5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
Found 940 products of "5-HT Receptor"
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LY 344864 hydrochloride
CAS:<p>LY 344864 hydrochloride is a selective receptor agonist with an affinity of 6 nM (Ki) at the 5-HT1F receptor.</p>Formula:C21H23ClFN3OColor and Shape:SolidMolecular weight:387.88Bifeprunox Mesylate
CAS:<p>Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.</p>Formula:C25H27N3O5SPurity:98%Color and Shape:SolidMolecular weight:481.56AS1069562
CAS:<p>AS1069562 inhibits 5-HT/NE reuptake, boosts IGF-1, FGF2 mRNA in dorsal root ganglia, spinal cord.</p>Formula:C20H23NO5SPurity:98%Color and Shape:SolidMolecular weight:389.46LP 20 hydrochloride
CAS:<p>ligand of the 5-HT7 receptor</p>Formula:C17H21ClN2OPurity:98%Color and Shape:SolidMolecular weight:304.815-HT7 agonist 2
CAS:<p>Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.</p>Formula:C23H29N3OColor and Shape:SolidMolecular weight:363.5CP 135807
CAS:<p>CP 135807 is a 5-HT1D receptor agonist.</p>Formula:C19H21N5O2Purity:98%Color and Shape:SolidMolecular weight:351.4SDZ 21009
CAS:<p>β-adrenoceptor and 5-HT1A/1B receptor antagonist</p>Formula:C19H28N2O4Purity:98%Color and Shape:SolidMolecular weight:348.445-HT6/5-HT2A receptor ligand-2
CAS:<p>Compound 42: brain-penetrant, dual 5-HT6/5-HT2A antagonist, Ki of 25 nM/32 nM, pro-cognitive.</p>Formula:C20H18FN3O2Color and Shape:SolidMolecular weight:351.37SEP-363856
CAS:<p>SEP-363856, a non-D2/5-HT2A, orally active CNS psychotropic may treat schizophrenia.</p>Formula:C9H13NOSPurity:98%Color and Shape:SolidMolecular weight:183.27CGS 12066B dimaleate
CAS:<p>5-HT1B full agonist</p>Formula:C25H25F3N4O8Purity:98%Color and Shape:SolidMolecular weight:566.48Tedatioxetine hydrobromide
CAS:<p>Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.</p>Formula:C18H22BrNSPurity:99.65%Color and Shape:SolidMolecular weight:364.34CP 93129 dihydrochloride
CAS:<p>5-HT1B agonist, potent and highly selective</p>Formula:C12H14ClN3OPurity:98%Color and Shape:SolidMolecular weight:251.71Ro 04-6790 dihydrochloride
CAS:<p>Ro 04-6790 dihydrochloride is an effective and selective antagonist of the serotonin 5-HT6 receptor.</p>Formula:C12H18Cl2N6O2SPurity:98%Color and Shape:SolidMolecular weight:381.28Belaperidone
CAS:<p>Belaperidone, an antipsychotic, resembles clozapine, binds D(4) and 5-HT(2A) receptors, minimally extends Q-T without causing arrhythmias.</p>Formula:C22H22FN3O2Color and Shape:SolidMolecular weight:379.43LY 393558
CAS:<p>Dual 5-HT1B/1D receptor antagonist</p>Formula:C26H31FN4O4S2Purity:98%Color and Shape:SolidMolecular weight:546.68Amitifadine hydrochloride
CAS:<p>Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).</p>Formula:C11H12Cl3NPurity:98%Color and Shape:SolidMolecular weight:264.58Alaproclate
CAS:<p>Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.</p>Formula:C13H18ClNO2Purity:98.29% - 98.64%Color and Shape:SolidMolecular weight:255.74WAY208466 dihydrochloride
CAS:<p>WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.</p>Formula:C17H20Cl2FN3O2SPurity:98.43%Color and Shape:SolidMolecular weight:420.33TC-2153
CAS:<p>TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.</p>Formula:C7H5ClF3NS5Color and Shape:SolidMolecular weight:355.89FR260010
CAS:<p>FR260010 is a novel potent serotonin 5-HT2C receptor antagonist.</p>Formula:C22H19N5Color and Shape:SolidMolecular weight:353.42DAT 582
CAS:<p>DAT 582 is a novel serotonin3 receptor antagonist. It is also an effective and long-lasting antiemetic agent</p>Formula:C22H28ClN5OPurity:98%Color and Shape:SolidMolecular weight:413.95Penbutolol
CAS:<p>Penbutolol is a nonselective beta-blocker utilized as an antihypertensive and an antianginal.</p>Formula:C18H29NO2Purity:98%Color and Shape:SolidMolecular weight:291.435-Nonyloxytryptamine oxalate
CAS:<p>5-HT1B agonist</p>Formula:C21H32N2O5Purity:98%Color and Shape:SolidMolecular weight:392.49PF-04781340
CAS:<p>PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.</p>Formula:C17H21N3Purity:98%Color and Shape:SolidMolecular weight:267.37LP44 hydrochloride
