5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
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LY266097 hydrochloride
CAS:172895-39-5
LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression …
Formula:
C21H24Cl2N2O2
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
407.33
Ref: TM-T22947
| 5mg | 50.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 107.00 € | ||
| 50mg | 159.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Rilapine
CAS:79781-95-6
Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can …
Formula:
C22H20ClN3
Purity:
99% - 99.66%
Color and Shape:
Solid
Molecular weight:
361.87
Ref: TM-T26085
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Anpirtoline hydrochloride
CAS:99201-87-3
Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in …
Formula:
C10H14Cl2N2S
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
265.20
Ref: TM-T22576
| 1mg | 52.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 421.00 € | ||
| 100mg | 606.00 € | ||
| 500mg | 1,253.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
PNU-282987 free base
CAS:711085-63-1
PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for …
Formula:
C14H17ClN2O
Purity:
99.64%
Color and Shape:
Liquid
Molecular weight:
264.75
Ref: TM-T60437
| 1mg | 55.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 201.00 € | ||
| 25mg | 392.00 € | ||
| 50mg | 727.00 € | ||
| 100mg | 1,020.00 € | ||
| 500mg | 2,039.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
5-HT3 antagonist 3
CAS:120635-47-4
5-HT3 antagonist 3 (Compound 15b) is a high-affinity 5-HT3 receptor antagonist. It binds to 5-HT3 …
Formula:
C20H21N3O
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
319.4
Ref: TM-T10162
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 775.00 € | ||
| 100mg | 1,040.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 31 Mar 2025
R 59-022 hydrochloride
CAS:93076-98-3
R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and …
Formula:
C27H27ClFN3OS
Purity:
97.7%
Color and Shape:
Liquid
Molecular weight:
496.04
Ref: TM-T72322
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 447.00 € | ||
| 100mg | 643.00 € | ||
| 500mg | 1,319.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Ricasetron
CAS:117086-68-7
Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used …
Formula:
C19H27N3O
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
313.44
Ref: TM-T28537
| 1mg | 214.00 € | ||
| 5mg | 543.00 € | ||
| 10mg | 771.00 € | ||
| 25mg | 1,199.00 € | ||
| 50mg | 1,621.00 € | ||
| 100mg | 2,183.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
DA-6886
CAS:1645260-76-9
DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: …
Formula:
C19H28Cl2N6O2
Purity:
99% - 99.89%
Color and Shape:
Solid
Molecular weight:
443.37
Ref: TM-T27117
| 1mg | 136.00 € | ||
| 5mg | 316.00 € | ||
| 10mg | 474.00 € | ||
| 25mg | 772.00 € | ||
| 50mg | 1,068.00 € | ||
| 100mg | 1,448.00 € | ||
| 500mg | 2,775.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Femoxetine hydrochloride
CAS:56222-04-9
Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression …
Formula:
C20H26ClNO2
Purity:
99.48%
Color and Shape:
Liquid
Molecular weight:
347.88
Ref: TM-T69096
| 1mg | 195.00 € | ||
| 5mg | 493.00 € | ||
| 10mg | 714.00 € | ||
| 25mg | 1,100.00 € | ||
| 50mg | 1,483.00 € | ||
| 100mg | 2,004.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Cyamemazine
CAS:3546-03-0
Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and …
Formula:
C19H21N3S
Purity:
97.01%
Color and Shape:
Solid
Molecular weight:
323.46
Ref: TM-T15026
| 1mg | 36.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 103.00 € | ||
| 25mg | 208.00 € | ||
| 50mg | 353.00 € | ||
| 100mg | 603.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Faxeladol
CAS:433265-65-7
Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.
Formula:
C15H23NO
Purity:
99.11% - 99.13%
Color and Shape:
Solid
Molecular weight:
233.35
Ref: TM-T31750
| 1mg | 597.00 € | ||
| 5mg | 1,258.00 € | ||
| 25mg | 1,692.00 € | ||
| 50mg | 2,023.00 € | ||
| 100mg | 2,610.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Cinitapride Hydrogen Tartrate
CAS:1207859-16-2
Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 …
Formula:
C25H36N4O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
552.581
Ref: TM-T22294
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Palonosetron
CAS:135729-61-2
Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and …
Formula:
C19H24N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
296.41
Ref: TM-T22393
| 25mg | 1,406.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Landipirdine
CAS:1000308-25-7
Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders …
Formula:
C18H19FN2O3S
Purity:
97.50% - 99.33%
Color and Shape:
Solid
Molecular weight:
362.42
Ref: TM-T27795
| 1mg | 227.00 € | ||
| 5mg | 541.00 € | ||
| 10mg | 726.00 € | ||
| 25mg | 1,172.00 € | ||
| 50mg | 1,493.00 € | ||
| 100mg | 2,124.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
p-MPPF dihydrochloride
CAS:223699-41-0
p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.
Formula:
C25H29Cl2FN4O2
Purity:
99.78%
Color and Shape:
Liquid
Molecular weight:
507.43
Ref: TM-T69750
| 1mg | 266.00 € | ||
| 5mg | 655.00 € | ||
| 10mg | 896.00 € | ||
| 25mg | 1,437.00 € | ||
| 50mg | 1,872.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Repinotan HCl
CAS:144980-77-8
Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study …
Formula:
C21H25ClN2O4S
Purity:
99.57%
Color and Shape:
Solid
Molecular weight:
436.95
Ref: TM-T28518
| 1mg | 380.00 € | ||
| 5mg | 820.00 € | ||
| 10mg | 1,168.00 € | ||
| 25mg | 1,564.00 € | ||
| 50mg | 1,899.00 € | ||
| 100mg | 2,396.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
RS 42358-197
CAS:135729-55-4
RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.
Formula:
C19H23ClN2O
Purity:
98.23%
Color and Shape:
Solid
Molecular weight:
330.85
Ref: TM-T20739
| 1mg | 162.00 € | ||
| 5mg | 362.00 € | ||
| 10mg | 542.00 € | ||
| 25mg | 804.00 € | ||
| 50mg | 1,081.00 € | ||
| 100mg | 1,450.00 € | ||
| 200mg | 1,958.00 € | ||
| 1mL*10mM (DMSO) | 359.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
AS19
CAS:1000578-26-6
AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM).
Formula:
C18H25N3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
283.41
Ref: TM-T10380
| 25mg | 1,549.00 € | ||
| 50mg | 2,031.00 € | ||
| 100mg | 2,609.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
5-HT4 antagonist 1
CAS:261766-73-8
5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).
Formula:
C23H36N4O5S
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
480.62
Ref: TM-T10169
| 1mg | 63.00 € | ||
| 5mg | 143.00 € | ||
| 10mg | 207.00 € | ||
| 25mg | 350.00 € | ||
| 50mg | 499.00 € | ||
| 100mg | 680.00 € | ||
| 500mg | 1,365.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
L-694,247
CAS:137403-12-4
L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E …
Formula:
C20H21N5O3S
Purity:
98.36%
Color and Shape:
White Solid
Molecular weight:
411.48
Ref: TM-T19701
| 1mg | 83.00 € | ||
| 5mg | 264.00 € | ||
| 10mg | 451.00 € | ||
| 25mg | 722.00 € | ||
| 50mg | 1,010.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
