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Androgen Receptor

Androgen Receptor

The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.

Found 207 products of "Androgen Receptor"

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  • N-desmethyl Enzalutamide
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    N-desmethyl Enzalutamide

    CAS:
    <p>N-desmethyl Enzalutamide (N-desmethyl MDV 3100) is the active Enzalutamide metabolite.It is the active metabolite of Enzalutamide.</p>
    Formula:C20H14F4N4O2S
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:450.41

    Ref: TM-T19450

  • Enzalutamide carboxylic acid
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    Enzalutamide carboxylic acid

    CAS:
    <p>Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .</p>
    Formula:C20H13F4N3O3S
    Purity:97.88%
    Color and Shape:Solid
    Molecular weight:451.39

    Ref: TM-T8217

  • Clascoterone
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    Clascoterone

    CAS:
    <p>Clascoterone (CB-03-01) is a new topical and peripherally selective androgen antagonist.</p>
    Formula:C24H34O5
    Purity:99.2% - 99.64%
    Color and Shape:Solid
    Molecular weight:402.52

    Ref: TM-T3357

  • LY2452473
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    LY2452473

    CAS:
    <p>LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer activity for the study of prostate cancer.</p>
    Formula:C22H22N4O2
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:374.44

    Ref: TM-T15804

  • Masofaniten
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    Masofaniten

    CAS:
    <p>Masofaniten (EPI-7386) is an orally active androgen receptor (AR) inhibitor with antitumor activity for the study of prostate and breast cancer.</p>
    Formula:C24H24Cl2N4O4S
    Purity:98.42% - 98.66%
    Color and Shape:Solid
    Molecular weight:535.44

    Ref: TM-T72985

  • AR antagonist 6
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    AR antagonist 6

    CAS:
    <p>AR antagonist 6 (compound 6i), a diphenyl ether androgen receptor (AR) antagonist, binds to the AR with an affinity of 120 nM. It demonstrates low toxicity and effective in vitro activity in the golden Syrian hamster ear model. [19] [1]</p>
    Formula:C16H12F3NO2
    Color and Shape:Solid
    Molecular weight:307.27

    Ref: TM-T85718

  • GDC-2992
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    GDC-2992

    CAS:
    <p>GDC-2992 is a selective androgen receptor (AR) degradator that degrades AR and inhibits proliferation in VCaP cells,CRPC.</p>
    Formula:C45H51ClN8O5
    Purity:99.82%
    Color and Shape:Soild
    Molecular weight:819.39

    Ref: TM-T204088

  • Estromustine
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    Estromustine

    CAS:
    <p>Estromustine, an active metabolite of estramustine phosphate, is used to treat prostate cancer.</p>
    Formula:C23H29Cl2NO3
    Color and Shape:Solid
    Molecular weight:438.39

    Ref: TM-T25391

  • Procymidone
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    Procymidone

    CAS:
    <p>Procymidone is a broad-spectrum fungicide that inhibits fungal glycerol triester synthesis, thereby disrupting hyphal growth. androgen receptor (AR) antagonist</p>
    Formula:C13H11Cl2NO2
    Purity:99.86%
    Color and Shape:Colorless Solid
    Molecular weight:284.14

    Ref: TM-T20811

  • JNJ-37654032
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    JNJ-37654032

    CAS:
    <p>JNJ-37654032: orally active, nonsteroidal SARM. Mixed AR agonist/antagonist. Selective for muscle, grows levator ani, max at 3mg/kg, ED(50) 0.8mg/kg.</p>
    Formula:C11H7Cl2F3N2O
    Color and Shape:Solid
    Molecular weight:311.09

    Ref: TM-T27676

  • BMS-564929
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    BMS-564929

    CAS:
    <p>BMS-564929 is an AR agonist that upregulates the expression and activity of fat-producing enzymes, reducing VAT content and lipid levels.</p>
    Formula:C14H12ClN3O3
    Purity:98.17%
    Color and Shape:Solid
    Molecular weight:305.72

    Ref: TM-T14675

  • (R)-Bicalutamide
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    (R)-Bicalutamide

    CAS:
    <p>(R)-Bicalutamide, an AR antagonist with antitumor properties, is crucial in prostate cancer research.</p>
    Formula:C18H14F4N2O4S
    Color and Shape:Solid
    Molecular weight:430.37

    Ref: TM-T62386

  • LG-121071
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    LG-121071

    CAS:
    <p>LG-121071: oral SARM, high-affinity AR full agonist, Ki=17 nM.</p>
    Formula:C15H15F3N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:296.29

    Ref: TM-T27824

  • Honokiol DCA
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    Honokiol DCA

    CAS:
    <p>Honokiol DCA inhibits DRP1, enhances respiration via mitochondrial repair, and is active against Vemurafenib-resistant melanoma.</p>
    Formula:C22H18Cl4O4
    Color and Shape:Solid
    Molecular weight:488.19

    Ref: TM-T27551

  • Lubabegron fumarate
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    Lubabegron fumarate

    CAS:
    <p>Lubabegron (LY591281, LY488756 fumarate) is a beta-agonist approved in 2018 to lower ammonia in cattle waste, aiding environment and health.</p>
    Formula:C29H29N3O3SC4H4O4
    Color and Shape:Solid
    Molecular weight:557.66

    Ref: TM-T69306

  • Gumelutamide
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    Gumelutamide

    CAS:
    <p>Gumelutamide, a tetrahydropyridopyrimidine compound, functions as both an antiandrogen and an antineoplastic agent by acting as an androgen antagonist.</p>
    Formula:C22H21ClN6O
    Color and Shape:Solid
    Molecular weight:420.89

    Ref: TM-T72955

  • TFM-4AS-1
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    TFM-4AS-1

    CAS:
    <p>androgen receptor modulator</p>
    Formula:C27H33F3N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:474.56

    Ref: TM-T23455

  • HG122
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    HG122

    CAS:
    <p>HG122 promotes AR degradation via proteasome, inhibiting castration-resistant prostate cancer.</p>
    Formula:C15H13N5O5
    Color and Shape:Solid
    Molecular weight:343.29

    Ref: TM-T61109

  • Androgen receptor antagonist 4
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    Androgen receptor antagonist 4

    CAS:
    <p>Compound AT2 is an AR inhibitor with anticancer effects, blocking DHT action and AR nuclear translocation (IC50=0.15μM).</p>
    Formula:C22H18ClN
    Color and Shape:Solid
    Molecular weight:331.84

    Ref: TM-T60988

  • AZD3514
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    AZD3514

    CAS:
    <p>AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM and has ability of reducing AR protein expression.Phase 1.</p>
    Formula:C25H32F3N7O2
    Purity:98.09%
    Color and Shape:Solid
    Molecular weight:519.56

    Ref: TM-T6400