Androgen Receptor
The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.
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D4-abiraterone
CAS:154229-21-7
D4-Abiraterone is an inhibitor of CYP17A1, 3b-hydroxysteroid dehydrogenase (3βHSD) and steroid 5a-reductase (SRD5A), the main …
Formula:
C24H29NO
Color and Shape:
Solid
Molecular weight:
347.49
Ref: TM-T10946
| 1mg | 46.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Ligandrol
CAS:1165910-22-4
Ligandrol is a novel nonsteroidal, oral SARM that binds to the androgen receptor with high …
Formula:
C14H12F6N2O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
338.25
Ref: TM-T15750
| 25mg | 45.00 € | ||
| 50mg | 63.00 € | ||
| 100mg | 93.00 € | ||
| 200mg | 123.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
2,2,5,7,8-Pentamethyl-6-Chromanol
CAS:950-99-2
2,2,5,7,8-Pentamethyl-6-Chromanol (PMC) is the anti-oxidant moiety of vitamin E (α-tocopherol), which has potent androgen receptor …
Formula:
C14H20O2
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
220.31
Ref: TM-T14008
| 1g | 82.00 € | ||
| 500mg | 56.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Ostarine
CAS:841205-47-8
Ostarine (MK-2866) is a non-steroidal SARM mimicking testosterone to boost muscle growth, libido, fertility, and …
Formula:
C19H14F3N3O3
Purity:
99.35% - 99.9%
Color and Shape:
Solid
Molecular weight:
389.33
Ref: TM-T2408
| 25mg | 42.00 € | ||
| 50mg | 78.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
UT-34
CAS:2168525-92-4
UT-34 is a selective and orally active antagonist of second-generation pan-androgen receptor (AR) and degrader(IC50s …
Formula:
C15H12F4N4O2
Purity:
98.12%
Color and Shape:
Solid
Molecular weight:
356.27
Ref: TM-T13273
| 1mg | 52.00 € | ||
| 2mg | 80.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 621.00 € | ||
| 100mg | 891.00 € | ||
| 1mL*10mM (DMSO) | 130.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
ORM-15341
CAS:1297537-33-7
ORM-15341 is a potent and full antagonist for human AR (hAR)( with IC50 values of …
Formula:
C19H17ClN6O2
Purity:
98.01%
Color and Shape:
Solid
Molecular weight:
396.83
Ref: TM-T12323
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 296.00 € | ||
| 100mg | 443.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
SK33
CAS:1928724-23-5
SK33 is a potent and tissue selective anti-androgen agent. SK33 reduces androgen receptor (AR) transcriptional …
Formula:
C20H13F9N2O3
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
500.31
Ref: TM-T12928
| 1mg | 79.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 218.00 € | ||
| 25mg | 364.00 € | ||
| 50mg | 520.00 € | ||
| 100mg | 703.00 € | ||
| 200mg | 903.00 € | ||
| 1mL*10mM (DMSO) | 181.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Dehydroisoandrosterone 3-acetate
CAS:853-23-6
Dehydroisoandrosterone 3-acetate (Prasterone acetate) is a primary C19 steroid generated by the adrenal cortex.
Formula:
C21H30O3
Purity:
100% - 99.81%
Color and Shape:
Solid
Molecular weight:
330.46
Ref: TM-T0856
| 1g | 52.00 € | ||
| 500mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
N-Desmethyl-Apalutamide
CAS:1332391-11-3
N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.
Formula:
C20H13F4N5O2S
Purity:
97.83%
Color and Shape:
Solid
Molecular weight:
463.41
Ref: TM-T12146
| 1mg | 114.00 € | ||
| 5mg | 253.00 € | ||
| 10mg | 363.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 754.00 € | ||
| 100mg | 1,007.00 € | ||
| 200mg | 1,367.00 € | ||
| 1mL*10mM (DMSO) | 271.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Spironolactone
CAS:52-01-7
Spironolactone (SC9420) is an Aldosterone Antagonist. The mechanism of action of spironolactone is as an …
Formula:
C24H32O4S
Purity:
99.63%
Color and Shape:
White Powder
Molecular weight:
416.57
Ref: TM-T0476
| 50mg | 39.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Medroxyprogesterone Acetate
CAS:71-58-9
Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. Farlutin is a …
Formula:
C24H34O4
Purity:
99.45%
Color and Shape:
White Powder
Molecular weight:
386.52
Ref: TM-T1261
| 200mg | 36.00 € | ||
| 500mg | 47.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
3,3'-Diindolylmethane
CAS:1968-05-4
3,3'-Diindolylmethane (DIM), a small molecule compound, is a proposed Y preventive agent.
