5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
Found 1025 products of "5-HT Receptor"
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AVN-322
CAS:AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.Formula:C17H20ClN5O2SPurity:>99.99%Color and Shape:SolidMolecular weight:393.89MS 245 oxalate
CAS:MS 245 oxalate is a 5-HT6 antagonist.Formula:C21H24N2O7SPurity:98%Color and Shape:SolidMolecular weight:448.49LY 334370 hydrochloride
CAS:5-HT1F receptor agonistFormula:C21H23ClFN3OPurity:98%Color and Shape:SolidMolecular weight:387.88Methiothepin maleate
CAS:Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.Formula:C24H28N2O4S2Purity:98%Color and Shape:SolidMolecular weight:472.62Irindalone
CAS:IrindaloneIrindalone is a potent serotonin (5-HT2) antagonist.Formula:C24H29FN4OPurity:98%Color and Shape:SolidMolecular weight:408.51EGIS-7625
CAS:EGIS-7625 is a selective and competitive antagonist of 5-HT2B receptor.Formula:C18H24Cl2N4O2Purity:98%Color and Shape:SolidMolecular weight:399.32Glemanserin
CAS:Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.Formula:C20H25NOPurity:99.93%Color and Shape:SolidMolecular weight:295.42Ref: TM-T22964
1mg38.00€5mg84.00€1mL*10mM (DMSO)84.00€10mg119.00€25mg259.00€50mg409.00€100mg605.00€500mg1,288.00€DV 7028 hydrochloride
CAS:DV 7028 hydrochloride is a 5-HT2A receptor antagonist.Formula:C21H26ClFN4O3Purity:98%Color and Shape:SolidMolecular weight:436.91Org37684
CAS:5-HT2 receptors agonistFormula:C14H20ClNO2Purity:98%Color and Shape:SolidMolecular weight:269.77L-775,606
CAS:L-775,606 is a selective agonist of 5-hydroxytryptamine 1D.Formula:C25H29FN6Purity:98%Color and Shape:SolidMolecular weight:432.54AR-A 2
CAS:AR-A 2, a selective 5-HT1B antagonist; high guinea pig 5-HT1B/1D affinity (Ki: 0.24, 0.47 nM); 10x less for 5-HT1D (Ki: 5 nM).Formula:C27H36N4O2Purity:98%Color and Shape:SolidMolecular weight:448.6PNU-282987 S enantiomer hydrochloride
CAS:(S)-PNU-282987, selective α7 nAChR agonist; Ki=26 nM (rat), weak on other receptors except 5-HT3; Ki=930 nM.Formula:C14H18Cl2N2OPurity:98%Color and Shape:SolidMolecular weight:301.21Donitriptan
CAS:Donitriptan 是一种 5-HT 受体激动剂，对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。
Formula:C23H25N5O2Purity:98.76%Color and Shape:SolidMolecular weight:403.48Quinupramine
CAS:Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.Formula:C21H24N2Purity:99.77%Color and Shape:SolidMolecular weight:304.43PNU-282987 free base
CAS:PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.
Formula:C14H17ClN2OPurity:99.64%Color and Shape:SolidMolecular weight:264.75Masupirdine free base
CAS:Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.Formula:C21H24BrN3O3SPurity:98.36% - 99.65%Color and Shape:SolidMolecular weight:478.4(Z)-Thiothixene
CAS:(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.
Formula:C23H29N3O2S2Purity:99.21%Color and Shape:Yellow To Yellow With A Tan Cast PowderMolecular weight:443.63Teniloxazine
CAS:Teniloxazine is an orally available antidepressant compound with anti-hypoxic properties.Formula:C16H19NO2SPurity:99.29%Color and Shape:SolidMolecular weight:289.39R 59-022 hydrochloride
CAS:R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.
Formula:C27H27ClFN3OSPurity:97.7%Color and Shape:SolidMolecular weight:496.04RS 42358-197
CAS:RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.Formula:C19H23ClN2OPurity:99.70%Color and Shape:SolidMolecular weight:330.85Ref: TM-T20739
1mg158.00€1mL*10mM (DMSO)349.00€5mg351.00€10mg527.00€25mg783.00€50mg1,054.00€100mg1,414.00€200mg1,908.00€Lecozotan HCl
CAS:Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.
