Calcium Channel
Calcium channels are membrane proteins that regulate the flow of calcium ions into and out of cells, which is essential for various cellular functions, including muscle contraction, neurotransmitter release, and gene expression. Dysregulation of calcium channel activity is associated with conditions such as hypertension, cardiac arrhythmias, and neurological disorders. At CymitQuimica, we provide a wide selection of calcium channel modulators to support your research in cardiovascular health, neurobiology, and signal transduction.
Found 493 products of "Calcium Channel"
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BX430
CAS:<p>BX430 is used for chronic pain and cardiovascular disease and it is a potent and selective noncompetitive allosteric human P2X4 receptor channels antagonist</p>Formula:C15H15Br2N3OPurity:97.34%Color and Shape:SolidMolecular weight:413.11Trimethadione
CAS:<p>Trimethadione (3,5,5,-Trimethyloxazolidine-2,4-dione) is a dione-type anticonvulsant with antiepileptic activity.</p>Formula:C6H9NO3Purity:99.67% - >99.99%Color and Shape:SolidMolecular weight:143.145,5-Dimethyloxazolidine-2,4-dione
CAS:<p>5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.</p>Formula:C5H7NO3Purity:99.12%Color and Shape:Drypowder PelletslargecrystalsMolecular weight:129.11GSK-7975A
CAS:<p>GSK-7975A is a potent and orally available inhibitor of CRAC channel.</p>Formula:C18H12F5N3O2Purity:98.92%Color and Shape:SolidMolecular weight:397.3Bupivacaine hydrochloride
CAS:<p>Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.</p>Formula:C18H28N2O·HClPurity:99.9% - >99.99%Color and Shape:SolidMolecular weight:324.89Praziquantel
CAS:<p>Praziquantel (Droncit) is an anthelmintic that paralyzes worms by increasing calcium in muscle cells, causing tegument damage and immune response.</p>Formula:C19H24N2O2Purity:99.67% - 99.69%Color and Shape:SolidMolecular weight:312.41Ca2+ channel agonist 1
CAS:<p>Ca2+ channel agonist 1 activates N-type Ca2+ channels and inhibits Cdk2 (EC50: 14.23 μM/3.34 μM) for motor nerve issues.</p>Formula:C19H26N6OPurity:97.71%Color and Shape:SolidMolecular weight:354.45Caloxin 2A1 TFA
<p>Caloxin 2A1 TFA is a PM Ca2+ pump inhibitor that inhibits human red blood cell Ca2+-Mg2+-ATPase leakage.</p>Formula:C66H92F3N19O24Purity:99.89%Color and Shape:SolidMolecular weight:1592.55Strontium ranelate
CAS:<p>Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis and can slow the course of osteoarthritis of the knee.</p>Formula:C12H6N2O8S·2SrPurity:98.97%Color and Shape:Crystalline SolidMolecular weight:513.49GV-58
CAS:<p>GV-58 agonizes N/P-Q-type Ca2+ channels (EC50: 7.21/8.81 μM) with 20x less inhibition on CDK kinases.</p>Formula:C18H26N6OSPurity:97.36%Color and Shape:SolidMolecular weight:374.5Penfluridol
CAS:<p>Penfluridol (TLP-607) is a highly potent antipsychotic.</p>Formula:C28H27ClF5NOPurity:98.9% - 99.87%Color and Shape:Off-White To White Crystalline PowderMolecular weight:523.97Catharanthine tartrate
CAS:<p>Catharanthine tartrate (Catharanthine hemitartrate) is an alkaloid from periwinkle that inhibits voltage-gated L-type calcium channels and has antitumor effect.</p>Formula:C25H30N2O8Purity:99.91%Color and Shape:SolidMolecular weight:486.51PACAP-38 (31-38), human, mouse, rat
CAS:<p>PACAP-38 (31-38), human, mouse, rat demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal NPY and catecholamine production</p>Formula:C47H83N17O11Purity:98%Color and Shape:SolidMolecular weight:1062.27D-myo-Inositol-1,3-diphosphate (sodium salt)
CAS:<p>D-myo-Inositol-1,3-phosphate (Ins(1,3)P) is an inositol phosphate involved in cellular signal transduction.</p>Formula:C6H12Na2O12P2Color and Shape:SolidMolecular weight:384.08PACAP-38 (31-38), human, mouse, rat TFA
<p>PACAP-38 (31-38), human, mouse, rat (TFA) demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal.</p>Formula:C49H84F3N17O13Purity:98%Color and Shape:SolidMolecular weight:1176.29Nesiritide
