GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
Found 373 products of "GABA Receptor"
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L-822179
CAS:L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.Formula:C17H14N8O2Purity:98.5% - 99.61%Color and Shape:SolidMolecular weight:362.35L 663581
CAS:L 663581 is the benzodiazepine receptor partial agonist.Formula:C17H16ClN5O2Purity:98%Color and Shape:SolidMolecular weight:357.79Piperidine-4-sulfonic acid
CAS:Piperidine-4-sulfonic acid is a potent GABA agonist, demonstrating an IC50 value of 0.034 μM for the inhibition of H-GABA binding [1].Formula:C5H11NO3SPurity:98%Color and Shape:SolidMolecular weight:165.21CGP 54626 hydrochloride
CAS:CGP 54626 hydrochloride is a GABAB receptor antagonist.Formula:C18H29Cl3NO3PPurity:98%Color and Shape:SolidMolecular weight:444.76CGP 64213
CAS:CGP 64213 is a GABAb receptor agonist.Formula:C26H36IN2O7PPurity:98%Color and Shape:SolidMolecular weight:646.45Adipiplon
CAS:Adipiplon(NG2-73, NG273) is a novel selective gamma-aminobutyric acid (GABA) partial agonist.Formula:C18H18FN7Color and Shape:SolidMolecular weight:351.38ADX71441
CAS:ADX71441, a GABAB PAM, lengthens urinary latencies, lessens events & volume, and may aid in alcoholism and bladder pain.Formula:C19H15ClF2N4O4Color and Shape:SolidMolecular weight:436.8mGAT-IN-1
CAS:mGAT-IN-1 is a potent, non-selective GAT inhibitor that inhibits mGAT3 activity well (IC50: 2.5 μM, pIC50: 5.61).Formula:C28H34ClN3O2S2Color and Shape:SolidMolecular weight:544.17Afizagabar
CAS:Afizagabar, a first-in-class α5-GABAAR antagonist, IC50: 585 nM, Ki: 66 nM, may boost memory.Formula:C19H12FN3O2SColor and Shape:SolidMolecular weight:365.38PHP 501 trifluoroacetate
CAS:GABAA antagonistFormula:C20H21N3OPurity:98%Color and Shape:SolidMolecular weight:319.4FGIN-1-27
CAS:FGIN-1-27 is a high-affinity agonist of the translocator protein and a specific peripheral benzodiazepine receptor (PBR) ligand(Ki = 5.0 nM).Formula:C28H37FN2OPurity:99.86%Color and Shape:SolidMolecular weight:436.6CGP-54626 free base
CAS:CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).Formula:C18H28Cl2NO3PPurity:98%Color and Shape:SolidMolecular weight:408.3Diproqualone
CAS:Diproqualone, analogous to methaqualone, exhibits sedative, anxiolytic, anti-inflammatory, and analgesic properties [1].Formula:C12H14N2O3Color and Shape:SolidMolecular weight:234.255COR659
CAS:COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.Formula:C16H16ClNO3SPurity:99.75%Color and Shape:SolidMolecular weight:337.82Ref: TM-T36520
1mg38.00€5mg86.00€1mL*10mM (DMSO)94.00€10mg123.00€25mg215.00€50mg299.00€100mg411.00€200mg560.00€mGAT3/4-IN-2
CAS:mGAT3/4-IN-2 are potent inhibitors of mGAT3/mGAT4 with their pIC50 values of 5.44 and 5.25, respectively.Formula:C26H32ClN3OS2Color and Shape:SolidMolecular weight:502.13GMA-839
CAS:GMA-839 is a selective modulator of gamma-aminobutyric acid(A) receptors.Formula:C21H31F3O3Purity:98%Color and Shape:SolidMolecular weight:388.46NCS-382 sodium
CAS:NCS-382 (sodium) is a potent antagonist of the GABA receptor, exhibiting anti-sedative and anti-hypnotic properties, with applications in neurological diseaseFormula:C13H13NaO3Purity:98%Color and Shape:SolidMolecular weight:240.23NO-711ME
CAS:NO-711ME (N-O711 Methyl ester) is a prodrug of NO-711. It also is a potent and selective GABA uptake inhibitor.Formula:C22H24N2O3Purity:99.54%Color and Shape:SolidMolecular weight:364.44Ref: TM-T24540
1mg64.00€5mg129.00€1mL*10mM (DMSO)138.00€10mg188.00€25mg299.00€50mg427.00€100mg575.00€200mg767.00€U 89843A
CAS:U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.Formula:C16H23N5Purity:99.62%Color and Shape:SolidMolecular weight:285.39CP-409092
CAS:CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.Formula:C17H19N3O2Purity:98%Color and Shape:SolidMolecular weight:297.35
