5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
Found 1025 products of "5-HT Receptor"
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Way 100289
CAS:Way 100289 is a selective 5-HT3 receptor antagonist.Formula:C20H27N3O3Color and Shape:SolidMolecular weight:357.45Cinitapride Hydrogen Tartrate
CAS:Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptorsFormula:C25H36N4O10Purity:98%Color and Shape:SolidMolecular weight:552.581LP44 hydrochloride
CAS:LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.Formula:C27H38ClN3OSPurity:98.06%Color and Shape:SolidMolecular weight:488.13CUMI-101
CAS:CUMI-101 is an agonist of 5-HT1A receptor.Formula:C19H27N5O3Color and Shape:SolidMolecular weight:373.45FK-1052 HCl
CAS:FK-1052 HCl is a serotonin 3 & 4 dual receptor antagonist.Formula:C18H20ClN3OColor and Shape:SolidMolecular weight:329.83Deramciclane fumarate
CAS:Deramciclane fumarate is a 5-HT(2A/C) antagonist with putative anxiolytic activity.Formula:C24H35NO5Color and Shape:SolidMolecular weight:417.54PF-4522654
CAS:PF-4522654 is a potent and selective 5-HT2C receptor agonist.Formula:C16H18F2N4Color and Shape:SolidMolecular weight:304.34Zimelidine dihydrochloride
CAS:5-HT re-uptake inhibitorFormula:C16H18BrClN2Purity:98%Color and Shape:SolidMolecular weight:353.69Ifoxetine sulfate
CAS:Ifoxetine sulfate, an atypical 5-HT inhibitor, may show unique therapeutic effects and side-effects.Formula:C13H19NO2H2O4SPurity:98%Color and Shape:SolidMolecular weight:270.34Ro 63-0563
CAS:Ro 63-0563 is a potent, 5-HT6 receptors selective antagonist.Formula:C13H17N5O2SPurity:98%Color and Shape:SolidMolecular weight:307.37Usmarapride free base
CAS:Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.Formula:C21H29N5O2Purity:99.91% - 99.91%Color and Shape:SolidMolecular weight:383.495-HT6/5-HT2A receptor ligand-1
CAS:Compound 33 is a dual 5-HT6/5-HT2A antagonist with Ki values of 2 nM and 11 nM, respectively, useful in neuro/psychiatric research.Formula:C21H19FN2O2Color and Shape:SolidMolecular weight:350.39Isamoltane
CAS:Isamoltane is a serotonin 5-HT1 Receptor AntagonistFormula:C16H23ClN2O2Color and Shape:SolidMolecular weight:310.82Blonanserin HCl
CAS:Blonanserin is an antagonist of dopamine-D2 and serotonin-S2.Formula:C23H32Cl2FN3Purity:98%Color and Shape:SolidMolecular weight:440.42EMD 56551
CAS:EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.Formula:C24H31N3O2Purity:95.64% - 99.39%Color and Shape:SolidMolecular weight:393.522Usmarapride
CAS:Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.Formula:C23H31N5O6Color and Shape:SolidMolecular weight:473.53RS 64459-193
CAS:RS 64459-193 has a high affinity for the 5-HT1A binding site.Formula:C26H36Cl2N2O2Color and Shape:SolidMolecular weight:479.48EMDT
CAS:EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.Formula:C15H22N2OPurity:97.66% - 99.78%Color and Shape:SolidMolecular weight:246.35Ref: TM-T11183
1mg87.00€2mg118.00€1mL*10mM (DMSO)166.00€5mg167.00€10mg202.00€25mg449.00€50mg652.00€100mg888.00€500mg1,783.00€Benzoctamine
CAS:Benzoctamine: oral psychoactive with tranquillizing effects; boosts catecholamine turnover; enhances rat heart [3H]noradrenaline uptake.Formula:C18H19NColor and Shape:SolidMolecular weight:249.35SB 714786
CAS:SB 714786 is a selective antagonist of 5-HT1D.Formula:C26H28N4OPurity:98%Color and Shape:SolidMolecular weight:412.53Repinotan HCl
CAS:Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.
