GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
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Bamaluzole
CAS:87034-87-5
Bamaluzole is an agonist of GABA receptor.
Formula:
C14H12ClN3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
273.72
Ref: TM-T10456
| 25mg | 1,406.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
RWJ-51204
CAS:205701-85-5
RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.
Formula:
C21H19F2N3O3
Purity:
100% - 99.57%
Color and Shape:
Solid
Molecular weight:
399.39
Ref: TM-T16811
| 1mg | 327.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,850.00 € | ||
| 100mg | 2,322.00 € | ||
| 500mg | 4,549.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
6,2'-Dihydroxyflavone
CAS:92439-20-8
6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.
Formula:
C15H10O4
Purity:
99.03%
Color and Shape:
Solid
Molecular weight:
254.24
Ref: TM-T8268
| 25mg | 39.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
NO-711ME
CAS:127586-66-7
NO-711ME (N-O711 Methyl ester) is a prodrug of NO-711. It also is a potent and …
Formula:
C22H24N2O3
Purity:
96.14%
Color and Shape:
Solid
Molecular weight:
364.44
Ref: TM-T24540
| 1mg | 94.00 € | ||
| 2mg | 120.00 € | ||
| 5mg | 181.00 € | ||
| 10mg | 273.00 € | ||
| 25mg | 436.00 € | ||
| 50mg | 621.00 € | ||
| 100mg | 835.00 € | ||
| 200mg | 1,116.00 € | ||
| 1mL*10mM (DMSO) | 195.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
L-822179
CAS:215874-86-5
L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with …
Formula:
C17H14N8O2
Purity:
98.34% - 98.74%
Color and Shape:
Solid
Molecular weight:
362.35
Ref: TM-T24381
| 1mg | 44.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 180.00 € | ||
| 50mg | 268.00 € | ||
| 100mg | 383.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
L-DABA hydrobromide
CAS:73143-97-2
L-DABA hydrobromide (L-2,4-Diaminobutyric acid hydrobromide) , GABA transaminase inhibitor with antitumor and anticonvulsant activity.
Formula:
C4H11BrN2O2
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
199.05
Ref: TM-T77795
| 100mg | 48.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
TPA 023
CAS:252977-51-8
TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 …
Formula:
C20H22FN7O
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
395.43
Ref: TM-T17144
| 1mg | 222.00 € | ||
| 5mg | 538.00 € | ||
| 10mg | 806.00 € | ||
| 25mg | 1,188.00 € | ||
| 50mg | 1,605.00 € | ||
| 100mg | 2,162.00 € | ||
| 1mL*10mM (DMSO) | 591.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
(+)-Bicuculline methiodide
CAS:40709-69-1
(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in …
Formula:
C21H20INO6
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
509.29
Ref: TM-T22604
| 1mg | 37.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
CP-409092
CAS:194098-25-4
CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.
Formula:
C17H19N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
297.35
Ref: TM-T10869L
| 25mg | 1,688.00 € | ||
| 50mg | 2,225.00 € | ||
| 100mg | 2,897.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
PZ-II-029
CAS:164025-44-9
PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.
Formula:
C18H15N3O3
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
321.33
Ref: TM-T28479
| 1mg | 91.00 € | ||
| 5mg | 166.00 € | ||
| 10mg | 257.00 € | ||
| 25mg | 480.00 € | ||
| 50mg | 693.00 € | ||
| 100mg | 981.00 € | ||
| 500mg | 1,930.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
COR659
CAS:544450-68-2
COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.
Formula:
C16H16ClNO3S
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
337.82
Ref: TM-T36520
| 1mg | 51.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 112.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 313.00 € | ||
| 50mg | 436.00 € | ||
| 100mg | 598.00 € | ||
| 200mg | 814.00 € | ||
| 1mL*10mM (DMSO) | 124.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
NCS-382 sodium
CAS:131733-92-1
NCS-382 (sodium) is a potent antagonist of the GABA receptor, exhibiting anti-sedative and anti-hypnotic properties, …
Formula:
C13H13NaO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
240.23
Ref: TM-T78111
| 10mg | 221.00 € | ||
| 50mg | 936.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
(-)-Bicuculline methochloride
CAS:53552-05-9
(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.
Formula:
C21H20ClNO6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
417.84
Ref: TM-T12044
| 5mg | 157.00 € | ||
| 10mg | 274.00 € | ||
| 25mg | 598.00 € | ||
| 50mg | 936.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
U 89843A
CAS:157013-32-6
U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.
Formula:
C16H23N5
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
285.39
Ref: TM-T23481
| 1mg | 46.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 130.00 € | ||
| 25mg | 295.00 € | ||
| 50mg | 522.00 € | ||
| 100mg | 704.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Xilmenolone
CAS:2368807-26-3
Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].
Formula:
C26H37N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
423.59
Ref: TM-T78670
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
SCS
CAS:3232-36-8
SCS is a GABAA receptor antagonist.
Formula:
C14H12N2O3
Purity:
98.89%
Color and Shape:
Solid
Molecular weight:
256.26
Ref: TM-T23339
| 10mg | 42.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | 89.00 € | ||
| 100mg | 130.00 € | ||
| 200mg | 182.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
TP003
CAS:628690-75-5
TP003 is a novel non-selective GABAA receptor benzodiazepine site agonist with affinity for α1β2gam2, α2β3gam2, …
Formula:
C23H16F3N3O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
407.39
Ref: TM-T23466
| 1mg | 46.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 274.00 € | ||
| 50mg | 410.00 € | ||
| 100mg | 592.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
T-2000
CAS:97846-21-4
T-2000 (DMMDPB) is a GABA receptor agonist that can be used to study myoclonus and …
Formula:
C20H20N2O5
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
368.38
Ref: TM-T28900
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information |
N-Arachidonyl-GABA
CAS:128201-89-8
N-Arachidonyl-GABA (NA-GABA) is a novel active fatty amino acid related to anandamide (ANA) found in …
Formula:
C24H39NO3
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
389.57
Ref: TM-T23039
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Indiplon
CAS:325715-02-4
Indiplon is a short-acting hypnotic with high-affinity allosteric potentiator of GABAA responses that demonstrates preference …
Formula:
C20H16N4O2S
Purity:
98.45%
Color and Shape:
Solid
Molecular weight:
376.43
Ref: TM-T21362
| 2mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information |