Formula:
C17H14N2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
246.31
Ref: TM-T2991
| 50mg | 46.00 € | ||
| 100mg | 57.00 € | ||
| 200mg | 67.00 € | ||
| 500mg | 87.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Bicalutamide
CAS:90357-06-5
Bicalutamide (ICI-176334), a synthetic, nonsteroidal antiandrogen, competitively binds to cytosolic androgen receptors in target tissues, …
Formula:
C18H14F4N2O4S
Purity:
98% - 99.97%
Color and Shape:
Off-White Crystalline Solid
Molecular weight:
430.37
Ref: TM-T0380
| 1g | 97.00 € | ||
| 50mg | 43.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 57.00 € | ||
| 500mg | 78.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Andarine
CAS:401900-40-1
Andarine (GTx-007) (S-4) is an active partial agonist and an investigational selective androgen receptor modulator …
Formula:
C19H18F3N3O6
Purity:
99.84%
Color and Shape:
Pale Yellow Solid
Molecular weight:
441.36
Ref: TM-T2108
| 5mg | 46.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 119.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Cyproterone acetate
CAS:427-51-0
Cyproterone acetate (Cyproterone 17-O-acetate) binds the androgen receptor (AR), thereby preventing androgen-induced receptor activation in …
Formula:
C24H29ClO4
Purity:
98.43%
Color and Shape:
Crystals From Diisopropyl Ether Odour
Molecular weight:
416.94
Ref: TM-T1167
| 100mg | 44.00 € | ||
| 250mg | 64.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Flutamide
CAS:13311-84-7
Flutamide (SCH 13521) is an antiandrogen with about the same potency as cyproterone in rodent …
Formula:
C11H11F3N2O3
Purity:
100% - 99.92%
Color and Shape:
Solid
Molecular weight:
276.21
Ref: TM-T0489
| 1g | 52.00 € | ||
| 5g | 90.00 € | ||
| 200mg | 35.00 € | ||
| 500mg | 50.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
UT-155
CAS:2031161-35-8
UT-155 is a selective and potent antagonist of the androgen receptor (AR) (Ki: 267 nM …
Formula:
C20H15F4N3O2
Purity:
98.94%
Color and Shape:
Solid
Molecular weight:
405.35
Ref: TM-T13272
| 1mg | 91.00 € | ||
| 2mg | 134.00 € | ||
| 5mg | 214.00 € | ||
| 10mg | 341.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 744.00 € | ||
| 100mg | 1,060.00 € | ||
| 500mg | 2,149.00 € | ||
| 1mL*10mM (DMSO) | 238.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Nilutamide
CAS:63612-50-0
Nilutamide, a nonsteroidal anti-androgen, treats prostate cancer by blocking androgen receptors, not affecting other hormone …
Formula:
C12H10F3N3O4
Purity:
98.45% - 98.67%
Color and Shape:
Crystalline Solid
Molecular weight:
317.22
Ref: TM-T0272
| 100mg | 51.00 € | ||
| 200mg | 64.00 € | ||
| 500mg | 88.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Vosilasarm
CAS:1182367-47-0
RAD140 is an investigational selective androgen receptor modulator (SARM) for the treatment of conditions such …
Formula:
C20H16ClN5O2
Purity:
99.01%
Color and Shape:
A Crystalline Solid
Molecular weight:
393.82
Ref: TM-T4358
| 2mg | 39.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 136.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Adrenosterone
CAS:382-45-6
Adrenosterone (11-ketoandrostenedione) is a steroid hormone isolated from the adrenal cortex.
Formula:
C19H24O3
Purity:
97.04% - 98.13%
Color and Shape:
Solid
Molecular weight:
300.39
Ref: TM-T2207
| 50mg | 51.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