CAS:<p>LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.</p>Formula:C27H38ClN3OSPurity:98.06%Color and Shape:SolidMolecular weight:488.13Bemesetron
CAS:<p>Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.</p>Formula:C15H17Cl2NO2Purity:99.77%Color and Shape:SolidMolecular weight:314.21Zicronapine
CAS:<p>Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.</p>Formula:C22H27ClN2Color and Shape:SolidMolecular weight:354.92SCH-23390 maleate
CAS:<p>SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,</p>Formula:C21H22ClNO5Purity:98%Color and Shape:SolidMolecular weight:403.86Indisetron Dihydrochloride
CAS:<p>Indisetron Dihydrochloride is a 5-HT(3) and 5-HT(4) receptor antagonist. Indisetron reduces 2-methyl-5-serotonin (HT)-induced bradycardia.</p>Formula:C17H24ClN5OColor and Shape:SolidMolecular weight:349.86(RS)-Minesapride
CAS:<p>Minesapride is a serotonin receptor agonist.</p>Formula:C21H31ClN4O5Purity:98%Color and Shape:SolidMolecular weight:454.95LY 206130
CAS:<p>LY 206130 is an antagonist of serotonin 5-HT1A.</p>Formula:C17H24N2O2Color and Shape:SolidMolecular weight:288.38SUN-C5174
CAS:<p>"SUN-C5174 is a selective 5-HT2 antagonist with pA2=8.98; inhibits platelet aggregation and reduces thromboembolic death in mice at ≥0.3 mg/kg."</p>Formula:C22H29FN4O2Purity:98%Color and Shape:SolidMolecular weight:400.49Deramciclane
CAS:<p>Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.</p>Formula:C20H31NOColor and Shape:SolidMolecular weight:301.47RGH 1756
CAS:<p>RGH 1756 is an atypical antipsychotic with high affinity to dopamine D(3) receptors that leads to c-Fos induction in a unique pattern.</p>Formula:C26H30N4O2SPurity:98%Color and Shape:SolidMolecular weight:462.61WAY 161503 hydrochloride
CAS:<p>WAY 161503 hydrochloride is a 5-HT2C receptor agonist.</p>Formula:C11H12Cl3N3OPurity:98%Color and Shape:SolidMolecular weight:308.59Altanserin hydrochloride
CAS:<p>Altanserin hydrochloride is a 5-HT2A receptor antagonist.</p>Formula:C22H23ClFN3O2SPurity:98%Color and Shape:SolidMolecular weight:447.95SB 258585 hydrochloride
CAS:<p>SB 258585 hydrochloride is a 5-HT6 receptor antagonist.</p>Formula:C18H23ClIN3O3SPurity:98%Color and Shape:SolidMolecular weight:523.82EMD 56551
CAS:<p>EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.</p>Formula:C24H31N3O2Purity:95.64% - 99.39%Color and Shape:SolidMolecular weight:393.522(Rac)-SEP-363856
CAS:<p>(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a unique</p>Formula:C9H13NOSPurity:98%Color and Shape:SolidMolecular weight:183.27SGS518 oxalate
CAS:<p>SGS518 oxalate is a 5-HT6 antagonist.</p>Formula:C23H24F2N2O7SPurity:98%Color and Shape:SolidMolecular weight:510.51Opiranserin
CAS:<p>Opiranserin is a development as an injectable agent for the treatment of postoperative pain.</p>Formula:C21H34N2O5Purity:98%Color and Shape:SolidMolecular weight:394.51Palonosetron
CAS:<p>Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).</p>Formula:C19H24N2OPurity:98%Color and Shape:SolidMolecular weight:296.41LY 334370 hydrochloride
CAS:<p>5-HT1F receptor agonist</p>Formula:C21H23ClFN3OPurity:98%Color and Shape:SolidMolecular weight:387.88ML 10375
CAS:<p>ML 10375 is an antagonist of 5-HT4 receptor.</p>Formula:C17H25ClN2O3Color and Shape:SolidMolecular weight:340.85YM 114
CAS:<p>YM 114 is an anatagonist of 5-HT(3) receptor.</p>Formula:C16H18ClN3OPurity:98%Color and Shape:SolidMolecular weight:303.79LY314228
CAS:<p>LY314228 is an antagonist of 5-HT2A receptor.</p>Formula:C20H24N4O3Color and Shape:SolidMolecular weight:368.43ATC0065 HCl
CAS:<p>ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.</p>Formula:C25H31BrCl2F3N5OColor and Shape:SolidMolecular weight:625.35GR-55562 dihydrobromide
CAS:<p>GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.</p>Formula:C23H26ClN3O2Purity:98%Color and Shape:SolidMolecular weight:411.93Pancopride
CAS:<p>Pancopride（LAS 30451） is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen mustard and dacarbazine-induced</p>Formula:C18H24ClN3O2Purity:93.64%Color and Shape:SolidMolecular weight:349.86Tacitin
CAS:<p>Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.</p>Formula:C18H20ClNPurity:98%Color and Shape:SolidMolecular weight:285.81
