Androgen Receptor
The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.
Found 229 products of "Androgen Receptor"
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Ralaniten triacetate
CAS:Ralaniten triacetate (EPI-506) is a precursor of Ralaniten, an AR-NTD inhibitor, which can be used in the study of prostate and breast cancer.Formula:C27H33ClO8Purity:98.69%Color and Shape:SolidMolecular weight:521.00Ref: TM-T36375
1mg154.00€5mg371.00€10mg620.00€25mg1,341.00€50mg1,783.00€100mg2,250.00€1mL*10mM (DMSO)425.00€ONC1-13B
CAS:ONC1-13B, an androgen receptor antagonist, is used potentially for the treatment of prostate cancer.Formula:C22H16F4N4O3SPurity:99.36% - 99.85%Color and Shape:SolidMolecular weight:492.45GLPG0492
CAS:GLPG0492 is a novel selective androgen receptor modulator.Formula:C19H14F3N3O3Purity:99.58%Color and Shape:SolidMolecular weight:389.33Ref: TM-T11410L
1mg71.00€5mg156.00€10mg224.00€25mg358.00€50mg515.00€100mg692.00€200mg888.00€1mL*10mM (DMSO)166.00€Androgen receptor antagonist 5
CAS:AR antagonist 5 blocks AR (IC50: 6.17 μM), hinders LNCaP cell growth, and has anti-tumor effects in mouse models.Formula:C21H15F4N5O3SColor and Shape:SolidMolecular weight:493.43Celiprolol hydrochloride
CAS:Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.Formula:C20H33N3O4·HClColor and Shape:White Crystalline SolidMolecular weight:415.96VPC-14228
CAS:VPC-14228 is a specific AR-DBD inhibitor that acts by inhibiting both Y594A and Q592A mutants.Formula:C13H14N2OSPurity:99.96%Color and Shape:SolidMolecular weight:246.33N-Nitrosodicyclohexylamine
CAS:N-Nitrosodicyclohexylamine (NDCHA), an N-nitrosocompound, exhibits anti-androgenic activity by competitively binding to the androgen receptor (AR) in oppositionFormula:C12H22N2OPurity:98%Color and Shape:SolidMolecular weight:210.32Androgen receptor degrader-2
CAS:Androgen Receptor Degrader-2 (Compound 9) is a potent degrader of androgen receptors, with potential application in cancer research [1].Formula:C16H16ClN3O4Purity:98%Color and Shape:SolidMolecular weight:349.77(rel)-BMS-641988
CAS:(rel)-BMS-641988, a relative configuration of the potent nonsteroidal androgen receptor antagonist BMS-641988, holds potential for prostate cancer research.Formula:C20H20F3N3O5SPurity:98%Color and Shape:SolidMolecular weight:471.45JNJ-26146900
CAS:JNJ-26146900 is a nonsteroidal androgen receptor (AR) ligand with tissue-selective activity in rats. JNJ-26146900 binds to the rat AR with a K(i) of 400nM.Formula:C15H15F3N2O3SPurity:98%Color and Shape:SolidMolecular weight:360.35Trimegestone
CAS:Trimegestone, a highly effective oral progestogen, is used for endometrial protection, all doses inducing secretory endometrial transformation.Formula:C22H30O3Purity:98%Color and Shape:SolidMolecular weight:342.47YXG-158
CAS:YXG-158 (Compound 23-h), an orally active androgen receptor (AR) degrader and cytochrome P450 17A1 (CYP17A1) inhibitor, exhibits AR degradation with a DC50 of 1Formula:C30H36FN3OPurity:98%Color and Shape:SolidMolecular weight:473.62Androgen receptor degrader-3
CAS:Androgen Receptor Degrader-3 (ARD-3) is a compound that inhibits androgen receptor signaling and promotes the degradation of the receptor, with potentialFormula:C45H51ClN8O5Purity:98%Color and Shape:SolidMolecular weight:819.39PLK1/BRD4-IN-1
CAS:PLK1/BRD4-IN-1 (9b) is an orally active dual inhibitor of PLK1 (IC50: 22 nM) and BRD4 (IC50: 109 nM).Formula:C31H43N9O2Color and Shape:SolidMolecular weight:573.73Androgen receptor-IN-5
CAS:Androgen receptor-IN-5 is a potent inhibitor of the androgen receptor with anticancer properties.Formula:C22H10Cl2F4N4OSPurity:98%Color and Shape:SolidMolecular weight:525.31Androgen receptor degrader-1
CAS:Androgen Receptor Degrader-1 (Compound 18) is a potent agent for androgen receptor degradation, applicable in cancer research [1].Formula:C15H14ClN3O4Purity:98%Color and Shape:SolidMolecular weight:335.74JJH260
CAS:JJH260, a N-hydroxy hydantoin carbamate, inhibits AIG1 and ADTRP with IC50 values of 0.57 μM and 8.5 μM, respectively, and targets ABHD6, LYPLA1/2.Formula:C29H34ClN5O5Color and Shape:SolidMolecular weight:568.06EPI-7170
CAS:EPI-7170: Ralaniten analogue, blocks androgen receptor, inhibits transcription in AR & variants, fights enzalutamide-resistant prostate cancer.Formula:C22H28Cl3NO6SColor and Shape:SolidMolecular weight:540.88LGD-2941
CAS:LGD-2941 is an androgen receptor modulator. LGD-2941 is used for the treatment of hypogonadism, female sexual dysfunction and menopausal syndrome.Formula:C17H16F6N2O2Color and Shape:SolidMolecular weight:394.31RU 59063
CAS:RU 59063 is a prototype of a new class of high-affinity nonsteroidal androgen receptor (AR) ligands.Formula:C17H18F3N3O2SPurity:99.09%Color and Shape:SolidMolecular weight:385.4Ref: TM-T20761
1mg93.00€5mg182.00€10mg269.00€25mg429.00€50mg610.00€100mg820.00€200mg1,071.00€1mL*10mM (DMSO)197.00€
