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Aminopeptidase

Aminopeptidase

Aminopeptidases are a group of enzymes that catalyze the cleavage of amino acids from the N-terminus of peptides and proteins, playing a crucial role in protein maturation and degradation. These enzymes are involved in various physiological processes, including antigen processing, peptide hormone regulation, and cellular homeostasis. Inhibitors of aminopeptidases are of interest in the treatment of diseases such as cancer, inflammation, and infectious diseases. At CymitQuimica, we provide a variety of aminopeptidase inhibitors to support your research in proteomics, drug development, and disease treatment.

Found 67 products of "Aminopeptidase"

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  • Leucinal
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    Leucinal

    CAS:
    <p>Leucinal inhibits the activity of brain aminopeptidase and potentiates analgesia induced by leu-enkephalen.</p>
    Formula:C6H13NO
    Color and Shape:Solid
    Molecular weight:115.17

    Ref: TM-T25675

  • M8891
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    M8891

    CAS:
    <p>M8891: Oral, reversible MetAP-2 inhibitor, brain-penetrant (IC50: 54nM; Ki: 4.33nM), hinders endothelial &amp; tumor cell growth, antiangiogenic &amp; antitumor.</p>
    Formula:C20H17F2N3O3
    Color and Shape:Solid
    Molecular weight:385.36

    Ref: TM-T11930

  • HFI-437
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    HFI-437

    CAS:
    <p>HFI-437 is a potent, non-peptidic, insulin-regulated aminopeptidase (IRAP) inhibitor with a K i of 20 nM and functions as a cognitive enhancer [1].</p>
    Formula:C23H20N2O5
    Color and Shape:Solid
    Molecular weight:404.42

    Ref: TM-T86574

  • Amastatin
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    Amastatin

    CAS:
    <p>Amastatin is a non-toxic inhibitor of aminopeptidase A and leucine aminopeptidase, and its Ki for aminopeptidase A is 1 μM .</p>
    Formula:C21H38N4O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:474.55

    Ref: TM-T22255

  • Aminopeptidase-IN-1
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    Aminopeptidase-IN-1

    CAS:
    <p>Aminopeptidase-IN-1: potent IRAP blocker, Ki 7.7 μM, useful for cognitive/memory disorder research.</p>
    Formula:C18H16N2O6
    Purity:98.37%
    Color and Shape:Solid
    Molecular weight:356.33

    Ref: TM-T61278

  • SC-22716
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    SC-22716

    CAS:
    <p>SC-22716 is a LTA4 hydrolase inhibitor.SC-22716 has anti-inflammatory activity and may be used in the study of inflammatory bowel disease and psoriasis.</p>
    Formula:C18H21NO
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:267.37

    Ref: TM-T28698

  • TP-004
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    TP-004

    CAS:
    <p>TP-004 is a potent and reversible methionine aminopeptidase 2 (MetAP2) inhibitor (IC50: 6 nM).</p>
    Formula:C17H16F3N5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:363.34

    Ref: TM-T13188

  • BDM14471
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    BDM14471

    CAS:
    <p>BDM14471 is a selective inhibitor of hydroxamate PfAM1.</p>
    Formula:C17H15FN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:314.31

    Ref: TM-T25141

  • LYS006
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    LYS006

    CAS:
    <p>LYS006 is a highly efficient and selective LTA4H (leukotriene A4 hydrolase) inhibitor,for neutrophil-driven inflammatory diseases ulcerative colitis.</p>
    Formula:C16H14ClFN6O3
    Purity:99.33%
    Color and Shape:Soild
    Molecular weight:392.77

    Ref: TM-T9690

  • JNJ-40929837
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    JNJ-40929837

    CAS:
    <p>JNJ-40929837 is an oral inhibitor of LTA4 hydrolase, which catalyzes LTB4 production.</p>
    Formula:C22H24N4O2S
    Color and Shape:Solid
    Molecular weight:408.52