CAS:<p>Nesiritide, recombinant human B-type natriuretic peptide, binds NPR-A/C with Kd 7.3/13 pM.</p>Formula:C143H244N50O42S4Purity:98%Color and Shape:SolidMolecular weight:3464.04NAADP tetrasodium salt
CAS:<p>Ca2+ mobilizing agent</p>Formula:C21H27N6O18P3Purity:98%Color and Shape:SolidMolecular weight:744.39NSC156529
CAS:<p>NSC156529 suppresses AKT1, reduces cancer cell growth in vitro, and inhibits prostate tumors in vivo.</p>Formula:C28H21ClS2Purity:98%Color and Shape:SolidMolecular weight:457.05D-myo-Inositol-1,3,4,5-tetraphosphate (sodium salt)
CAS:<p>Ins(1,3,4,5)-P4, made via Ins(1,4,5)P3 phosphorylation, boosts calcium by opening ER and plasma membrane channels.</p>Formula:C6H8Na8O18P4Color and Shape:SolidMolecular weight:675.93Triphenylethylene
CAS:<p>Compound PDK0283, with CAS No. 58-72-0, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0283 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Formula:C20H16Color and Shape:White PowderMolecular weight:256.34G-Glu-Ser
CAS:<p>G-Glu-Ser is a calcium receptor activator and Flavor-enriching agent.</p>Formula:C8H14N2O6Color and Shape:SolidMolecular weight:234.21Ryanodine
CAS:<p>Ryanodine: a diterpenoid modulating Ca2+ release via ryanodine receptors; concentration-dependent effects; found in Ryania speciosa; toxic.</p>Formula:C25H35NO9Purity:98%Color and Shape:White SolidMolecular weight:493.553BTT-266
CAS:<p>BTT-266 is a blocker of voltage-gated calcium channel for pain management.</p>Formula:C34H28N4O4Purity:98.34%Color and Shape:SolidMolecular weight:556.61ω-Conotoxin MVIIC
CAS:<p>Peptide neurotoxin; wide spectrum blocker of N, P and Q type calcium channels.</p>Formula:C106H178N40O32S7Purity:98%Color and Shape:White Lyophilised SolidMolecular weight:2749Ziconotide
CAS:<p>Ziconotide: analgesic from cone snail for severe, chronic pain; synthetic ω-conotoxin.</p>Formula:C102H172N36O32S7Purity:98%Color and Shape:White PowderMolecular weight:2639.13UK-59811 hydrochloride
CAS:<p>UK-59811 hydrochloride, Br-dihydropyridine derivative, blocks Ca V Ab channels in bacteria, IC50: 194 nM.</p>Formula:C22H30BrClN2O5Color and Shape:SolidMolecular weight:517.85Calcium Channel antagonist 3
CAS:<p>Calcium Channel antagonist 3 is a voltage-gated calcium channel inhibitor (IC50 : 5-20 μM).</p>Formula:C23H26N2O4SPurity:>99.99%Color and Shape:SolidMolecular weight:426.53Cavα2δ-IN-1
CAS:<p>Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a Ki</p>Formula:C18H27N5OColor and Shape:SolidMolecular weight:329.448ω-Conotoxin MVIIC TFA
<p>ω-Conotoxin MVIIC TFA is a peptide and neurotoxin blocks P-type and q-type voltage-sensitive neuronal Ca ++ channels (VGCCs) radiolabel immunoprecipitation.</p>Formula:C106H178N40O32S7·C2HF3O2Color and Shape:SolidMolecular weight:2863.27Elgodipine
CAS:<p>Elgodipine decreases angina severity, inhibits muscle growth, and is voltage-sensitive, showing promise for angina treatment.</p>Formula:C29H33FN2O6Purity:98.95% - 99.50%Color and Shape:SolidMolecular weight:524.58Mast cell degranulating peptide (28-49)
CAS:<p>Mast cell degranulating peptide (28-49) is a bee venom depolarizer that can improve the cGMP content of cerebellum tablets in mice.</p>Formula:C110H196N40O24S4Purity:98%Color and Shape:SolidMolecular weight:2591.25Calcium Channel antagonist 2
CAS:<p>Calcium Channel antagonist 2 is a calcium channel antagonist (IC50=5-20 μM) that can be used to study diseases due to Ca2+ channels like pain and diabetes.</p>Formula:C23H25FN2O4SPurity:99.34%Color and Shape:SolidMolecular weight:444.52Calcium Channel antagonist 4
CAS:<p>Calcium Channel antagonist 4 is a voltage-gated calcium channel inhibitor (IC50 : 5-20 μM).</p>Formula:C23H26N2O4SPurity:98.09%Color and Shape:SolidMolecular weight:426.53Chlorocresol
CAS:<p>Chlorocresol (4-Chloro-3-methylphenol) is an antiseptic medication.</p>Formula:C7H7ClOColor and Shape:SolidMolecular weight:142.58Candidalysin
