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GABA Receptor

GABA Receptor

GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.

Found 364 products of "GABA Receptor"

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  • CymitQuimica logo
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    β-CCM

    CAS:
    β-CCM is a benzodiazepine receptor inverse agonist with anxiogenic and convulsant effects. It enhances emotional reactivity and reduces interference sensitivity in spatial working memory tasks. β-CCM is applicable in research related to anxiety disorders.
    Formula:C13H10N2O2
    Molecular weight:226.231

    Ref: TM-T206213

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    CGS-​9895

    CAS:
    CGS-9895 is a GABA antagonist that operates by interacting with the benzodiazepine binding site on GABA receptors containing the γ subunit (ag).
    Formula:C17H13N3O2
    Molecular weight:291.304

    Ref: TM-T204818

  • BGT1-IN-1
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    BGT1-IN-1

    CAS:
    BGT1-IN-1 (compound 9) is an effective inhibitor of BGT1, demonstrating IC50 values of 13.9 µM for hBGT1 and 58.3 µM for GAT3. It exhibits no cytotoxic effects and possesses neuroprotective activity.
    Formula:C6H9NO2
    Color and Shape:Solid
    Molecular weight:127.14

    Ref: TM-T200935

  • EF1502 free base
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    EF1502 free base

    CAS:
    EF1502 is a potent and selective GABA transporter inhibitor.
    Formula:C22H26N2O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.58

    Ref: TM-T27241

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    GABAA receptor agonist 1

    Compound 3e, a potent GABAA agonist, targets GABA sites and has potential anti-depressive effects in mice.
    Formula:C20H30O3
    Color and Shape:Solid
    Molecular weight:318.45

    Ref: TM-T60842

  • ZK 93426 hydrochloride
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    ZK 93426 hydrochloride

    CAS:
    benzodiazepine receptor antagonist,competitive
    Formula:C18H21ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.82

    Ref: TM-T23562

  • Cyproflanilide
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    Cyproflanilide

    CAS:
    Cyproflanilide is a GABAR antagonist that exhibits high activity against a variety of pests, including those from the Lepidoptera, Coleoptera, and Thysanoptera orders.
    Formula:C28H17BrF12N2O2
    Color and Shape:Solid
    Molecular weight:721.33

    Ref: TM-T201028

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    GABAA receptor agonist 2

    Compound 4c, a potent GABAA agonist with anti-depressive effects in mouse FST/TST, shows promise in depression research.
    Formula:C22H36O5
    Color and Shape:Solid
    Molecular weight:380.52

    Ref: TM-T61625

  • GABA-IN-4
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    GABA-IN-4

    CAS:
    GABA-IN-4 (Compound 17) is a derivative of N-(indol-3-ylglyoxylyl)benzylamine. It exhibits high affinity for the benzodiazepine receptor (BzR), the binding site within the GABAA receptor complex, with a Ki value of 67 nM. Benzodiazepines are widely used as anxiolytic, sedative-hypnotic, and anticonvulsant agents.
    Formula:C17H13ClN2O2
    Color and Shape:Solid
    Molecular weight:312.75

    Ref: TM-T205501

  • Moxetomidate
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    Moxetomidate

    CAS:
    <p>Moxetomidate is a GABAA receptor (GABAA receptor) agonist with hypnotic properties.</p>
    Formula:C15H18N2O3
    Color and Shape:Solid
    Molecular weight:274.315

    Ref: TM-T205308

  • Gabaculine HCl
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    Gabaculine HCl

    CAS:
    Gabaculine, an irreversible GABA-T inhibitor (Ki: 2.9 μM), impacts plastid development and affects DPOR/GluTR levels.
    Formula:C7H10ClNO2
    Color and Shape:Solid
    Molecular weight:175.61

    Ref: TM-T24080

  • Thiomuscimol hydrobromide
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    Thiomuscimol hydrobromide

    CAS:
    Thiomuscimol hydrobromide is an agonist of GABAA receptor.
    Formula:C4H6N2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:130.17

    Ref: TM-T28965

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    Refisolone

    CAS:
    Refisolone is an antagonist of the GABAA receptor.
    Formula:C18H24O3
    Molecular weight:288.381

    Ref: TM-T206497

  • S-8510 phosphate
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    S-8510 phosphate

    CAS:
    S-8510 phosphate is an agonist of inverse Benzodiazepine (BDZ) receptor(Kis of 34.6 nM, 36.2 nM for –GABA and +GABA respectively).
    Formula:C12H13N4O6P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:340.23

    Ref: TM-T12792

  • SGE-516
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    SGE-516

    CAS:
    <p>SGE516: neuroactive steroid, enhances GABAA, lowers neuronal activity, protects from seizures.</p>
    Formula:C23H35N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:385.54

    Ref: TM-T28766

  • (-)-Bicuculline methobromide
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    (-)-Bicuculline methobromide

    CAS:
    (-)-Bicuculline methobromide is a potent antagonist of GABAA receptor .
    Formula:C21H20BrNO6
    Color and Shape:White
    Molecular weight:462.29

    Ref: TM-T12043

    1mg
    Discontinued
    Discontinued product
  • 2-AEMP TFA
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    2-AEMP TFA

    CAS:
    2-AEMP TFA is a potent and rapidly acting antagonist of GABA(A)-ρ1 receptors. 2-AEMP is an analog of GABA.
    Formula:C3H10NO3P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:139.091

    Ref: TM-T26380

    5mg
    Discontinued
    25mg
    Discontinued
    Discontinued product
  • 3-Methylglutaconic acid
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    3-Methylglutaconic acid

    CAS:
    3-Methylglutaconic acid, a primary metabolite accumulating in 3-Methylglutaconic aciduria (MGTA), induces lipid and protein oxidation, while diminishing non-enzymatic antioxidant defenses in cerebral cortex supernatants, thereby promoting oxidative stress in the cerebral cortex. This compound is utilized in research concerning brain damage diseases [1].
    Formula:C6H8O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:144.13

    Ref: TM-T78071

    1mg
    Discontinued
    Discontinued product
  • Alfadolone acetate
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    Alfadolone acetate

    CAS:
    Alfadolone acetate is a gamma-aminobutyric acid (GABA) receptor agonist.
    Formula:C23H34O5
    Color and Shape:Solid
    Molecular weight:390.51

    Ref: TM-T26592

    ne
    Discontinued
    Discontinued product
  • Pipequaline
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    Pipequaline

    CAS:
    Pipequaline (PK-8165) is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It possesses a novel chemical structure that is not closely related to other drugs of this type. The drug has a similar pharmacological profile to the benzodiazepine family of drugs, but with mainly anxiolytic properties and very little sedative, amnestic or anticonvulsant effects, and so is classified as a nonbenzodiazepine anxiolytic.
    Formula:C22H24N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:316.44

    Ref: TM-T4655

    5mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    1ml*10 (DMSO)
    Discontinued
    Discontinued product