Androgen Receptor
The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.
Found 229 products of "Androgen Receptor"
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Galeterone
CAS:Galeterone (VN 124) is an oral androgen receptor modulator/CYP17 inhibitor with antiandrogen properties, targeting prostate cancer growth.Formula:C26H32N2OPurity:99.47% - 99.773%Color and Shape:SolidMolecular weight:388.55CLP-3094
CAS:CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor.Formula:C15H13ClN2OSPurity:99.84%Color and Shape:SolidMolecular weight:304.79JNJ-63576253 free base
CAS:JNJ-63576253 free base (TRC253) is a potent and orally active full antagonist of androgen receptor (AR). JNJ-63576253 can be used for the research of CRPC.Formula:C23H21F3N6O2SPurity:98.32%Color and Shape:SolidMolecular weight:502.51Ref: TM-T8933
2mg38.00€5mg50.00€10mg85.00€25mg159.00€50mg244.00€100mg359.00€200mg512.00€1mL*10mM (DMSO)86.00€CTK8A3536
CAS:CTK8A3536 ((2-MORPHOLIN-4-YL-4-PHENYL-1,3-THIAZOL-5-YL)METHANOL) is an inhibitor of Androgen receptor.Formula:C14H16N2O2SPurity:99.62%Color and Shape:SolidMolecular weight:276.35Ref: TM-T8592
1mg84.00€5mg167.00€10mg245.00€25mg404.00€50mg567.00€100mg767.00€200mg1,018.00€1mL*10mM (DMSO)160.00€Ailanthone
CAS:Ailanthone (Δ13-Dehydrochaparrinone) is an effective inhibitor of both full-length androgen receptor (AR) (IC50: 69 nM) and constitutively active truncated ARFormula:C20H24O7Purity:99.71% - 99.96%Color and Shape:SolidMolecular weight:376.4ARD-2128
CAS:ARD-2128: potent oral PROTAC that degrades AR, curbing prostate cancer growth with no toxicity.Formula:C45H50ClN7O6Purity:98.8%Color and Shape:SolidMolecular weight:820.37Boldenone Undecylenate
CAS:Boldenone Undecylenate (Parenabol) is a synthetic steroid.Formula:C30H44O3Purity:99.39%Color and Shape:Light Yellow Oily MatterMolecular weight:452.67Ref: TM-T3137
1mg35.00€2mg48.00€5mg52.00€10mg85.00€25mg140.00€50mg246.00€100mg396.00€500mg939.00€1mL*10mM (DMSO)52.00€Triptophenolide
CAS:Triptophenolide (Hypolide) is a compound isolated from Tripterygium wilfordii Hook with anti-inflammatory activity.Formula:C20H24O3Purity:98.07% - ≥95%Color and Shape:White PowderMolecular weight:312.40AC-262536
CAS:AC-262536 is a selective androgen receptor (SAR) modulator and exhibits potent agonist activity at the androgen receptor.Formula:C18H18N2OPurity:99.88%Color and Shape:SolidMolecular weight:278.35Ref: TM-T26539
5mg46.00€10mg74.00€25mg145.00€50mg240.00€100mg359.00€200mg510.00€1mL*10mM (DMSO)49.00€Enzalutamide
CAS:Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist (IC50=36 nM in LNCaP).Formula:C21H16F4N4O2SPurity:99% - 99.93%Color and Shape:SolidMolecular weight:464.44Ref: TM-T6002
5mg48.00€10mg56.00€25mg74.00€50mg96.00€100mg154.00€200mg187.00€500mg274.00€1mL*10mM (DMSO)52.00€RU 58841
CAS:RU 58841 (PSK-3841) is a specific androgen receptor antagonist or anti-androgen; RU 58841(PSK-3841) has a significant effect on hair regrowth.Formula:C17H18F3N3O3Purity:99.31% - 99.70%Color and Shape:SolidMolecular weight:369.34Ref: TM-T2236
5mg40.00€10mg63.00€25mg99.00€50mg130.00€100mg177.00€200mg245.00€500mg371.00€1mL*10mM (DMSO)48.00€EPI-001
CAS:EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ～6 μM and a selective PPAR-gamma modulator.Formula:C21H27ClO5Purity:99% - 99.67%Color and Shape:SolidMolecular weight:394.89Ref: TM-T6829
2mg34.00€5mg48.00€10mg73.00€25mg120.00€50mg192.00€100mg286.00€200mg425.00€1mL*10mM (DMSO)49.00€Clascoterone
CAS:Clascoterone (CB-03-01) is a new topical and peripherally selective androgen antagonist.Formula:C24H34O5Purity:99.2% - 99.72%Color and Shape:SolidMolecular weight:402.52DSRM-3716
CAS:Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery ofFormula:C9H6INPurity:97.28% - 99.785%Color and Shape:SolidMolecular weight:255.06p,p'-DDE
CAS:p,p'-DDE (p,p'-dichlorodiphenyldichloroethylene) is a metabolite and degradation product of the organochlorine pesticide DDTFormula:C14H8Cl4Purity:99.68%Color and Shape:White Crystalline Solid Physical Description White Crystalline Solid Or White Powder (Ntp 1992)Molecular weight:318.03CSRM617 hydrochloride
CAS:CSRM617 hydrochloride: selective OC2 inhibitor, Kd 7.43 uM, binds OC2-HOX, induces apoptosis, tolerable in mouse prostate cancer.Formula:C10H14ClN3O5Purity:99.59%Color and Shape:SoildMolecular weight:291.69LY2452473
CAS:LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer activity for the study of prostate cancer.Formula:C22H22N4O2Purity:99.72%Color and Shape:SolidMolecular weight:374.44Ref: TM-T15804
1mg34.00€5mg67.00€10mg96.00€25mg133.00€50mg170.00€100mg253.00€200mg386.00€1mL*10mM (DMSO)73.00€Masofaniten
CAS:Masofaniten (EPI-7386) is an orally active androgen receptor (AR) inhibitor with antitumor activity for the study of prostate and breast cancer.Formula:C24H24Cl2N4O4SPurity:98.42% - 98.66%Color and Shape:SolidMolecular weight:535.44Estromustine
CAS:Estromustine, an active metabolite of estramustine phosphate, is used to treat prostate cancer.Formula:C23H29Cl2NO3Color and Shape:SolidMolecular weight:438.39GDC-2992
CAS:GDC-2992 is a selective androgen receptor (AR) degradator that degrades AR and inhibits proliferation in VCaP cells,CRPC.Formula:C45H51ClN8O5Purity:99.82%Color and Shape:SoildMolecular weight:819.39
