ERK
ERK is a key protein in the MAPK (Mitogen-Activated Protein Kinase) signaling pathway, which is involved in transmitting signals from cell surface receptors to the DNA in the cell nucleus. ERK plays a crucial role in the regulation of various cellular processes, including proliferation, differentiation, and survival. Dysregulation of ERK signaling is associated with the development of cancer and other diseases, making it an important target for therapeutic intervention. At CymitQuimica, we offer a selection of high-quality ERK inhibitors and modulators to support your research in cell signaling, oncology, and therapeutic development.
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ERK1/2 inhibitor 9
CAS:2169302-75-2
ERK1/2 Inhibitor 9 (Probe 1), a covalent antagonist of ERK1/2, exhibits sub-micromolar efficacy in cellular …
Formula:
C31H32ClN7O3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
586.08
Ref: TM-T78190
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 3 Feb 2025
Laxiflorin B
CAS:165337-71-3
Laxiflorin B, a novel selective inhibitor of ERK 1/2 derived from herbal sources, exhibits antitumor …
Formula:
C20H24O5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
344.4
Ref: TM-T79785
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 3 Feb 2025
MEK-IN-6
CAS:2845151-86-0
MEK-IN-6 (Example 69), a potent MEK inhibitor, effectively inhibits ERK1/2 (Thr202/Tyr204) phosphorylation in A375 cells, …
Formula:
C18H20FN3O4S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
393.43
Ref: TM-T79047
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
MK-8353
CAS:1184173-73-6
MK-8353 (SCH900353) is a potent, selective and orally available inhibitor of ERK1/2 (IC50s of 23.0 …
Formula:
C37H41N9O3S
Purity:
96.15% - 99.89%
Color and Shape:
Solid
Molecular weight:
691.84
Ref: TM-T12069
| 1mg | 79.00 € | ||
| 5mg | 153.00 € | ||
| 10mg | 268.00 € | ||
| 25mg | 451.00 € | ||
| 50mg | 655.00 € | ||
| 100mg | 933.00 € | ||
| 1mL*10mM (DMSO) | 229.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
ERK-IN-2
CAS:2743576-56-7
ERK-IN-2, an ERK2 inhibitor, exhibits an IC50 value of 1.8 nM. At doses greater than …
Formula:
C16H18ClN5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
347.8
Ref: TM-T11225
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Ergosterol peroxide
CAS:2061-64-5
Ergosterol peroxide inhibits osteoclasts, has antiviral/antitumor effects, stimulates Foxo3a, and may prevent renal fibrosis.
Formula:
C28H44O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
428.65
Ref: TM-TMA1743
| 1mg | 361.00 € | ||
| 5mg | 1,404.00 € | ||
| 500µg | 188.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
12(S)-HETE
CAS:54397-83-0
12(S)-HETE, made by platelets, promotes tumor cell adhesion to endothelium and matrix at 0.1μM-181M.
Formula:
C20H32O3
Color and Shape:
Solid
Molecular weight:
320.47
Ref: TM-T37047
| 10µg | 404.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
KU004
CAS:1260401-93-1
KU004, a potent dual EGFR/HER2 inhibitor, exhibits anticancer properties. It inhibits the proliferation of human …
Formula:
C29H27ClFN4O2P
Color and Shape:
Liquid
Molecular weight:
548.98
Ref: TM-T89998
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 3 Mar 2025
SJ-C1044
CAS:2121503-76-0
SJ-C1044 is an orally effective pan-RAF inhibitor demonstrating immunomodulatory and antitumor activities. It targets wild-type …
Formula:
C25H14F7N7O
Color and Shape:
Liquid
Molecular weight:
561.41
Ref: TM-T200357
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 3 Mar 2025
DOR agonist 2
CAS:1212540-02-7
Compound 3 (DOR agonist 2) acts as a Delta Opioid Receptor agonist. It inhibits the …
Formula:
C29H26N2O3
Color and Shape:
Liquid
Molecular weight:
450.53
Ref: TM-T200382
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 3 Mar 2025
ERK2 IN-1
CAS:1093061-47-2
ERK2 IN-1 is a selective ERK2 inhibitor with an IC50 of 7 nM.
Formula:
C36H34FN7O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
647.76
Ref: TM-T11228
| 25mg | 2,106.00 € | ||
| 50mg | 2,785.00 € | ||
| 100mg | 3,739.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Rineterkib
CAS:1715025-32-3
Rineterkib (ERK-IN-1) is an inhibitor of RAF and ERK1/2 activating mutations in the MAPK pathway.
Formula:
C26H27BrF3N5O2
Purity:
98.4%
Color and Shape:
Solid
Molecular weight:
578.42
Ref: TM-T11224
| 1mg | 96.00 € | ||
| 5mg | 190.00 € | ||
| 10mg | 357.00 € | ||
| 25mg | 604.00 € | ||
| 50mg | 860.00 € | ||
| 100mg | 1,170.00 € | ||
| 1mL*10mM (DMSO) | 252.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
