GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
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Radequinil
CAS:219846-31-8
Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) …
Formula:
C18H14N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
334.33
Ref: TM-T16717
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
3α,21-Dihydroxy-5α-pregnan-20-one
CAS:567-02-2
3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like …
Formula:
C21H34O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
334.49
Ref: TM-T26390
| 1mg | 146.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Monday 16 Jun 2025
NO 711
CAS:159094-94-7
NNC-711: Strong GABA uptake blocker for GAT-1, IC50 = 0.04µM; weak on rGAT-2/hGAT-3/hBGT-1. Anticonvulsant in …
Formula:
C21H22N2O3
Purity:
99.83%
Color and Shape:
Liquid
Molecular weight:
350.41
Ref: TM-T70414
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
Divaplon
CAS:90808-12-1
Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics …
Formula:
C17H17N3O2
Purity:
96.90% - 97.49%
Color and Shape:
Solid
Molecular weight:
295.34
Ref: TM-T27186
| 1mg | 143.00 € | ||
| 5mg | 333.00 € | ||
| 10mg | 504.00 € | ||
| 25mg | 817.00 € | ||
| 50mg | 1,121.00 € | ||
| 100mg | 1,510.00 € | ||
| 500mg | 3,030.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
DMCM hydrochloride
CAS:1215833-62-7
DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.
Formula:
C17H19ClN2O4
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
350.8
Ref: TM-T11061
| 1mg | 37.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 464.00 € | ||
| 100mg | 655.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
Lesogaberan
CAS:344413-67-8
Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity …
Formula:
C3H9FNO2P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
141.08
Ref: TM-T15737
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
GS 39783
CAS:39069-52-8
GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties …
Formula:
C15H23N5O2S
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
337.44
Ref: TM-T22813
| 1mg | 46.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 137.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 406.00 € | ||
| 100mg | 592.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
Bamaluzole
CAS:87034-87-5
Bamaluzole is an agonist of GABA receptor.
Formula:
C14H12ClN3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
273.72
Ref: TM-T10456
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
Ru-32514
CAS:90807-98-0
Ru-32514 is a benzodiazepine receptor agonist.
Formula:
C18H17N3O2
Purity:
98.74%
Color and Shape:
Solid
Molecular weight:
307.35
Ref: TM-T12779
| 1mg | 279.00 € | ||
| 2mg | 414.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
SCH 50911
CAS:733717-87-8
SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow …
Formula:
C8H15NO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
173.21
Ref: TM-T12867L
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Jun 2025
Anxiolytic/nonsedative agent-1
CAS:355022-97-8
TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy …
Formula:
C18H15N3O4
Purity:
97.05%
Color and Shape:
Solid
Molecular weight:
337.33
Ref: TM-T23445
| 1mg | 64.00 € | ||
| 2mg | 96.00 € | ||
| 5mg | 115.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 330.00 € | ||
| 50mg | 472.00 € | ||
| 100mg | 655.00 € | ||
| 500mg | 1,293.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
NNC 05-711
CAS:145645-62-1
NNC 711 is a GABA uptake inhibitor.
Formula:
C21H23ClN2O3
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
386.87
Ref: TM-T23075
| 1mg | 69.00 € | ||
| 5mg | 164.00 € | ||
| 10mg | 235.00 € | ||
| 25mg | 399.00 € | ||
| 50mg | 567.00 € | ||
| 100mg | 820.00 € | ||
| 200mg | 1,103.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
NCS-382 sodium
CAS:131733-92-1
NCS-382 (sodium) is a potent antagonist of the GABA receptor, exhibiting anti-sedative and anti-hypnotic properties, …
Formula:
C13H13NaO3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
240.23
Ref: TM-T78111
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 30 Jun 2025
L-DABA hydrobromide
CAS:73143-97-2
L-DABA hydrobromide (L-2,4-Diaminobutyric acid hydrobromide) , GABA transaminase inhibitor with antitumor and anticonvulsant activity.
Formula:
C4H11BrN2O2
Purity:
99.11%
Color and Shape:
Liquid
Molecular weight:
199.05
Ref: TM-T77795
| 100mg | 48.00 € |
Estimated delivery in United States, on Monday 30 Jun 2025
COR659
CAS:544450-68-2
COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.
Formula:
C16H16ClNO3S
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
337.82
Ref: TM-T36520
| 1mg | 52.00 € | ||
| 2mg | 75.00 € | ||
| 5mg | 116.00 € | ||
| 10mg | 178.00 € | ||
| 25mg | 324.00 € | ||
| 50mg | 452.00 € | ||
| 100mg | 620.00 € | ||
| 200mg | 843.00 € | ||
| 1mL*10mM (DMSO) | 128.00 € |
Estimated delivery in United States, on Monday 30 Jun 2025
6,2'-Dihydroxyflavone
CAS:92439-20-8
6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.
Formula:
C15H10O4
Purity:
99.03%
Color and Shape:
Solid
Molecular weight:
254.24
Ref: TM-T8268
| 25mg | 39.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 30 Jun 2025
Xilmenolone
CAS:2368807-26-3
Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].
Formula:
C26H37N3O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
423.59
Ref: TM-T78670
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 30 Jun 2025
CP-409092
CAS:194098-25-4
CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.
Formula:
C17H19N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
297.35
Ref: TM-T10869L
| 25mg | 1,730.00 € | ||
| 50mg | 2,262.00 € | ||
| 100mg | 2,945.00 € |
Estimated delivery in United States, on Monday 30 Jun 2025
L-822179
CAS:215874-86-5
L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with …
Formula:
C17H14N8O2
Purity:
98.34% - 98.74%
Color and Shape:
Solid
Molecular weight:
362.35
Ref: TM-T24381
| 1mg | 46.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 278.00 € | ||
| 100mg | 398.00 € |
Estimated delivery in United States, on Monday 30 Jun 2025
PZ-II-029
CAS:164025-44-9
PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.
Formula:
C18H15N3O3
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
321.33
Ref: TM-T28479
| 1mg | 52.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 305.00 € | ||
| 50mg | 472.00 € | ||
| 100mg | 723.00 € | ||
| 500mg | 1,454.00 € | ||
| 1mL*10mM (DMSO) | 202.00 € |
Estimated delivery in United States, on Monday 30 Jun 2025