Formula:C28H30ClN5O3Purity:99.04%Color and Shape:SolidMolecular weight:520.02DA-6886
CAS:DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.Formula:C19H28Cl2N6O2Purity:99.91% - 99.99%Color and Shape:SolidMolecular weight:443.37Adoprazine
CAS:Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.Formula:C24H24FN3O2Purity:99.83%Color and Shape:SolidMolecular weight:405.46Ref: TM-T10249
1mg60.00€5mg130.00€1mL*10mM (DMSO)142.00€10mg205.00€25mg363.00€50mg580.00€100mg782.00€Femoxetine hydrochloride
CAS:Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.Formula:C20H26ClNO2Purity:99.63%Color and Shape:SolidMolecular weight:347.88Goxalapladib
CAS:Goxalapladib（GSK 677116） is a small molecule compound that can be used to treat cardiovascular risks associated with atherosclerosis.Formula:C40H39F5N4O3Purity:99.64% - 99.93%Color and Shape:SolidMolecular weight:718.75Cyamemazine
CAS:Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.Formula:C19H21N3SPurity:97.01%Color and Shape:SolidMolecular weight:323.46Tedatioxetine
CAS:Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.Formula:C18H21NSPurity:99.76% - >99.99%Color and Shape:SolidMolecular weight:283.43Landipirdine
CAS:Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.Formula:C18H19FN2O3SPurity:97.61% - 99.99%Color and Shape:SolidMolecular weight:362.42Faxeladol
CAS:Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.Formula:C15H23NOPurity:98.77% - 99.67%Color and Shape:SolidMolecular weight:233.35Cianopramine
CAS:Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.Formula:C20H23N3Purity:99.92% - 99.92%Color and Shape:SolidMolecular weight:305.42BL-1020 Mesylate
CAS:BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.Formula:C28H45ClN4O11S4Purity:>99.99%Color and Shape:SolidMolecular weight:777.39Viloxazine
CAS:Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activityFormula:C13H19NO3Purity:99.65%Color and Shape:SolidMolecular weight:237.29CP 96021
CAS:"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."
Formula:C29H21FN4OSPurity:97.81% - 99.62%Color and Shape:SoildMolecular weight:492.57Cilansetron
CAS:Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.Formula:C20H21N3OPurity:99.82% - 99.98%Color and Shape:SolidMolecular weight:319.4E6801
CAS:E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.Formula:C17H18ClN5O2S2Purity:96.32% - 97.24%Color and Shape:SolidMolecular weight:423.94Ticalopride
CAS:Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.Formula:C14H20ClN3O3Purity:99.51%Color and Shape:SolidMolecular weight:313.78SPD-473 citrate
CAS:SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.Formula:C23H31Cl2NO8SPurity:99.37%Color and Shape:SolidMolecular weight:552.47Roxindole
CAS:Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.Formula:C23H26N2OPurity:98.03% - 98.93%Color and Shape:SolidMolecular weight:346.47Aplindore Fumarate
CAS:Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.Formula:C22H22N2O7Purity:99.66%Color and Shape:SolidMolecular weight:426.42Nexopamil
CAS:Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.
Formula:C24H40N2O3Purity:97.87% - >99.99%Color and Shape:SolidMolecular weight:404.59ATC 0175
CAS:ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.Formula:C23H26ClF2N5OPurity:99.98%Color and Shape:SolidMolecular weight:461.93Perphenazine dihydrochloride
CAS:Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.Formula:C21H28Cl3N3OSPurity:99.67%Color and Shape:SolidMolecular weight:476.89Liafensine
CAS:Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.Formula:C24H22N4Purity:99.91%Color and Shape:SolidMolecular weight:366.46Piromelatine
CAS:Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity withFormula:C17H16N2O4Purity:99.83%Color and Shape:SolidMolecular weight:312.32Ref: TM-T34081
1mg60.00€5mg130.00€1mL*10mM (DMSO)142.00€10mg178.00€25mg334.00€50mg522.00€100mg713.00€Lensiprazine
CAS:Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder andFormula:C24H27FN4O2Purity:97.86%Color and Shape:SolidMolecular weight:422.5H-9 dihydrochloride
CAS:H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.Formula:C11H15Cl2N3O2SPurity:97.3%Color and Shape:SolidMolecular weight:324.235-HT6/7 antagonist 1
CAS:5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.Formula:C22H20FN3O3Purity:98.78% - 99.26%Color and Shape:SolidMolecular weight:393.41Litoxetine
CAS:Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.Formula:C16H19NOPurity:99.68%Color and Shape:SolidMolecular weight:241.33Ref: TM-T67956
1mg92.00€1mL*10mM (DMSO)178.00€5mg207.00€10mg309.00€25mg527.00€50mg755.00€100mg1,044.00€500mg2,088.00€BMY-14802 hydrochloride
CAS:BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.Formula:C18H23ClF2N4OPurity:99.97%Color and Shape:SolidMolecular weight:384.85Tiospirone
CAS:Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.Formula:C24H32N4O2SPurity:99.74%Color and Shape:SolidMolecular weight:440.6Ref: TM-T24885
1mg123.00€5mg293.00€1mL*10mM (DMSO)354.00€10mg537.00€25mg863.00€50mg1,161.00€100mg1,558.00€
