86%Color and Shape:White SolidMolecular weight:535.04
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