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CGRP Receptor

CGRP Receptor

CGRP receptors are involved in the transmission of pain and the regulation of blood flow. CGRP is a neuropeptide that plays a critical role in migraine pathophysiology by dilating blood vessels and modulating pain signaling pathways. Targeting CGRP receptors has become a promising approach in the development of migraine therapies. At CymitQuimica, we offer a range of CGRP receptor modulators to support your research in pain management, neurobiology, and vascular health.

Found 56 products for "CGRP Receptor".

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  • Calcitonin (salmon) Acetate
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    Calcitonin (salmon) Acetate

    Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5
    Formula:C147H243N44O50S2
    Purity:99.29% - 99.63%
    Color and Shape:White Solid
    Molecular weight:3490.94

    Ref: TM-TP1040L

  • HCGRP-(8-37) acetate
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    HCGRP-(8-37) acetate

    HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor.
    Formula:C141H234N44O40
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:3185.64

    Ref: TM-TP1134L

  • Atogepant
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    Atogepant

    CAS:
    Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist for the study of migraine.
    Formula:C29H23F6N5O3
    Purity:99.77% - 99.78%
    Color and Shape:Solid
    Molecular weight:603.515

    Ref: TM-T26682

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    Fremanezumab

    CAS:
    Fremanezumab (TEV-48125) is a humanised monoclonal antibody targeting CGRP, capable of neutralising human, mouse and rat CGRP, migraine.
    Purity:97.6% (SDS-PAGE); 95.9% (SEC-HPLC) - 97.6% (SDS-PAGE); 95.9% (SEC-HPLC)
    Color and Shape:Transparent Liquid
    Molecular weight:145.49 kDa (Predicted)

    Ref: TM-T76680

  • Eptinezumab
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    Eptinezumab

    CAS:
    Eptinezumab is a humanised monoclonal antibody targeting CGRP (calcitonin gene-related peptide), which prevents CGRP binding to its receptor, migraine.
    Purity:96.9% (SDS-PAGE); 99.8% (SEC-HPLC) - 96.9% (SDS-PAGE); 99.8% (SEC-HPLC)
    Color and Shape:Transparent Liquid
    Molecular weight:143.27 kDa (Predicted)

    Ref: TM-T76678

  • SB 268262
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    SB 268262

    CAS:
    CGRP1 antagonist
    Formula:C18H15N3O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.46

    Ref: TM-T23320

  • Calcitonin (salmon)
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    Calcitonin (salmon)

    CAS:
    Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.
    Formula:C145H240N44O48S2
    Purity:99.41% - 99.88%
    Color and Shape:Solid
    Molecular weight:3431.85

    Ref: TM-TP1040

  • CGRP antagonist 1
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    CGRP antagonist 1

    CAS:
    CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the
    Formula:C29H26N4O4
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:494.5411

    Ref: TM-T13453

  • β-CGRP, human
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    β-CGRP, human

    CAS:
    β-CGRP, human ,a 37-amino acid peptide,is the beta form of Calcitonin-gene-related peptide (β-CGRP), involved extensively in regulation of the cardiovascular
    Formula:C162H267N51O48S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3793.41

    Ref: TM-TP1130

  • Ubrogepant
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    Ubrogepant

    CAS:
    Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in the acute treatment of migraine studies.
    Formula:C29H26F3N5O3
    Purity:99.45% - 99.78%
    Color and Shape:Yellow Solid
    Molecular weight:549.5436

    Ref: TM-T17194

  • Rimegepant sulfate hydrate
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    Rimegepant sulfate hydrate

    CAS:
    Rimegepant (BMS-927711/BHV-3000): oral CGRP blocker for migraines, effective without vasoconstriction, beats placebo, well-tolerated.
    Formula:C56H64F4N12O13S
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:1221.2526

    Ref: TM-T70837

  • CGRP antagonist 7
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    CGRP antagonist 7

    CAS:
    CGRP antagonist 7 is a potent calcitonin gene-related peptide receptor (CGRP) antagonist with a Ki value of 0.029 nM. It effectively inhibits CGRP receptor-mediated cyclic adenosine monophosphate (cAMP) production, with an IC50 value of 1.5 nM. This compound is useful in migraine research.
    Formula:C30H32FN5O3
    Color and Shape:Solid
    Molecular weight:529.61

    Ref: TM-T211975

  • HTL22562
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    HTL22562

    CAS:
    HTL22562 is a calcitonin gene-related peptide (CGRP) receptor antagonist for acute treatment of migraine.
    Formula:C40H49N11O5
    Color and Shape:Solid
    Molecular weight:763.904

    Ref: TM-T39522

  • BI-44370
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    BI-44370

    CAS:
    BI-44370, a CGRP (calcitonin gene-related peptide) receptor antagonist, can be used to treat migraines and other chronic pain.
    Formula:C35H47N5O6
    Color and Shape:Solid
    Molecular weight:633.78

    Ref: TM-T26796

  • DNA crosslinker 6
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    DNA crosslinker 6

    CAS:
    DNA crosslinker 6 (compound 1) is an anti-mitotic agent known for its strong binding affinity to AT-DNA and inhibition of AT-hook 1 binding to DNA (IC50=0.03 µM). Additionally, it exhibits anti-protozoal activity, effectively inhibiting T. brucei with an EC50 of 0.83 µM.
    Formula:C19H21N7O
    Color and Shape:Solid
    Molecular weight:363.42

    Ref: TM-T201475

  • MK-3207 Hydrochloride
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    MK-3207 Hydrochloride

    CAS:
    MK-3207 Hydrochloride (MK-3207 HCl) is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 nM and 0.022 nM, highly selective versus human AM1, AM2, CTR, and AMY3. Phase 2.
    Formula:C31H30ClF2N5O3
    Purity:98.19%
    Color and Shape:Yellow Solid
    Molecular weight:594.051

    Ref: TM-T6590