    Ref: TM-T71283

  • RB 101
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    RB 101

    CAS:
    <p>RB 101 suppresses enkephalinase and aminopeptidases; biologically cleaved at disulfide to produce inhibitors of both aminopeptidase N and neutral endopeptidase.</p>
    Formula:C31H38N2O3S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:582.84

    Ref: TM-T26048

  • MetAP2-IN-1
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    MetAP2-IN-1

    CAS:
    <p>MetAP2-IN-1 is a selective inhibitor of MetAP2, a target involved in angiogenesis-related conditions, suitable for research applications [1].</p>
    Formula:C8H6BrN3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:224.06

    Ref: TM-T78129

  • Arphamenine A
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    Arphamenine A

    CAS:
    <p>Arphamenine A is an inhibitor of aminopeptidase B (aminopeptidaseB) found in HMG361-CF4 of Actinomadura azurea. It exhibits inhibitory effects against Sarcoma 180 and invasive micropapillary carcinoma (IMC).</p>
    Formula:C16H24N4O3
    Color and Shape:Solid
    Molecular weight:320.387

    Ref: TM-TN10713

  • A-800141
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    A-800141

    CAS:
    <p>A-800141 is an orally active and selective MetAP2 inhibitor with an IC50 of 12 nM, while showing weaker inhibitory activity against MetAP1 (IC50: 36 μM). GAPDH can serve as a biomarker for monitoring the inhibition of MetAP2 by A-800141. This compound exhibits anti-angiogenic and anticancer properties in various xenograft tumor models.</p>
    Formula:C24H30N2O4S
    Color and Shape:Solid
    Molecular weight:442.571

    Ref: TM-T204983

  • EC33
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    EC33

    CAS:
    <p>EC33, a selective aminopeptidase A (APA) inhibitor, blocks the pressor response of exogenous Ang II and does not cross the blood-brain barrier, making it a potential candidate for salt-dependent hypertension research [1].</p>
    Formula:C4H11NO3S2
    Color and Shape:Solid
    Molecular weight:185.27

    Ref: TM-T86337

  • LTA4H-IN-3
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    LTA4H-IN-3

    CAS:
    <p>LTA4H-IN-3 (compound 9) functions as an inhibitor of LTA4H, demonstrating an IC50 of 28 nM [1].</p>
    Formula:C17H15ClN4O3
    Color and Shape:Solid
    Molecular weight:358.78

    Ref: TM-T86828

  • LTA4H-IN-2
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    LTA4H-IN-2

    CAS:
    <p>LTA4H-IN-2 (compound (S)-2) acts as an orally active inhibitor targeting Leukotriene A4 Hydrolase, exhibiting potent activity with an IC 50 of less than 3 nM [1].</p>
    Formula:C20H19FN6O2
    Color and Shape:Solid
    Molecular weight:394.4

    Ref: TM-T86827

  • Bestatin methyl ester
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    Bestatin methyl ester

    CAS:
    <p>Bestatin methyl ester (600, 900 µM; 24 h) inhibits spore cell differentiation in Dictyostelium discoideum.</p>
    Formula:C17H26N2O4
    Color and Shape:Solid
    Molecular weight:322.4

    Ref: TM-T88754

  • Ketomethylenebestatin
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    Ketomethylenebestatin

    CAS:
    <p>Ketomethylenebestatin, a weaker carba-analog of aminopeptidase inhibitor bestatin, is 10x less potent.</p>
    Formula:C17H25NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:307.38

    Ref: TM-T25573

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    SDX-7539

    CAS:
    <p>SDX-7539 is a selective MetAP2 inhibitor that inhibits the proliferation of HUVEC, with an IC50 of 120 μM. It has demonstrated antitumor activity in xenografted NSCLC in athymic nude mice.</p>
    Formula:C23H38N2O5
    Molecular weight:422.56

    Ref: TM-T209478