Formula:C21H25ClN2O4SPurity:99.57%Color and Shape:SolidMolecular weight:436.95CJ 033466
CAS:CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.Formula:C19H28ClN5OPurity:99.72%Color and Shape:SolidMolecular weight:377.91Trelanserin
CAS:Trelanserin (SL-650472) is an antagonist of the serotonin receptor.Formula:C24H24FN5O2SColor and Shape:SolidMolecular weight:465.54MHP 133
CAS:MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).Formula:C17H20ClN5O3Purity:98%Color and Shape:SolidMolecular weight:377.83Bopindolol
CAS:Bopindolol: oral β1/β2-ARs antagonist and partial agonist; prodrug of pindolol for hypertension research.Formula:C23H28N2O3Color and Shape:SolidMolecular weight:380.48AP521
CAS:AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).Formula:C20H19ClN2O3SPurity:98%Color and Shape:SolidMolecular weight:402.89WAY 163909
CAS:WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).Formula:C14H18N2Purity:98%Color and Shape:SolidMolecular weight:214.31Iloperidone hydrochloride
CAS:Iloperidone hydrochloride is a D(2)/5-HT(2) receptor antagonist. It is also an atypical antipsychotic for the treatment of schizophrenia symptoms.Formula:C24H28ClFN2O4Purity:98%Color and Shape:SolidMolecular weight:462.95Isamoltane hemifumarate
CAS:5-HT1B antagonistFormula:C16H22N202C4H404Purity:98%Color and Shape:SolidMolecular weight:332.4Eplivanserin
CAS:Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.Formula:C19H21FN2O2Purity:97.04%Color and Shape:SolidMolecular weight:328.38UCSF648
CAS:UCSF648 (Compound 5A6-48) weakly activates MTNR1A and ADRA2A. UCSF648 is a chemical probe for the serotonin receptor 5-HT 5A [1].Formula:C15H19ClN2O2SColor and Shape:SolidMolecular weight:326.84SB 258719 hydrochloride
CAS:Selective 5-HT7 receptor antagonistFormula:C18H31ClN2O2SPurity:98%Color and Shape:SolidMolecular weight:374.97Bifeprunox
CAS:Bifeprunox: potent antipsychotic, partial agonist at D2-like/5-HT1A receptors; treats schizophrenia.Formula:C24H23N3O2Purity:98%Color and Shape:SolidMolecular weight:385.46NPS ALX Compound 4a dihydrochloride
CAS:NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Formula:C25H27Cl2N3O2SPurity:98%Color and Shape:SolidMolecular weight:504.47E55888
CAS:E55888 is a potent and selective full agonist of the 5HT7 serotonin receptor.Formula:C16H23N3Color and Shape:SolidMolecular weight:257.37Lintopride
CAS:Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.Formula:C14H19ClN4O2Purity:98%Color and Shape:SolidMolecular weight:310.78(R)-DOI hydrochloride
CAS:(R)-DOI hydrochloride is the salt form of 2,5-Dimethoxy-4-iodoamphetamine (DOI), a potent 5-HT2A and 5-HT2C receptor agonist, orally active and hallucinogenic.Formula:C11H17ClINO2Purity:99.88% - >99.99%Color and Shape:SolidMolecular weight:357.62Enciprazine
CAS:Enciprazine (D-3112) shows anxiolytic activity, is used to treat anxiety disorders, and can be used to study depression.Formula:C23H32N2O6Purity:98.63%Color and Shape:SolidMolecular weight:432.51OPC-14523 free base
CAS:OPC-14523, a 5-HT1A receptor agonist, is used potentially for the treatment of depression and neuropathic pain.Formula:C23H28ClN3O2Purity:98%Color and Shape:SolidMolecular weight:413.94S 14506 hydrochloride
CAS:S 14506 hydrochloride is a 5-HT1A receptor full agonist.Formula:C24H27ClFN3O2Purity:99.92%Color and Shape:SolidMolecular weight:443.94MK-212
CAS:MK-212 is a 5HT2C agonist; boosts corticosterone and lowers activity at 0.5-1mg/kg; reduces anxiety without affecting movement at 0.1-0.2mg/kg in mice.Formula:C8H11ClN4Color and Shape:SolidMolecular weight:198.655-HT7 agonist 1
CAS:5-HT7 agonist 1 (4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-1H-indole) is a selective agonist of 5-HT7 (IC50 = 222.93 nM).Formula:C19H20ClN3Purity:98.61%Color and Shape:SolidMolecular weight:325.84Ref: TM-T10170
1mg109.00€2mg163.00€5mg241.00€1mL*10mM (DMSO)241.00€10mg355.00€25mg532.00€50mg745.00€100mg1,018.00€Ziprasidone mesylate trihydrate
CAS:Ziprasidone mesylate hydrate is an oral 5-HT/D2 antagonist with Ki: D2=4.8nM, 5-HT2A=0.42nM, 5-HT1A=3.4nM in rats.Formula:C22H31ClN4O7S2Color and Shape:SolidMolecular weight:563.08PF-184298
CAS:PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.Formula:C15H20Cl2N2OPurity:98.67%Color and Shape:SolidMolecular weight:315.24PNU-96391
CAS:PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.Formula:C15H23NO2SPurity:99.53%Color and Shape:SolidMolecular weight:281.41Ref: TM-T28435
1mg73.00€1mL*10mM (DMSO)138.00€5mg146.00€10mg210.00€25mg319.00€50mg447.00€100mg600.00€200mg800.00€S 32212 hydrochloride
CAS:S 32212 hydrochloride is a high-affinity inverse agonist at the 5-HT2C receptor and an antagonist at the α2-adrenergic receptor, which is antidepressant .Formula:C25H29ClN4O2Purity:97.11% - 99.57%Color and Shape:SolidMolecular weight:452.98Org-12962 hydrochloride
CAS:Org-12962 hydrochloride is a 5-HT2C receptor agonist.Formula:C10H12Cl2F3N3Purity:98%Color and Shape:SolidMolecular weight:302.12Org-12962
CAS:Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).Formula:C10H11ClF3N3Purity:98.34%Color and Shape:SolidMolecular weight:265.66Zatosetron maleate
CAS:Zatosetron maleate（LY 277359 maleate） is a potent and selective serotonin 5HT3 receptor antagonist for the study of acute migraine.Formula:C23H29ClN2O6Purity:98.07%Color and Shape:SolidMolecular weight:464.94Org-13011 fumarate
CAS:Org-13011 fumarate1 is an agonist of the 5-HT1A receptor and can be used to study neurological disorders.Formula:C22H29F3N4O5Purity:98.92%Color and Shape:SolidMolecular weight:486.48
