Calcium Channel
Calcium channels are membrane proteins that regulate the flow of calcium ions into and out of cells, which is essential for various cellular functions, including muscle contraction, neurotransmitter release, and gene expression. Dysregulation of calcium channel activity is associated with conditions such as hypertension, cardiac arrhythmias, and neurological disorders. At CymitQuimica, we provide a wide selection of calcium channel modulators to support your research in cardiovascular health, neurobiology, and signal transduction.
Found 573 products of "Calcium Channel"
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BX430
CAS:BX430 is used for chronic pain and cardiovascular disease and it is a potent and selective noncompetitive allosteric human P2X4 receptor channels antagonistFormula:C15H15Br2N3OPurity:97.34%Color and Shape:SolidMolecular weight:413.115,5-Dimethyloxazolidine-2,4-dione
CAS:5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.Formula:C5H7NO3Purity:99.12%Color and Shape:Drypowder PelletslargecrystalsMolecular weight:129.11CRAC intermediate 2
CAS:CRAC intermediate 2 is a intermediate compound for CRAC inhibitor synthesis.Formula:C11H7F6N3Purity:99.69%Color and Shape:SolidMolecular weight:295.18GSK-7975A
CAS:GSK-7975A is a potent and orally available inhibitor of CRAC channel.Formula:C18H12F5N3O2Purity:98.92%Color and Shape:SolidMolecular weight:397.3Ref: TM-T15423
1mg42.00€2mg55.00€5mg88.00€10mg130.00€25mg250.00€50mg378.00€100mg570.00€500mg1,189.00€1mL*10mM (DMSO)87.00€Nitrendipine
CAS:Nitrendipine is a vasodilating calcium channel blocker and antihypertensive that preserves kidney function and promotes sodium excretion.Formula:C18H20N2O6Purity:99% - 99.55%Color and Shape:SolidMolecular weight:360.36Ref: TM-T0119
1g414.00€10mg35.00€25mg52.00€50mg67.00€100mg113.00€200mg172.00€500mg268.00€1mL*10mM (DMSO)52.00€Caloxin 2A1 TFA
Caloxin 2A1 TFA is a PM Ca2+ pump inhibitor that inhibits human red blood cell Ca2+-Mg2+-ATPase leakage.Formula:C66H92F3N19O24Purity:99.89%Color and Shape:SolidMolecular weight:1592.55Strontium ranelate
CAS:Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis and can slow the course of osteoarthritis of the knee.Formula:C12H6N2O8S·2SrPurity:98.97%Color and Shape:Crystalline SolidMolecular weight:513.49Nimodipine
CAS:Nimodipine (BAY-e 9736), a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle cells.Formula:C21H26N2O7Purity:99.64% - 99.79%Color and Shape:SolidMolecular weight:418.44GV-58
CAS:GV-58 agonizes N/P-Q-type Ca2+ channels (EC50: 7.21/8.81 μM) with 20x less inhibition on CDK kinases.Formula:C18H26N6OSPurity:97.36%Color and Shape:SolidMolecular weight:374.5Ref: TM-T11517
1mg49.00€5mg137.00€10mg205.00€25mg409.00€50mg592.00€100mg827.00€500mg1,648.00€1mL*10mM (DMSO)150.00€Penfluridol
CAS:Penfluridol (TLP-607) is a highly potent antipsychotic.Formula:C28H27ClF5NOPurity:98.9% - 99.87%Color and Shape:Off-White To White Crystalline PowderMolecular weight:523.97Felodipine
CAS:Felodipine (CGH-869) is a longlasting 1, 4-dihydropyridine calcium channel repressor.Formula:C18H19Cl2NO4Purity:99.91%Color and Shape:SolidMolecular weight:384.25Ref: TM-T0145
2mg34.00€5mg50.00€10mg67.00€25mg96.00€50mg123.00€100mg168.00€500mg409.00€1mL*10mM (DMSO)54.00€Boc-LRR-AMC TFA
Boc-LRR-AMC TFA is a fluorogenic protease substrate for detecting trypsin-like activity in the 26S proteasome or 20S proteasome core.Formula:C35H53F3N10O9Purity:97.70%Color and Shape:SolidMolecular weight:814.85PACAP-38 (31-38), human, mouse, rat TFA
PACAP-38 (31-38), human, mouse, rat (TFA) demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal.Formula:C49H84F3N17O13Purity:98%Color and Shape:SolidMolecular weight:1176.29Isotachysterol 3
CAS:Isotachysterol 3 boosts calcium transport in gut and bone mobilization in kidneyless rats.Formula:C27H44OColor and Shape:SolidMolecular weight:384.64Nesiritide
