GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
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3α,21-Dihydroxy-5α-pregnan-20-one
CAS:567-02-2
3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like …
Formula:
C21H34O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
334.49
Ref: TM-T26390
| 1mg | 141.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Friday 27 Dec 2024
DMCM hydrochloride
CAS:1215833-62-7
DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.
Formula:
C17H19ClN2O4
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
350.8
Ref: TM-T11061
| 1mg | 37.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 248.00 € | ||
| 50mg | 461.00 € | ||
| 100mg | 650.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Nerisopam
CAS:102771-12-0
Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.
Formula:
C18H19N3O2
Purity:
97.27%
Color and Shape:
Solid
Molecular weight:
309.36
Ref: TM-T28159
| 1mg | 138.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 496.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,477.00 € | ||
| 500mg | 2,960.00 € | ||
| 1mL*10mM (DMSO) | 449.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Fengabine
CAS:80018-06-0
Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat …
Formula:
C17H17Cl2NO
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
322.23
Ref: TM-T27310
| 1mg | 82.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 242.00 € | ||
| 25mg | 470.00 € | ||
| 50mg | 643.00 € | ||
| 100mg | 912.00 € | ||
| 500mg | 1,829.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Radequinil
CAS:219846-31-8
Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) …
Formula:
C18H14N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
334.33
Ref: TM-T16717
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
SCH 50911 hydrochloride
CAS:160415-07-6
SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) …
Formula:
C8H16ClNO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
209.67
Ref: TM-T12867
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Divaplon
CAS:90808-12-1
Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics …
Formula:
C17H17N3O2
Purity:
96.90% - 97.49%
Color and Shape:
Solid
Molecular weight:
295.34
Ref: TM-T27186
| 1mg | 141.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 797.00 € | ||
| 50mg | 1,100.00 € | ||
| 100mg | 1,476.00 € | ||
| 500mg | 2,980.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Pazinaclone
CAS:103255-66-9
Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.
Formula:
C25H23ClN4O4
Purity:
98.12% - 99%
Color and Shape:
Solid
Molecular weight:
478.93
Ref: TM-T28303
| 1mg | 138.00 € | ||
| 5mg | 325.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 797.00 € | ||
| 50mg | 1,100.00 € | ||
| 100mg | 1,476.00 € | ||
| 500mg | 2,980.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
E2730
CAS:1520073-91-9
E2730 is a selective and noncompetitive inhibitor of the gamma-aminobutyric acid (GABA) transporter 1 (GAT1) …
Formula:
C9H8F4N2O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
284.23
Ref: TM-T79399
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
U-89843A
CAS:157013-85-9
U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents …
Formula:
C16H24ClN5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
321.85
Ref: TM-T78560
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
(R)-Baclofen hydrochloride
CAS:63701-55-3
Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.
Formula:
C10H13Cl2NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
250.12
Ref: TM-T17306
| 10mg | 87.00 € | ||
| 25mg | 200.00 € | ||
| 50mg | 328.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Pipequaline
CAS:77472-98-1
Pipequaline (PK-8165) is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that …
Formula:
C22H24N2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
316.44
Ref: TM-T4655
| 5mg | 49.00 € | ||
| 25mg | 121.00 € | ||
| 50mg | 219.00 € | ||
| 100mg | 379.00 € | ||
| 1ml*10 (DMSO) | 50.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
GABAB receptor antagonist 1
CAS:797-17-1
(E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM.GABAB …
Formula:
C18H24O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
304.38
Ref: TM-T11350
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
(E)-GABAB receptor antagonist 1
CAS:1611483-29-4
(E)-GABAB antagonist 1 inhibits GABA IP3 production, with an IC50 of 37.9 μM and acts …
Formula:
C18H24O4
Purity:
95.26%
Color and Shape:
Solid
Molecular weight:
304.38
Ref: TM-T11137
| 1mg | 112.00 € | ||
| 5mg | 248.00 € | ||
| 10mg | 365.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 765.00 € | ||
| 100mg | 1,044.00 € | ||
| 200mg | 1,413.00 € | ||
| 1mL*10mM (DMSO) | 240.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
AZD 3043
CAS:579494-66-9
AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a …
Formula:
C19H29NO5
Purity:
98.19% - ≥98%
Color and Shape:
Solid
Molecular weight:
351.44
Ref: TM-T30248
| 1mg | 273.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,416.00 € | ||
| 50mg | 1,845.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Alpidem
CAS:82626-01-5
Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.
Formula:
C21H23Cl2N3O
Purity:
100% - 99.49%
Color and Shape:
White To Off-White Solid
Molecular weight:
404.33
Ref: TM-T26600
| 1mg | 60.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 230.00 € | ||
| 25mg | 388.00 € | ||
| 50mg | 552.00 € | ||
| 100mg | 800.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Ru-32514
CAS:90807-98-0
Ru-32514 is a benzodiazepine receptor agonist.
Formula:
C18H17N3O2
Purity:
98.74%
Color and Shape:
Solid
Molecular weight:
307.35
Ref: TM-T12779
| 1mg | 274.00 € | ||
| 2mg | 408.00 € | ||
| 5mg | 675.00 € | ||
| 10mg | 922.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Golexanolone
CAS:2089238-18-4
Golexanolone can be used to study neurological diseases.
Formula:
C21H31NO2
Purity:
98.81% - 99.98%
Color and Shape:
Solid
Molecular weight:
329.48
Ref: TM-T25458
| 1mg | 273.00 € | ||
| 5mg | 672.00 € | ||
| 10mg | 918.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
NS-2710
CAS:184220-36-8
NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.
Formula:
C22H20N4O
Purity:
98.10% - 99.82%
Color and Shape:
Solid
Molecular weight:
356.42
Ref: TM-T28197
| 1mg | 273.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Lesogaberan
CAS:344413-67-8
Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity …
Formula:
C3H9FNO2P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
141.08
Ref: TM-T15737
| 25mg | 1,406.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