CAS:<p>Candidalysin is a cytolytic peptide toxin initially isolated from *Candida albicans*, exhibiting both toxic and non-toxic properties. It activates epithelial cell signaling pathways by interacting with the epithelial growth factor receptor (EGFR) on host cells, leading to the activation of matrix metalloproteinases (MMP) and calcium ion influx, which results in inflammatory responses and immune cell recruitment. Additionally, Candidalysin exhibits cytotoxicity by causing membrane damage to host cells.</p>Formula:C153H266N38O38S2Color and Shape:SolidMolecular weight:3310.112-Nitrobenzoic acid
CAS:<p>2-Nitrobenzoic acid is an anti-growth agent with an IC50 of 8.3 μM against Jurkat cells with T-type Ca²⁺ channel alpha 1H/delta 25.</p>Formula:C7H5NO4Purity:99.97%Color and Shape:SoildMolecular weight:167.12ω-Conotoxin GVIA
CAS:<p>Peptide neurotoxin; selectively and reversibly blocks N-type calcium channels (IC50 = 0.15 nM). Reduces (RS)-3,5-DHPG -induced long term depression in vivo.</p>Formula:C120H182N38O43S6Purity:98%Color and Shape:SolidMolecular weight:3037Levamlodipine besylate Hemipentahydrate
CAS:<p>Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.</p>Formula:C20H25ClN2O5·C6H6O3SH2OColor and Shape:SolidMolecular weight:1224.18(±)5(6)-DiHETE
CAS:<p>Eicosapentaenoic acid is an ω-3 polyunsaturated fatty acid that is abundant in marine organisms and fish oils.</p>Formula:C20H32O4Color and Shape:SolidMolecular weight:336.472MMK 1
CAS:<p>Potent hFPR2 agonist; EC50: 1 nM (mFPR2), 2 nM (hFPR2), >10,000 nM (hFPR1). Induces monocyte/neutrophil migration, boosts IL-1β/IL-6, activates NADPH-oxidase.</p>Formula:C75H123N19O18SPurity:98%Color and Shape:SolidMolecular weight:1610.97Cyclic ADP-ribose ammonium
<p>cADPR ammonium is a second messenger that boosts cytosolic calcium via Ryanodine receptors and TRPM2 channels.</p>Color and Shape:LiquidSulcardine 2HCl
CAS:<p>Sulcardine 2HCl is a multi-ion channel blocker that blocks the properties of hERG and hNav1.5 channels and can be used to study atrial fibrillation.</p>Formula:C24H35Cl2N3O4SPurity:99.33% - 99.76%Color and Shape:SoildMolecular weight:532.523Kurtoxin
<p>Kurtoxin is a selective Cav3 (T-type) voltage-gated Ca2+ channel gating inhibitor, exhibiting a dissociation constant (Kd) of 15 nM for the Cav3.1 (α1G T-type)</p>Formula:C324H478N94O90S8Purity:98%Color and Shape:SolidMolecular weight:7386.36SG-094
CAS:<p>SG-094 inhibits TPC2, halts RIL175 cell growth, IC50: 3.7 μM for cancer research.</p>Formula:C30H29NO3Purity:97.06%Color and Shape:SoildMolecular weight:451.56Ethacrynic acid D5
CAS:<p>Ethacrynic acid: a diuretic, anti-inflammatory, inhibits calcium channels, GSTs, NF-kB pathway, and modulates leukotriene; has deuterium-labeled form.</p>Formula:C13H12Cl2O4Purity:98%Color and Shape:SolidMolecular weight:308.17(R)-IDHP
CAS:<p>(R)-IDHP, a salvia derivative, relaxes blood vessels by blocking calcium channels, aiding cardiovascular research.</p>Formula:C12H16O5Color and Shape:SolidMolecular weight:240.25KT-362 free base
CAS:<p>KT-362 is a calcium channel blocker with antihypertensive properties that can be used in the study of cardiovascular disease.</p>Formula:C22H28N2O3SPurity:99.76%Color and Shape:SoildMolecular weight:400.53Fasudil
CAS:<p>Fasudil (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.</p>Formula:C14H17N3O2SPurity:99.79% - 99.84%Color and Shape:SolidMolecular weight:291.37Ser-Ala-alloresact acetate
<p>Ser-Ala-alloresact acetate is a sperm-activating peptide (SAP) that is released by marine invertebrate eggs and plays an important role in fertilization.</p>Formula:C44H75N13O16S2Purity:99.73%Color and Shape:SolidMolecular weight:1106.281-(aminomethyl)cyclopropanecarboxylic acid hydrochloride
CAS:<p>1-(aminomethyl)cyclopropanecarboxylic acid hydrochloride inhibits L amino acid transporter proteins and the α2δ subunit of voltage-gated calcium channels.1-(</p>Formula:C5H10ClNO2Purity:>99.99%Color and Shape:SolidMolecular weight:151.59
