CGRP Receptor
CGRP receptors are involved in the transmission of pain and the regulation of blood flow. CGRP is a neuropeptide that plays a critical role in migraine pathophysiology by dilating blood vessels and modulating pain signaling pathways. Targeting CGRP receptors has become a promising approach in the development of migraine therapies. At CymitQuimica, we offer a range of CGRP receptor modulators to support your research in pain management, neurobiology, and vascular health.
Found 51 products of "CGRP Receptor"
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Eptinezumab
CAS:Eptinezumab is a humanised monoclonal antibody targeting CGRP (calcitonin gene-related peptide), which prevents CGRP binding to its receptor, migraine.
Purity:95% - 95%Color and Shape:LiquidSB 268262
CAS:CGRP1 antagonistFormula:C18H15N3O4S2Purity:98%Color and Shape:SolidMolecular weight:401.46CGRP antagonist 1
CAS:CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for theFormula:C29H26N4O4Purity:99.55%Color and Shape:SolidMolecular weight:494.54Ubrogepant
CAS:Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in the acute treatment of migraine studies.Formula:C29H26F3N5O3Purity:99.452% - 99.78%Color and Shape:SolidMolecular weight:549.54Ref: TM-T17194
1mg153.00€5mg378.00€10mg597.00€25mg929.00€50mg1,225.00€100mg1,681.00€1mL*10mM (DMSO)455.00€CGRP antagonist 7
CAS:CGRP antagonist 7 is a potent calcitonin gene-related peptide receptor (CGRP) antagonist with a Ki value of 0.029 nM. It effectively inhibits CGRP receptor-mediated cyclic adenosine monophosphate (cAMP) production, with an IC50 value of 1.5 nM. This compound is useful in migraine research.Formula:C30H32FN5O3Color and Shape:SolidMolecular weight:529.61Rimegepant sulfate hydrate
CAS:Rimegepant (BMS-927711/BHV-3000): oral CGRP blocker for migraines, effective without vasoconstriction, beats placebo, well-tolerated.Formula:C56H64F4N12O13SColor and Shape:SolidMolecular weight:1221.2526DNA crosslinker 6
CAS:DNA crosslinker 6 (compound 1) is an anti-mitotic agent known for its strong binding affinity to AT-DNA and inhibition of AT-hook 1 binding to DNA (IC50=0.03 µM). Additionally, it exhibits anti-protozoal activity, effectively inhibiting T. brucei with an EC50 of 0.83 µM.Formula:C19H21N7OColor and Shape:SolidMolecular weight:363.42MK-3207 Hydrochloride
CAS:MK-3207 Hydrochloride (MK-3207 HCl) is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 nM and 0.022 nM, highly selective versus human AM1, AM2, CTR, and AMY3. Phase 2.Formula:C31H30ClF2N5O3Purity:98.19%Color and Shape:SolidMolecular weight:594.05MK-3207
CAS:MK-3207 is a potent, oral CGRP receptor antagonist with high selectivity for human and monkey receptors, inhibiting blood flow in vivo.Formula:C31H29F2N5O3Color and Shape:SolidMolecular weight:557.59MK-8825
CAS:MK-8825 is a CGRP receptor antagonist.Formula:C31H30F2N6O3Color and Shape:SolidMolecular weight:572.61BI-44370
CAS:BI-44370, a CGRP (calcitonin gene-related peptide) receptor antagonist, can be used to treat migraines and other chronic pain.Formula:C35H47N5O6Color and Shape:SolidMolecular weight:633.78
