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Androgen Receptor

Androgen Receptor

The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.

Found 229 products of "Androgen Receptor"

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  • AR ligand-44
    Targetmol
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    AR ligand-44

    CAS:
    AR ligand-44 is an androgen receptor (androgen receptor) ligand that can be utilized in the synthesis of PROTACs such as [ARD-2051].
    Formula:C23H24ClN3O2
    Color and Shape:Solid
    Molecular weight:409.91

    Ref: TM-T212032

    10mg
    To inquire
    50mg
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  • Androgen receptor antagonist 11
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    Androgen receptor antagonist 11

    CAS:
    Androgen receptor antagonist 11 (compound N29) is a selective, orally available antagonist.
    Formula:C20H19F3N4O3S
    Color and Shape:Solid
    Molecular weight:452.45

    Ref: TM-T201269

    25mg
    1,602.00€
    50mg
    2,025.00€
    100mg
    2,600.00€
  • PROTAC Androgen receptor degrader-1
    Targetmol
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    PROTAC Androgen receptor degrader-1

    CAS:
    PROTACAndrogen receptor degrader-1 (Ex.14) is a PROTAC degrader targeting the androgen receptor, with a DC50 of 6 nM. This compound is applicable in prostate cancer research.
    Formula:C43H48ClN9O2
    Color and Shape:Solid
    Molecular weight:758.35

    Ref: TM-T212553

    10mg
    To inquire
    50mg
    To inquire
  • KF-19418
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    KF-19418

    CAS:
    KF-19418 is a follicle stimulant that directly activates follicles in vitro and promotes hair growth in vivo.
    Formula:C21H14N4O
    Color and Shape:Solid
    Molecular weight:338.36

    Ref: TM-T201487

    10mg
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    50mg
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  • Pentomone
    Targetmol
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    Pentomone

    CAS:
    Pentomone (LY-113935) is an anti-androgen compound that acts as a prostate growth inhibitor.
    Formula:C24H26O5
    Color and Shape:Solid
    Molecular weight:394.46

    Ref: TM-T201000

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • FL442
    Targetmol
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    FL442

    CAS:
    FL442 is an Androgen Receptor (AR) modulator. This compound exhibits potent inhibitory effects in AR-dependent prostate cancer cells, showing similar suppression efficiency to the traditional antiandrogen drugs Bicalutamide and Enzalutamide. It also maintains antiandrogen activity against the Enzalutamide-resistant AR mutant F876L. The pharmacokinetic properties of FL442 in mice reveal a longer half-life (8 hours), excellent targeting (prostate tissue), and metabolic stability. Additionally, it is effective at inhibiting LNCaP tumor growth at low plasma concentrations (30 ng/mL).
    Formula:C15H13F3N2O
    Color and Shape:Solid
    Molecular weight:294.27

    Ref: TM-T200138

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • LX1
    Targetmol
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    LX1

    CAS:
    LX1, an anti-prostate cancer compound, specifically targets the androgen receptor (AR), AR variants, and the steroidogenic enzyme AKR1C3. It inhibits AKR1C3's enzymatic function, decreases the conversion of androstenedione to testosterone, and reduces the expression of both AR and AR-V7, subsequently downregulating their target genes. Additionally, LX1 is effective in overcoming tumor cell resistance to Enzalutamide, and when combined with Enzalutamide, it further suppresses tumor growth.
    Formula:C22H15F6NO2
    Color and Shape:Solid
    Molecular weight:439.35

    Ref: TM-T200147

    25mg
    1,539.00€
    50mg
    1,941.00€
    100mg
    2,451.00€
  • Androstatrione
    Targetmol
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    Androstatrione

    CAS:

    Androstatrione is an androgenic compound.

    Formula:C19H26O3
    Color and Shape:Solid
    Molecular weight:302.41

    Ref: TM-T207371

    10mg
    To inquire
    50mg
    To inquire
  • PF-998425
    Targetmol
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    PF-998425

    CAS:
    non-steroidal androgen receptor (AR) antagonist
    Formula:C14H14F3NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:269.26

    Ref: TM-T23141

    25mg
    Discontinued
    Discontinued product