CAS:Nesiritide, recombinant human B-type natriuretic peptide, binds NPR-A/C with Kd 7.3/13 pM.Formula:C143H244N50O42S4Purity:98%Color and Shape:SolidMolecular weight:3464.04NSC156529
CAS:NSC156529 suppresses AKT1, reduces cancer cell growth in vitro, and inhibits prostate tumors in vivo.Formula:C28H21ClS2Purity:98%Color and Shape:SolidMolecular weight:457.05Ryanodine
CAS:Ryanodine: a diterpenoid modulating Ca2+ release via ryanodine receptors; concentration-dependent effects; found in Ryania speciosa; toxic.Formula:C25H35NO9Purity:98%Color and Shape:White SolidMolecular weight:493.553D-myo-Inositol-1,3,4,5-tetraphosphate (sodium salt)
CAS:Ins(1,3,4,5)-P4, made via Ins(1,4,5)P3 phosphorylation, boosts calcium by opening ER and plasma membrane channels.Formula:C6H8Na8O18P4Color and Shape:SolidMolecular weight:675.93G-Glu-Ser
CAS:G-Glu-Ser is a calcium receptor activator and Flavor-enriching agent.Formula:C8H14N2O6Color and Shape:SolidMolecular weight:234.21Elgodipine
CAS:Elgodipine decreases angina severity, inhibits muscle growth, and is voltage-sensitive, showing promise for angina treatment.Formula:C29H33FN2O6Purity:99.84% - 99.98%Color and Shape:SolidMolecular weight:524.58NAADP tetrasodium salt
CAS:Ca2+ mobilizing agentFormula:C21H27N6O18P3Purity:98%Color and Shape:SolidMolecular weight:744.39D-myo-Inositol-1,3-diphosphate (sodium salt)
CAS:D-myo-Inositol-1,3-phosphate (Ins(1,3)P) is an inositol phosphate involved in cellular signal transduction.
Formula:C6H12Na2O12P2Color and Shape:SolidMolecular weight:384.08Mast cell degranulating peptide (28-49)
CAS:Mast cell degranulating peptide (28-49) is a bee venom depolarizer that can improve the cGMP content of cerebellum tablets in mice.
Formula:C110H196N40O24S4Purity:98%Color and Shape:SolidMolecular weight:2591.25RyRs activator 5
Compound A-1 (RyRs activator 5) is an efficacious agonist of ryanodine receptors, exhibiting activity against Spodoptera frugiperda [1].Color and Shape:Odour SolidBTT-266
CAS:BTT-266 is a blocker of voltage-gated calcium channel for pain management.
Formula:C34H28N4O4Purity:98.34%Color and Shape:SolidMolecular weight:556.61Cd1a
Cd1a, a β-toxin from the African spider Ceratogyrus darlingi, modulates calcium ion channels and inhibits human calcium ion channels (Ca v 2.2)(IC 50 2.6 μM) asColor and Shape:Odour Solidω-Conotoxin MVIIC
CAS:Peptide neurotoxin; wide spectrum blocker of N, P and Q type calcium channels.Formula:C106H178N40O32S7Purity:98%Color and Shape:White Lyophilised SolidMolecular weight:2749Fasudil
CAS:Fasudil (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.Formula:C14H17N3O2SPurity:99.79% - 99.84%Color and Shape:SolidMolecular weight:291.37Triphenylethylene
CAS:Compound PDK0283, with CAS No. 58-72-0, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0283 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formula:C20H16Color and Shape:White PowderMolecular weight:256.34Cavα2δ-IN-1
CAS:Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a KiFormula:C18H27N5OColor and Shape:SolidMolecular weight:329.448Huwentoxin I
CAS:Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.Formula:C161H246N48O44S6Purity:98%Color and Shape:SolidMolecular weight:3750.36Mipsagargin
CAS:Mipsagargin (G-202) is a new antibiotic that inhibits DNA biosynthesis.Formula:C66H100N6O27Purity:98%Color and Shape:SolidMolecular weight:1409.52Nesiritide acetate
CAS:Nesiritide, a 32-amino acid natriuretic peptide and recombinant form of human brain natriuretic peptide, enhances vasorelaxation ex vivo in porcine hearts from an acute coronary occlusion model when given as a 2 µg/kg bolus dose followed by a 0.01 µg/kg per minute infusion, facilitated by the calcium ionophore A23187. Formulations containing nesiritide have been utilized in managing congestive heart failure.Formula:C143H244N50O42S4C2H4O2Color and Shape:SolidMolecular weight:3524.1Cyclic ADP-ribose ammonium
