
Enzyme
Enzyme inhibitors are molecules that bind to enzymes and decrease their activity. These inhibitors are widely used in research to study enzyme kinetics, regulation, and the role of specific enzymes in metabolic pathways. Enzyme inhibitors are also crucial in drug development, as many therapeutic agents function by inhibiting enzymes involved in disease processes. By targeting enzymes, these inhibitors can modulate biochemical pathways and offer potential treatments for various diseases. At CymitQuimica, we provide a comprehensive selection of high-quality enzyme inhibitors to support your research in biochemistry, pharmacology, and drug discovery.
Subcategories of "Enzyme"
- Carbonic Anhydrase(178 products)
- Hydroxylase(30 products)
- MPO(2 products)
- Reductase(52 products)
- Tyrosinase(67 products)
Found 3587 products of "Enzyme"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
hCAIX-IN-8
CAS:<p>hCAIX-IN-8, a selective hCAIX inhibitor, IC50: 0.024 μM. Also affects CAII, CAVA (IC50s: 1.99, 1.10 μM), limits cell migration, and induces apoptosis.</p>Formula:C19H16N4O6Color and Shape:SolidMolecular weight:396.35hCAIX-IN-5
CAS:<p>hCAIX-IN-5 was a selective hCAIX inhibitor, inhibiting hCAI, hCAII, hCAIV, and hCAIX with Ki values of >10000, >10000, 130.7, and 829.1 nM, respectively.</p>Formula:C18H12FNO3Purity:99.26%Color and Shape:SolidMolecular weight:309.29AHR-15010
CAS:<p>AHR-15010 is a novel anti-arthritic agent.</p>Formula:C10H16N2O8S2Purity:98%Color and Shape:SolidMolecular weight:356.37hCAIX-IN-7
CAS:<p>hCAIX-IN-7 (6c) selectively inhibits tumor-related isoform hCAIX (KI: 410.6 nM) and weakly affects hCAI/II (KI: >10000 nM).</p>Formula:C18H12FNO3Color and Shape:SolidMolecular weight:309.29CDK2-IN-11
CAS:<p>CDK2-IN-11 inhibits CDK2 (IC50: 6.4 μM) and targets hCA II, IX, XII (Ki: 23.4-56.3 nM); suited for cancer research.</p>Formula:C18H14ClN7O2SColor and Shape:SolidMolecular weight:427.87Carbonic anhydrase inhibitor 13
CAS:<p>Carbonic anhydrase inhibitor 13 (compound 7) is a potent inhibitor of carbonic anhydrase (CA).</p>Formula:C17H15N5O3S2Color and Shape:SolidMolecular weight:401.46Carbonic anhydrase inhibitor 11
CAS:<p>Potent carbonic anhydrase inhibitor VI targets CA II, IX, XII with Ki: 40, 39, 900 nM respectively.</p>Formula:C19H15F3N4O3S2Color and Shape:SolidMolecular weight:468.47hCAIX/XII-IN-4
CAS:<p>hCAIX/XII-IN-4 inhibits CAIX/XII with Ki: 4.5 nM (CAXII), 23.6 nM (CAIX), and >10000 nM (CAI/CAII).</p>Formula:C20H16N2O5Color and Shape:SolidMolecular weight:364.35hCAII-IN-2
CAS:<p>hCAII-IN-2 inhibits human carbonic anhydrases I, II, IX, XII with Ki values of 261.4, 3.8, 19.6, 45.2 nM respectively.</p>Formula:C25H18ClN5O4SColor and Shape:SolidMolecular weight:519.96PGDS Protein, Human, Recombinant
<p>Hematopoietic Prostaglandin D Synthase (HPGDS) belongs to the GST superfamily and Sigma family.</p>Color and Shape:Lyophilized PowderMolecular weight:26 KDa (reducing condition)hCAIX-IN-3
CAS:<p>hCAII-IN-3 (7e) selectively inhibits CA II/IX with Kis of 124.2/30.5 nM, showing promise for cancer treatment.</p>Formula:C21H21BrN6O4SColor and Shape:SolidMolecular weight:533.4hCAIX-IN-14
CAS:<p>hCAIX-IN-14 is a potent inhibitor of human CA IX with a K i value of 134.8 nM .</p>Formula:C11H17ClN6O2SColor and Shape:SolidMolecular weight:332.81Carbonic anhydrase inhibitor 7
CAS:<p>Potent hCA inhibitor; targets hCA IX, II, XII, I with Ki: 6.5, 7.1, 72.1, 255.8 nM respectively.</p>Formula:C23H17N3O5SColor and Shape:SolidMolecular weight:447.46hCAXII-IN-1
CAS:<p>hCAXII-IN-1 selectively inhibits HCA IX/XII, promising for new cancer drug development.</p>Formula:C20H17NO5Color and Shape:SolidMolecular weight:351.35hCA I-IN-2
CAS:<p>hCA I-IN-2 (6d) inhibits hCA I (Ki: 18.8 nM) more selectively over II, IX, XII (Ki: 375.1, 1721, 283.9 nM).</p>Formula:C26H20BrN5O3SColor and Shape:SolidMolecular weight:562.44hCA I-IN-1
CAS:<p>hCA I-IN-1 inhibits hCA I (Ki: 38.3 nM), II (Ki: 716.4 nM), IX (Ki: 940.1 nM), XII (Ki: 192.8 nM).</p>Formula:C27H23N5O4SColor and Shape:SolidMolecular weight:513.57CDK2-IN-12
CAS:<p>CDK2-IN-12 (10b), potent CDK2 inhibitor, IC50: 11.6 μM; inhibits hCA I/II/IX/XII, KI: 3534/638.4/44.3/48.8 nM; anti-cancer properties.</p>Formula:C20H17N9O2SColor and Shape:SolidMolecular weight:447.47hCAIX/XII-IN-3
CAS:<p>Compound 6q inhibits hCAIX/CAXII; K i : hCAI >10000 nM, hCAII >10000 nM, hCAIX 66.2 nM, hCAXII 4.4 nM.</p>Formula:C20H13F3N2O4Color and Shape:SolidMolecular weight:402.32FC11409B
CAS:<p>FC11409B is a CAIX inhibitor, inhibiting breast cancer invasion and metastasis.</p>Formula:C29H23BF4N2O3SColor and Shape:SolidMolecular weight:566.38Disulfamide
CAS:<p>Disulfamide: Oral carbonic anhydrase inhibitor, IC50 0.07 μM, diuretic by blocking Na+/HCO3- reabsorption.</p>Formula:C7H9ClN2O4S2Purity:98.1%Color and Shape:SolidMolecular weight:284.74
