Androgen Receptor
The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.
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Adrenosterone
CAS:382-45-6
Adrenosterone (11-ketoandrostenedione) is a steroid hormone isolated from the adrenal cortex.
Formula:
C19H24O3
Purity:
97.04% - 98.13%
Color and Shape:
Solid
Molecular weight:
300.39
Ref: TM-T2207
| 50mg | 47.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 14 Apr 2025
BWA-522
BWA-522 is a small molecule, orally available protein-targeting chimera (PROTAC) that potentates the degradation of …
Formula:
C43H51ClN4O7
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
771.34
Ref: TM-T78810
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Apr 2025
PROTAC AR-NTD degrader 1
PROTAC AR-NTD antagonist 1 (compound 18) is a small molecule belonging to the protein-targeting chimeras …
Formula:
C41H47ClN6O7
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
771.3
Ref: TM-T78811
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Anticancer agent 135
Anticancer agent 135 (compound 26h) acts as a potent androgen receptor (AR) antagonist, effectively blocking …
Formula:
C23H21F3N4OS
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
458.5
Ref: TM-T79465
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Apr 2025
(R)-SKBG-1
CAS:2955634-67-8
(R)-SKBG-1 is an inhibitor of the RNA-binding protein NONO, effectively downregulating androgen receptor expression by …
Formula:
C22H32ClN3O6S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
495.98
Ref: TM-T79156
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Gridegalutamide
CAS:2446929-86-6
Gridegalutamide exhibits anti-androgen and anti-tumor activities.
Formula:
C41H45F3N8O5S
Color and Shape:
Liquid
Molecular weight:
818.91
Ref: TM-T200967
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Apr 2025
BMS-986365
CAS:2446928-30-7
BMS-986365 (CC-94676) is an orally available, selective and highly potent AR degrader with potential anticancer …
Formula:
C41H45F3N8O5S
Purity:
98.77% - 99.96%
Color and Shape:
Soild
Molecular weight:
818.91
Ref: TM-T84297
| 1mg | 199.00 € | ||
| 5mg | 500.00 € | ||
| 10mg | 788.00 € | ||
| 25mg | 1,569.00 € | ||
| 50mg | 2,431.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Zanoterone
CAS:107000-34-0
Zanoterone is an AR antagonist (androgen receptor).Zanoterone has antitumor activity for the treatment of genitourinary …
Formula:
C23H32N2O3S
Purity:
99.85% - 99.96%
Color and Shape:
Soild
Molecular weight:
416.58
Ref: TM-T68020
| 1mg | 182.00 € | ||
| 5mg | 457.00 € | ||
| 10mg | 652.00 € | ||
| 25mg | 1,026.00 € | ||
| 50mg | 1,406.00 € | ||
| 100mg | 1,890.00 € | ||
| 500mg | 3,725.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
ARD-266
CAS:2666951-70-6
ARD-266 is a PROTAC degrader based on the von Hippel-Lindau E3 ligase that induces the …
Formula:
C52H59ClN6O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
915.51
Ref: TM-T13552
| 1mg | 705.00 € | ||
| 5mg | 1,549.00 € | ||
| 10mg | 2,431.00 € | ||
| 25mg | 3,617.00 € | ||
| 50mg | 4,882.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
ARD-1676
CAS:2632305-36-1
ARD-1676 is an orally administered androgen receptor (AR) PROTAC degrader that combines an AR ligand …
Formula:
C44H46ClN7O5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
788.33
Ref: TM-T79725
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Apr 2025
MK-0773 FA
MK-0773 FA (MK-0773 FA (606101-58-0 Free base)) is an androgen receptor modulator used for the …
Formula:
C28H36FN5O4
Purity:
99.17%
Color and Shape:
Soild
Molecular weight:
525.61
Ref: TM-T16090L
| 1mg | 87.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
ARD-2585
CAS:2757422-79-8
ARD-2585 is an orally active and selective androgen receptor PROTAC degrader with anticancer activity for …
Formula:
C41H43ClN8O5
Color and Shape:
Liquid
Molecular weight:
763.28
Ref: TM-T74141
| 1mg | 316.00 € | ||
| 5mg | 755.00 € | ||
| 10mg | 1,216.00 € | ||
| 25mg | 2,403.00 € | ||
| 50mg | 3,771.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Luxdegalutamide
CAS:2750830-09-0
Luxdegalutamide (ARV-766) is an orally available and effective protein degrader of protein hydrolysis-targeted chimeras (PROTAC).Luxdegalutamide …
Formula:
C45H54FN7O6
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
807.95
Ref: TM-T75129
| 1mg | 303.00 € | ||
| 5mg | 730.00 € | ||
| 10mg | 1,121.00 € | ||
| 25mg | 1,691.00 € | ||
| 50mg | 2,205.00 € | ||
| 100mg | 2,822.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
RD162
CAS:915087-27-3
RD162 is a non-steroidal antiandrogen (NSAA) specifically binding to the androgen receptor (AR).
Formula:
C22H16F4N4O2S
Purity:
97.74%
Color and Shape:
Solid
Molecular weight:
476.45
Ref: TM-T21740
| 1mg | 47.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 393.00 € | ||
| 50mg | 585.00 € | ||
| 100mg | 832.00 € | ||
| 1mL*10mM (DMSO) | 144.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
WCA-814
WCA-814, an androgen receptor (AR) antagonist-Hsp90 inhibitor conjugate, induces degradation of both full-length and AR-V7, …
Formula:
C46H53ClN10O5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
861.43
Ref: TM-T78945
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Apr 2025
AS-601811
CAS:194979-95-8
AS-601811 is a bio-active chemical.
Formula:
C15H17NO
Purity:
98.05% - 99.49%
Color and Shape:
Solid
Molecular weight:
227.3
Ref: TM-T30150
| 1mg | 279.00 € | ||
| 5mg | 683.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,415.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,612.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Masofaniten
CAS:2416716-62-4
Masofaniten (EPI-7386) is an orally active androgen receptor (AR) inhibitor with antitumor activity for the …
Formula:
C24H24Cl2N4O4S
Purity:
98.66%
Color and Shape:
Liquid
Molecular weight:
535.44
Ref: TM-T72985
| 25mg | 1,539.00 € | ||
| 50mg | 2,005.00 € | ||
| 100mg | 2,992.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Rezvilutamide
CAS:1572045-62-5
Rezvilutamide (SHR3680) is an orally available androgen receptor inhibitor that crosses the blood-brain barrier and …
Formula:
C22H20F3N3O4S
Purity:
99.97%
Color and Shape:
Solid
Molecular weight:
479.47
Ref: TM-T39044
| 1mg | 81.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Apr 2025
LY2452473
CAS:1029692-15-6
LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer …
Formula:
C22H22N4O2
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
374.44
Ref: TM-T15804
| 1mg | 46.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 160.00 € | ||
| 50mg | 188.00 € | ||
| 100mg | 311.00 € | ||
| 500mg | 747.00 € | ||
| 1mL*10mM (DMSO) | 97.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
MK-0773
CAS:606101-58-0
MK-0773 (PF-05314882) is a selective androgen receptor modulator that binds to AR (IC50: 6.6 nM) …
Formula:
C27H34FN5O2
Purity:
99.36% - 99.63%
Color and Shape:
Solid
Molecular weight:
479.59
Ref: TM-T16090
| 1mg | 162.00 € | ||
| 5mg | 329.00 € | ||
| 10mg | 474.00 € | ||
| 1mL*10mM (DMSO) | 187.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
