CGRP Receptor
CGRP receptors are involved in the transmission of pain and the regulation of blood flow. CGRP is a neuropeptide that plays a critical role in migraine pathophysiology by dilating blood vessels and modulating pain signaling pathways. Targeting CGRP receptors has become a promising approach in the development of migraine therapies. At CymitQuimica, we offer a range of CGRP receptor modulators to support your research in pain management, neurobiology, and vascular health.
Found 56 products for "CGRP Receptor".
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CRSP-1
CAS:Central CT receptor agonist, 350x stronger than CT, no CGRP or adrenomedullin action, inhibits osteoclasts, affects rat feeding, body temp, and calcium.Formula:C175H294N54O49S5Purity:98%Color and Shape:SolidMolecular weight:4098.88Cagrilintide acetate
.Cagrilintide is a long-acting amylin analog,treat diabetes and obesity by reducing appetite through activation of the AMY3R and calcitonin receptor.Formula:C196H316N54O61S2Purity:99.88%Color and Shape:White SolidMolecular weight:4469.06β-CGRP (mouse)
β-CGRP (mouse), a calcitonin gene-related peptide, induces vasodilation and is applicable in research areas including cardiovascular, pro-inflammatory, migraine, and metabolic studies.Formula:C165H265N49O55S2Color and Shape:SolidMolecular weight:3879.29CGRP 8-37 (rat)
CAS:CGRP 8-37 (rat) is a CGRP receptor antagonist, a CGRP fragment with potential anti-injury effects that induces arterial relaxation.Formula:C138H224N42O41Purity:99.28%Color and Shape:SolidMolecular weight:3127.51Adrenomedullin (AM) (22-52), human acetate
Adrenomedullin (AM) (22-52), human acetate is an antagonist of calcitonin generelated peptide receptor in the hindlimb vascular bed of the cat and anFormula:C161H256N46O50Purity:99.42%Color and Shape:SolidMolecular weight:3636.09α-CGRP (mouse, rat) TFA
α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is predominantly located at neuromuscular junctions andFormula:C162H262N50O52S2·C2HF3O2Purity:98%Color and Shape:SolidGalcanezumab
CAS:Galcanezumab: humanized IgG4 antibody that targets CGRP for migraine and cluster headache prevention/treatment.Purity:> 95%Color and Shape:LiquidMolecular weight:144.08 kDaUbrogepant-D5
Ubrogepant-D5 is the deuterium-labeled version of Ubrogepant. It is an orally active and selective antagonist of the calcitonin gene-related peptide receptor (CGRP). Ubrogepant (T17194) exhibits high affinity for CGRP receptors in humans and rhesus monkeys, effectively blocking the cAMP response induced by α-CGRP stimulation. This compound is utilized in studies focused on acute migraine.Color and Shape:Odour SolidCGRP antagonist 6
CGRP Antagonist 6 (Compound 23) is a potent CGRP receptor antagonist (Ki: 0.84 nM). It is utilized in the study of migraines.Color and Shape:Odour SolidAdrenomedullin (1-50), rat
CAS:Rat adrenomedullin (1-50) is a 50-AA peptide; induces arterial vasodilation by activating CGRP1 receptors.Formula:C248H381N77O75S5Purity:98%Color and Shape:SolidMolecular weight:5729.5Adrenomedullin (AM) (22-52), human
CAS:Adrenomedullin (ADM) is a 52-aa hypotensive peptide. Adrenomedullin (ADM) has structural similarity with amylin.Formula:C159H252N46O48Purity:98%Color and Shape:SolidMolecular weight:3576.04HCGRP-(8-37)
CAS:Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selective CGRP receptor antagonistFormula:C139H230N44O38Purity:98%Color and Shape:SolidMolecular weight:3125.59Calcitonin (human)
CAS:Endogenous calcitonin receptor agonist. Lowers systemic blood calcium levels and inhibits bone resorption.Formula:C151H226N40O45S3Purity:98%Color and Shape:White Lyophilized PowderMolecular weight:3417.87SUN B8155
CAS:SUN B8155 is a CT receptor agonist that induces cAMP formation in cells expressing recombinant human CT receptor.Formula:C14H15N3O3Purity:99.38% - 99.99%Color and Shape:Yellow SolidMolecular weight:273.29Telcagepant
CAS:Telcagepant (MK-0974) is an oral calcitonin gene-related peptide receptor (CGRP) antagonist that blocks CGRP receptors, migraines and for pain relief.Formula:C26H27F5N6O3Purity:98.98% - 98.98%Color and Shape:SolidMolecular weight:566.52Calcitonin (salmon)
CAS:Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.Formula:C145H240N44O48S2Purity:99.41% - 99.80%Color and Shape:SolidMolecular weight:3431.85Olcegepant
CAS:Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4Formula:C38H47Br2N9O5Purity:96.08% - 97.24%Color and Shape:SolidMolecular weight:869.65Calcitonin(salmon) Acetate(47931-85-1(free base))
Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5Formula:C147H243N44O50S2Purity:99.29% - 99.63%Color and Shape:White SolidMolecular weight:3490.94Vazegepant hydrochloride
CAS:Vazegepant hydrochloride (Vazegepant HCl) is the first intranasal gepant for the acute treatment of migraine and has announced a positive phase II/III study.Formula:C36H47ClN8O3Purity:98.93%Color and Shape:White SolidMolecular weight:675.3Ref: TM-T8682
1mg102.00€5mg215.00€1mL*10mM (DMSO)313.00€10mg316.00€25mg535.00€50mg763.00€100mg1,054.00€BCTC
CAS:BCTC is a potent TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 (IC50 of 35 and 6 nM, respectively)Formula:C20H25ClN4OPurity:99.21% - 99.74%Color and Shape:White SolidMolecular weight:372.89
