Androgen Receptor
The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.
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ACP-105
CAS:899821-23-9
ACP-105 is a novel and potent nonsteroidal selective androgen receptor modulator (SARM) with partial agonist …
Formula:
C16H19ClN2O
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
290.79
Ref: TM-T14116
| 2mg | 37.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | 218.00 € | ||
| 100mg | 314.00 € | ||
| 200mg | 439.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
AS-601811
CAS:194979-95-8
AS-601811 is a bio-active chemical.
Formula:
C15H17NO
Purity:
98.05% - 99.49%
Color and Shape:
Solid
Molecular weight:
227.3
Ref: TM-T30150
| 1mg | 274.00 € | ||
| 5mg | 670.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,389.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,563.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
ARD-1676
CAS:2632305-36-1
ARD-1676 is an orally administered androgen receptor (AR) PROTAC degrader that combines an AR ligand …
Formula:
C44H46ClN7O5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
788.33
Ref: TM-T79725
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
(R)-SKBG-1
CAS:2955634-67-8
(R)-SKBG-1 is an inhibitor of the RNA-binding protein NONO, effectively downregulating androgen receptor expression by …
Formula:
C22H32ClN3O6S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
495.98
Ref: TM-T79156
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
BWA-522
BWA-522 is a small molecule, orally available protein-targeting chimera (PROTAC) that potentates the degradation of …
Formula:
C43H51ClN4O7
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
771.34
Ref: TM-T78810
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
BMS-986365
CAS:2446928-30-7
BMS-986365 (CC-94676) is an orally available, selective and highly potent AR degrader with potential anticancer …
Formula:
C41H45F3N8O5S
Purity:
98.77% - 99.96%
Color and Shape:
Soild
Molecular weight:
818.91
Ref: TM-T84297
| 1mg | 196.00 € | ||
| 5mg | 493.00 € | ||
| 10mg | 773.00 € | ||
| 25mg | 1,539.00 € | ||
| 50mg | 2,384.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Zanoterone
CAS:107000-34-0
Zanoterone is an AR antagonist (androgen receptor).Zanoterone has antitumor activity for the treatment of genitourinary …
Formula:
C23H32N2O3S
Purity:
99.85% - 99.96%
Color and Shape:
Soild
Molecular weight:
416.58
Ref: TM-T68020
| 1mg | 179.00 € | ||
| 5mg | 448.00 € | ||
| 10mg | 638.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,380.00 € | ||
| 100mg | 1,855.00 € | ||
| 500mg | 3,639.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
WCA-814
WCA-814, an androgen receptor (AR) antagonist-Hsp90 inhibitor conjugate, induces degradation of both full-length and AR-V7, …
Formula:
C46H53ClN10O5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
861.43
Ref: TM-T78945
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
MK-0773 FA
MK-0773 FA (MK-0773 FA (606101-58-0 Free base)) is an androgen receptor modulator used for the …
Formula:
C28H36FN5O4
Purity:
99.17%
Color and Shape:
Soild
Molecular weight:
525.61
Ref: TM-T16090L
| 1mg | 86.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
PROTAC AR-NTD degrader 1
PROTAC AR-NTD antagonist 1 (compound 18) is a small molecule belonging to the protein-targeting chimeras …
Formula:
C41H47ClN6O7
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
771.3
Ref: TM-T78811
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
ARD-2585
CAS:2757422-79-8
ARD-2585 is an orally active and selective androgen receptor PROTAC degrader with anticancer activity for …
Formula:
C41H43ClN8O5
Color and Shape:
Liquid
Molecular weight:
763.28
Ref: TM-T74141
| 1mg | 308.00 € | ||
| 5mg | 735.00 € | ||
| 10mg | 1,183.00 € | ||
| 25mg | 2,337.00 € | ||
| 50mg | 3,667.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
RD162
CAS:915087-27-3
RD162 is a non-steroidal antiandrogen (NSAA) specifically binding to the androgen receptor (AR).
Formula:
C22H16F4N4O2S
Purity:
97.74%
Color and Shape:
Solid
Molecular weight:
476.45
Ref: TM-T21740
| 1mg | 46.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 384.00 € | ||
| 50mg | 575.00 € | ||
| 100mg | 819.00 € | ||
| 1mL*10mM (DMSO) | 144.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Luxdegalutamide
CAS:2750830-09-0
Luxdegalutamide (ARV-766) is an orally available and effective protein degrader of protein hydrolysis-targeted chimeras (PROTAC).Luxdegalutamide …
Formula:
C45H54FN7O6
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
807.95
Ref: TM-T75129
| 1mg | 296.00 € | ||
| 5mg | 713.00 € | ||
| 10mg | 1,103.00 € | ||
| 25mg | 1,655.00 € | ||
| 50mg | 2,157.00 € | ||
| 100mg | 2,762.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Anticancer agent 135
Anticancer agent 135 (compound 26h) acts as a potent androgen receptor (AR) antagonist, effectively blocking …
Formula:
C23H21F3N4OS
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
458.5
Ref: TM-T79465
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
Masofaniten
CAS:2416716-62-4
Masofaniten (EPI-7386) is an orally active androgen receptor (AR) inhibitor with antitumor activity for the …
Formula:
C24H24Cl2N4O4S
Purity:
98.66%
Color and Shape:
Liquid
Molecular weight:
535.44
Ref: TM-T72985
| 25mg | 1,477.00 € | ||
| 50mg | 1,924.00 € | ||
| 100mg | 2,872.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
MK-0773
CAS:606101-58-0
MK-0773 (PF-05314882) is a selective androgen receptor modulator that binds to AR (IC50: 6.6 nM) …
Formula:
C27H34FN5O2
Purity:
99.36% - 99.63%
Color and Shape:
Solid
Molecular weight:
479.59
Ref: TM-T16090
| 1mg | 85.00 € | ||
| 5mg | 176.00 € | ||
| 10mg | 274.00 € | ||
| 1mL*10mM (DMSO) | 185.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Rezvilutamide
CAS:1572045-62-5
Rezvilutamide (SHR3680) is an orally available androgen receptor inhibitor that crosses the blood-brain barrier and …
Formula:
C22H20F3N3O4S
Purity:
99.97%
Color and Shape:
Solid
Molecular weight:
479.47
Ref: TM-T39044
| 1mg | 80.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
LY2452473
CAS:1029692-15-6
LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer …
Formula:
C22H22N4O2
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
374.44
Ref: TM-T15804
| 1mg | 45.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | 186.00 € | ||
| 100mg | 308.00 € | ||
| 500mg | 738.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Nandrolone phenylpropionate
CAS:62-90-8
Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women …
Formula:
C27H34O3
Purity:
99.46%
Color and Shape:
White Or Milky Crystalline Powder
Molecular weight:
406.56
Ref: TM-T8709
| 10mg | 43.00 € | ||
| 25mg | 61.00 € | ||
| 50mg | 85.00 € | ||
| 100mg | 112.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
DJ-V-159
CAS:2253744-53-3
DJ-V-159 is a GPRC6A agonist, targeting the G protein-coupled receptor family C group 6 member …
Formula:
C24H12F6N4O2
Purity:
99.85% - 99.96%
Color and Shape:
Solid
Molecular weight:
502.37
Ref: TM-T5100
| 2mg | 36.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 266.00 € | ||
| 100mg | 427.00 € | ||
| 500mg | 931.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
