GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
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Fengabine
CAS:80018-06-0
Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat …
Formula:
C17H17Cl2NO
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
322.23
Ref: TM-T27310
| 1mg | 82.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 242.00 € | ||
| 25mg | 470.00 € | ||
| 50mg | 643.00 € | ||
| 100mg | 912.00 € | ||
| 500mg | 1,829.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
E2730
CAS:1520073-91-9
E2730 is a selective and noncompetitive inhibitor of the gamma-aminobutyric acid (GABA) transporter 1 (GAT1) …
Formula:
C9H8F4N2O2S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
284.23
Ref: TM-T79399
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Lesogaberan
CAS:344413-67-8
Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity …
Formula:
C3H9FNO2P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
141.08
Ref: TM-T15737
| 25mg | 1,406.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Bamaluzole
CAS:87034-87-5
Bamaluzole is an agonist of GABA receptor.
Formula:
C14H12ClN3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
273.72
Ref: TM-T10456
| 25mg | 1,406.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
RWJ-51204
CAS:205701-85-5
RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.
Formula:
C21H19F2N3O3
Purity:
100% - 99.57%
Color and Shape:
Solid
Molecular weight:
399.39
Ref: TM-T16811
| 1mg | 327.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,850.00 € | ||
| 100mg | 2,322.00 € | ||
| 500mg | 4,549.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Nerisopam
CAS:102771-12-0
Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.
Formula:
C18H19N3O2
Purity:
97.27%
Color and Shape:
Solid
Molecular weight:
309.36
Ref: TM-T28159
| 1mg | 138.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 496.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,477.00 € | ||
| 500mg | 2,960.00 € | ||
| 1mL*10mM (DMSO) | 449.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
3α,21-Dihydroxy-5α-pregnan-20-one
CAS:567-02-2
3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like …
Formula:
C21H34O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
334.49
Ref: TM-T26390
| 1mg | 141.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Thursday 23 Jan 2025
Progabide
CAS:62666-20-0
Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.
Formula:
C17H16ClFN2O2
Purity:
99.7%
Color and Shape:
Solid
Molecular weight:
334.77
Ref: TM-T16581
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 151.00 € | ||
| 100mg | 230.00 € | ||
| 200mg | 326.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Tracazolate hydrochloride
CAS:1135210-68-2
Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant …
Formula:
C16H25ClN4O2
Purity:
99.07%
Color and Shape:
Solid
Molecular weight:
340.85
Ref: TM-T23470
| 5mg | 41.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 114.00 € | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Thursday 23 Jan 2025
BPDBA
CAS:312281-74-6
BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory …
Formula:
C19H20Cl2N2O
Purity:
99.24% - 99.86%
Color and Shape:
Solid
Molecular weight:
363.28
Ref: TM-T26891
| 1g | 1,304.00 € | ||
| 2mg | 42.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 174.00 € | ||
| 50mg | 279.00 € | ||
| 100mg | 450.00 € | ||
| 500mg | 985.00 € | ||
| 1mL*10mM (DMSO) | 115.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Suriclone
CAS:53813-83-5
Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.
Formula:
C20H20ClN5O3S2
Purity:
98.17% - 98.52%
Color and Shape:
Solid
Molecular weight:
477.99
Ref: TM-T28887
| 1mg | 141.00 € | ||
| 5mg | 326.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 797.00 € | ||
| 50mg | 1,100.00 € | ||
| 100mg | 1,481.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Lirequinil
CAS:143943-73-1
Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.
Formula:
C26H25ClN2O3
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
448.94
Ref: TM-T27838
| 1mg | 155.00 € | ||
| 5mg | 372.00 € | ||
| 10mg | 561.00 € | ||
| 25mg | 891.00 € | ||
| 50mg | 1,196.00 € | ||
| 100mg | 1,635.00 € | ||
| 500mg | 3,240.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Phaclofen
CAS:114012-12-3
GABAB antagonist
Formula:
C9H13ClNO3P
Purity:
99.32%
Color and Shape:
White Solid
Molecular weight:
249.63
Ref: TM-T23147
| 1mg | 81.00 € | ||
| 5mg | 168.00 € | ||
| 10mg | 279.00 € | ||
| 25mg | 645.00 € | ||
| 50mg | 896.00 € | ||
| 100mg | 1,201.00 € | ||
| 200mg | 1,623.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Sarmazenil
CAS:78771-13-8
Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used …
Formula:
C15H14ClN3O3
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
319.74
Ref: TM-T16844
| 1mg | 278.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 936.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
U-89843A
CAS:157013-85-9
U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents …
Formula:
C16H24ClN5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
321.85
Ref: TM-T78560
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
Riluzole hydrochloride
CAS:850608-87-6
Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).
Formula:
C8H6ClF3N2OS
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
270.66
Ref: TM-T41265
| 25mg | 37.00 € | ||
| 50mg | 52.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
RO 4938581
CAS:883093-10-5
RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, …
Formula:
C13H8BrF2N5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
352.14
Ref: TM-T16794
| 25mg | 1,141.00 € | ||
| 50mg | 1,499.00 € | ||
| 100mg | 2,468.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
GS 39783
CAS:39069-52-8
GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties …
Formula:
C15H23N5O2S
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
337.44
Ref: TM-T22813
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 134.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 399.00 € | ||
| 100mg | 579.00 € |
Estimated delivery in United States, on Thursday 23 Jan 2025
NCS-382 sodium
CAS:131733-92-1
NCS-382 (sodium) is a potent antagonist of the GABA receptor, exhibiting anti-sedative and anti-hypnotic properties, …
Formula:
C13H13NaO3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
240.23
Ref: TM-T78111
| 10mg | 221.00 € | ||
| 50mg | 936.00 € |
Estimated delivery in United States, on Thursday 6 Feb 2025
U 89843A
CAS:157013-32-6
U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.
Formula:
C16H23N5
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
285.39
Ref: TM-T23481
| 1mg | 46.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 130.00 € | ||
| 25mg | 295.00 € | ||
| 50mg | 522.00 € | ||
| 100mg | 704.00 € |
Estimated delivery in United States, on Thursday 6 Feb 2025
