CGRP Receptor
CGRP receptors are involved in the transmission of pain and the regulation of blood flow. CGRP is a neuropeptide that plays a critical role in migraine pathophysiology by dilating blood vessels and modulating pain signaling pathways. Targeting CGRP receptors has become a promising approach in the development of migraine therapies. At CymitQuimica, we offer a range of CGRP receptor modulators to support your research in pain management, neurobiology, and vascular health.
Found 51 products of "CGRP Receptor"
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Adrenomedullin (AM) (22-52), human acetate
Adrenomedullin (AM) (22-52), human acetate is an antagonist of calcitonin generelated peptide receptor in the hindlimb vascular bed of the cat and anFormula:C161H256N46O50Purity:99.42%Color and Shape:SolidMolecular weight:3636.09Calcitonin Gene Related Peptide (CGRP) II, rat
CAS:CGRP II is a potent vasodilator that boosts pancreatic enzyme levels by activating β-cell receptors.Formula:C163H267N51O50S2Purity:98%Color and Shape:SolidMolecular weight:3805.31Adrenomedullin (11-50), rat
CAS:Adrenomedullin 11-50 rat is a peptide, stimulates CGRP1 receptor for vasodilation, used in bone growth research.Formula:C194H304N58O59S4Purity:98%Color and Shape:SolidMolecular weight:4521.17HTL22562
CAS:HTL22562 is a calcitonin gene-related peptide (CGRP) receptor antagonist for acute treatment of migraine.Formula:C40H49N11O5Color and Shape:SolidMolecular weight:763.904α-CGRP(human)
CAS:Endogenous calcitonin gene-related peptide receptor (CGRP) agonist.Formula:C163H267N51O49S2Purity:98%Color and Shape:SolidMolecular weight:3789.33Adrenomedullin (16-31), human
CAS:Adrenomedullin (16-31), human is amino acid residues 16-31 fragment of human adrenomedullin (hADM).Formula:C82H129N25O21S2Purity:98%Color and Shape:SolidMolecular weight:1865.19CGRP 8-37 (rat)
CAS:CGRP 8-37 (rat) is a CGRP receptor antagonist, a CGRP fragment with potential anti-injury effects that induces arterial relaxation.Formula:C138H224N42O41Purity:99.28%Color and Shape:SolidMolecular weight:3127.51α-CGRP(human) TFA
α-CGRP(human) TFA is a 37-amino acid regulatory neuropeptide that is extensively located within the central and peripheral nervous system, functioning as aFormula:C165H268F3N51O51S2Color and Shape:SolidMolecular weight:3903.33Adrenomedullin (16-31), human TFA
Human adrenomedullin (16-31) TFA, fragment 16-31, binds CGRP1 receptor, raises rat blood pressure, not cats’.Formula:C84H130F3N25O23S2Color and Shape:SolidMolecular weight:1979.21Telcagepant
CAS:Telcagepant (MK-0974) is an oral calcitonin gene-related peptide receptor (CGRP) antagonist that blocks CGRP receptors, migraines and for pain relief.Formula:C26H27F5N6O3Purity:98.98% - 98.98%Color and Shape:SolidMolecular weight:566.52SUN B8155
CAS:SUN B8155 is a CT receptor agonist that induces cAMP formation in cells expressing recombinant human CT receptor.Formula:C14H15N3O3Purity:99.38% - 99.38%Color and Shape:SolidMolecular weight:273.29Calcitonin (salmon)
CAS:Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.Formula:C145H240N44O48S2Purity:99.41% - 99.80%Color and Shape:PowderMolecular weight:3431.85BCTC
CAS:BCTC is a potent TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 (IC50 of 35 and 6 nM, respectively)Formula:C20H25ClN4OPurity:99.21%Color and Shape:SolidMolecular weight:372.89β-CGRP, human acetate
β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptorFormula:C164H271N51O50S3Purity:99.35%Color and Shape:SolidMolecular weight:3853.46Rimegepant
CAS:View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.Cited in 1 publications.Formula:C28H28F2N6O3Purity:99.1% - 99.99%Color and Shape:SolidMolecular weight:534.56Olcegepant
CAS:Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4Formula:C38H47Br2N9O5Purity:96.08% - 97.24%Color and Shape:SolidMolecular weight:869.65Vazegepant hydrochloride
CAS:Vazegepant hydrochloride (Vazegepant HCl) is the first intranasal gepant for the acute treatment of migraine and has announced a positive phase II/III study.Formula:C36H47ClN8O3Purity:98.93%Color and Shape:SolidMolecular weight:675.3Ref: TM-T8682
1mg107.00€5mg227.00€10mg334.00€25mg565.00€50mg805.00€100mg1,111.00€1mL*10mM (DMSO)329.00€Calcitonin(salmon) Acetate(47931-85-1(free base))
Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5Formula:C145H240N44O48S2Purity:99.29%Color and Shape:SolidMolecular weight:3431.85HCGRP-(8-37) acetate
HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor.Formula:C141H234N44O40Purity:99.29%Color and Shape:SolidMolecular weight:3185.64Atogepant
CAS:Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist for the study of migraine.Formula:C29H23F6N5O3Purity:99.66%Color and Shape:SolidMolecular weight:603.52Ref: TM-T26682
1mg147.00€5mg250.00€10mg313.00€25mg620.00€50mg1,108.00€100mg1,611.00€200mg2,178.00€1mL*10mM (DMSO)334.00€
