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5-HT Receptor

5-HT Receptor

5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.

Found 940 products of "5-HT Receptor"

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  • MR33317


    <p>MR33317 is an inhibitor of acetylcholinesterase with an IC50 value of 41 nM. Additionally, it acts as an agonist for brain 5-HT4 receptors.</p>
    Formula:C22H28ClN3O2
    Molecular weight:401.187
  • Naratriptan D3 Hydrochloride

    CAS:
    <p>Naratriptan D3 Hydrochloride is the deuterium labeled Naratriptan, is a selective agonist of 5-HT1 receptor subtype.</p>
    Formula:C17H26ClN3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:374.94
  • 5-MeO-pyr-T

    CAS:
    <p>5-MeO-pyr-T (5-Methoxy pyrrolidinyltryptamine) acts as a 5-HT1AR agonist, exhibiting Ki values of 0.577 μM and 373 μM for 5-HT1AR and 5-HT2AR, respectively. It inhibits the reuptake of 5-HT and triggers its release. Additionally, 5-MeO-pyr-T can induce reduced motor activity.</p>
    Formula:C15H20N2O
    Color and Shape:Solid
    Molecular weight:244.33
  • SB 699551

    CAS:
    <p>SB 699551 is a selective 5-HT5A antagonist (Ki=6.31 nM) that enhances 5-HT neuronal function. It inhibits SERT (Ki=25.12 nM),inhibit breast cancer.</p>
    Formula:C34H45N3O
    Purity:99.83%
    Molecular weight:511.74
  • Neocarzinostatin

    CAS:
    <p>Neocarzinostatin is an effective DNA-damaging, anti-tumor antibiotic.</p>
    Purity:98%
    Color and Shape:Solid
    Molecular weight:N/A
  • Paynantheine

    CAS:
    <p>Paynantheine is an alkaloid with antinociceptive properties, found in Mitragyna speciosa. It also acts as an agonist at 5-HT1AR and 5-HT2BR receptors, inducing lower lip contraction and providing antinociception in rats.</p>
    Formula:C23H28N2O4
    Color and Shape:Solid
    Molecular weight:396.48
  • Cinanserin hydrochloride

    CAS:
    <p>Cinanserin hydrochloride (SQ 10643) is a 5-HT2 receptor blocker (Ki: 41 nM) and SARS-CoV 3C-like protease inhibitor.</p>
    Formula:C20H25ClN2OS
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:376.94
  • Dehydro Aripiprazole (hydrochloride)

    CAS:
    <p>Dehydro aripiprazole, an active atypical antipsychotic metabolite of aripiprazole, is formed by CYP3A4 and CYP2D6.</p>
    Formula:C23H26Cl3N3O2
    Color and Shape:Solid
    Molecular weight:482.83
  • Donitriptan hydrochloride

    CAS:
    <p>Donitriptan hydrochloride (Donitriptan monohydrochloride) is a potent, high efficacy agonist of 5-HT1B/1D receptors with pKis of 9.4 and 9.3, respectively</p>
    Formula:C23H26ClN5O2
    Purity:99.8% - 99.86%
    Color and Shape:Solid
    Molecular weight:439.94
  • 1,8-Cineole

    CAS:
    <p>Eucalyptol, a natural monoterpenoid and cyclic ether found in eucalyptus species, effectively controls excessive airway mucus secretion and asthma by inhibiting pro-inflammatory cytokines. It serves as an efficacious treatment for non-purulent sinusitis, reducing inflammation and pain when applied topically, and demonstrating leukemic cell-killing capabilities in vitro.</p>
    Formula:C10H18O
    Purity:97.44% - 97.44%
    Color and Shape:Solid
    Molecular weight:154.25
  • (Rac)-Norcisapride

    CAS:
    <p>Norcisapride, a 5-HT3 and 5-HT4 agonist, treats GI, orofacial, and ENT disorders.</p>
    Formula:C14H20ClN3O3
    Purity:99.32%
    Color and Shape:Soild
    Molecular weight:313.78
  • (R,R)-Palonosetron Hydrochloride

    CAS:
    <p>(R,R)-Palonosetron Hydrochloride is the active enantiomer of Palonosetron</p>
    Formula:C19H25ClN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.87
  • 5-HT2A receptor agonist-5

    CAS:
    <p>5-HT2A receptor agonist-5 (compound I-3) is a potent 5-HT2A agonist with a Ki value of 0.017 µM and exhibits antidepressant activity.</p>
    Formula:C23H29N3O
    Color and Shape:Solid
    Molecular weight:363.5
  • Eletriptan

    CAS:
    <p>Eletriptan, second-generation triptans used to treat migraines, is used as an abortion drug.</p>
    Formula:C22H26N2O2S
    Color and Shape:Solid
    Molecular weight:382.52
  • LEK 8804

    CAS:
    <p>LEK 8804 is a 5-HT(2) receptor antagonist and 5-HT(1A) receptor agonist.</p>
    Formula:C19H19N3O
    Color and Shape:Solid
    Molecular weight:305.37
  • AMI-193

    CAS:
    <p>AMI-193 (Spiramide) is a selective 5-HT2 &amp; D2 receptor antagonist with antipsychotic properties.</p>
    Formula:C22H26FN3O2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:383.46
  • LE 300

    CAS:
    <p>LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.</p>
    Formula:C20H22N2
    Purity:97.91% - 98.79%
    Color and Shape:Solid
    Molecular weight:290.4
  • (-)-Eseroline fumarate

    CAS:
    <p>(-)-Eseroline fumarate, a Physostigmine metabolite and AChE inhibitor, triggers cancer cell LDH release and neuronal cell death.</p>
    Formula:C17H22N2O5
    Color and Shape:Solid
    Molecular weight:334.37
  • Ro60-0175

    CAS:
    <p>Ro60-0175 is a selective 5-HT2B and 5-HT2C serotonin receptor agonist, often used as fumarate.</p>
    Formula:C11H12ClFN2
    Purity:97.09%
    Color and Shape:Solid
    Molecular weight:226.68
  • LY 344864 racemate

    CAS:
    <p>LY 344864 racemate is a 5-HT1F receptor agonist.</p>
    Formula:C21H22FN3O
    Purity:99.75%
    Color and Shape:Soild
    Molecular weight:351.42