cADPR ammonium is a second messenger that boosts cytosolic calcium via Ryanodine receptors and TRPM2 channels.Color and Shape:LiquidChlorocresol
CAS:Chlorocresol (4-Chloro-3-methylphenol) is an antiseptic medication.Formula:C7H7ClOColor and Shape:SolidMolecular weight:142.58ω-Agatoxin TK
CAS:Selective blocker of CaV2.1 P/Q-type calcium channels.Formula:C215H337N65O70S10Purity:98%Color and Shape:SolidMolecular weight:5273.02PACAP-38 (31-38), human, mouse, rat
CAS:PACAP-38 (31-38), human, mouse, rat demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal NPY and catecholamine productionFormula:C47H83N17O11Purity:98%Color and Shape:SolidMolecular weight:1062.27Candidalysin
CAS:Candidalysin is a cytolytic peptide toxin initially isolated from *Candida albicans*, exhibiting both toxic and non-toxic properties. It activates epithelial cell signaling pathways by interacting with the epithelial growth factor receptor (EGFR) on host cells, leading to the activation of matrix metalloproteinases (MMP) and calcium ion influx, which results in inflammatory responses and immune cell recruitment. Additionally, Candidalysin exhibits cytotoxicity by causing membrane damage to host cells.Formula:C153H266N38O38S2Color and Shape:SolidMolecular weight:3310.11sFTX-3.3
CAS:sFTX-3.3 is a calcium ion channel antagonist, exhibiting IC50 values of approximately 0.24 mM and 0.70 mM against P-type and N-type channels respectively.Formula:C12H29N7OColor and Shape:SolidMolecular weight:287.412MMK 1
CAS:Potent hFPR2 agonist; EC50: 1 nM (mFPR2), 2 nM (hFPR2), >10,000 nM (hFPR1). Induces monocyte/neutrophil migration, boosts IL-1β/IL-6, activates NADPH-oxidase.Formula:C75H123N19O18SPurity:98%Color and Shape:SolidMolecular weight:1610.97Katacalcin
CAS:Katacalcin (PDN 21) is a potent plasma calcium-lowering peptide[1].Formula:C97H154N34O36S2Purity:98%Color and Shape:White PowderMolecular weight:2436.6Kurtoxin
Kurtoxin is a selective Cav3 (T-type) voltage-gated Ca2+ channel gating inhibitor, exhibiting a dissociation constant (Kd) of 15 nM for the Cav3.1 (α1G T-type)Formula:C324H478N94O90S8Purity:98%Color and Shape:SolidMolecular weight:7386.36SG-094
CAS:SG-094 inhibits TPC2, halts RIL175 cell growth, IC50: 3.7 μM for cancer research.
Formula:C30H29NO3Purity:97.06%Color and Shape:SoildMolecular weight:451.56(±)5(6)-DiHETE
CAS:Eicosapentaenoic acid is an ω-3 polyunsaturated fatty acid that is abundant in marine organisms and fish oils.Formula:C20H32O4Color and Shape:SolidMolecular weight:336.472Sulcardine 2HCl
CAS:Sulcardine 2HCl is a multi-ion channel blocker that blocks the properties of hERG and hNav1.5 channels and can be used to study atrial fibrillation.Formula:C24H35Cl2N3O4SPurity:99.33% - 99.76%Color and Shape:SoildMolecular weight:532.523Ethacrynic acid D5
CAS:Ethacrynic acid: a diuretic, anti-inflammatory, inhibits calcium channels, GSTs, NF-kB pathway, and modulates leukotriene; has deuterium-labeled form.Formula:C13H12Cl2O4Purity:98%Color and Shape:SolidMolecular weight:308.17ω-Conotoxin GVIA
CAS:Peptide neurotoxin; selectively and reversibly blocks N-type calcium channels (IC50 = 0.15 nM). Reduces (RS)-3,5-DHPG -induced long term depression in vivo.Formula:C120H182N38O43S6Purity:98%Color and Shape:SolidMolecular weight:3037UK-59811 hydrochloride
CAS:UK-59811 hydrochloride, Br-dihydropyridine derivative, blocks Ca V Ab channels in bacteria, IC50: 194 nM.Formula:C22H30BrClN2O5Color and Shape:SolidMolecular weight:517.85Ziconotide
CAS:Ziconotide: analgesic from cone snail for severe, chronic pain; synthetic ω-conotoxin.Formula:C102H172N36O32S7Purity:98%Color and Shape:White PowderMolecular weight:2639.131-(aminomethyl)cyclopropanecarboxylic acid hydrochloride
CAS:1-(aminomethyl)cyclopropanecarboxylic acid hydrochloride inhibits L amino acid transporter proteins and the α2δ subunit of voltage-gated calcium channels.1-(
Formula:C5H10ClNO2Purity:>99.99%Color and Shape:SolidMolecular weight:151.59
